Progress in the development of human carbonic anhydrase inhibitors and their pharmacological applications: Where are we today?
出版年份 2020 全文链接
标题
Progress in the development of human carbonic anhydrase inhibitors and their pharmacological applications: Where are we today?
作者
关键词
-
出版物
MEDICINAL RESEARCH REVIEWS
Volume -, Issue -, Pages -
出版商
Wiley
发表日期
2020-07-21
DOI
10.1002/med.21713
参考文献
相关参考文献
注意：仅列出部分参考文献，下载原文获取全部文献信息。- Perfluoroalkyl Substances of Significant Environmental Concern Can Strongly Inhibit Human Carbonic Anhydrase Isozymes
- (2020) Giang T. H. Nguyen et al. ANALYTICAL CHEMISTRY
- 1,3-Dipolar Cycloaddition, HPLC Enantioseparation, and Docking Studies of Saccharin/Isoxazole and Saccharin/Isoxazoline Derivatives as Selective Carbonic Anhydrase IX and XII Inhibitors
- (2020) Melissa D’Ascenzio et al. JOURNAL OF MEDICINAL CHEMISTRY
- Heterocyclic periphery in the design of carbonic anhydrase inhibitors: 1,2,4-Oxadiazol-5-yl benzenesulfonamides as potent and selective inhibitors of cytosolic h CA II and membrane-bound h CA IX isoforms
- (2018) Mikhail Krasavin et al. BIOORGANIC CHEMISTRY
- Unprotected primary sulfonamide group facilitates ring-forming cascade en route to polycyclic [1,4]oxazepine-based carbonic anhydrase inhibitors
- (2018) Alexander Sapegin et al. BIOORGANIC CHEMISTRY
- Synthesis and biological evaluation of novel pyrazoline-based aromatic sulfamates with potent carbonic anhydrase isoforms II, IV and IX inhibitory efficacy
- (2018) Alessio Nocentini et al. BIOORGANIC CHEMISTRY
- Synthesis and biological evaluation of novel N , N ′-diaryl cyanoguanidines acting as potent and selective carbonic anhydrase II inhibitors
- (2018) Suleyman Akocak et al. BIOORGANIC CHEMISTRY
- Synthesis, biological evaluation and computational studies of novel iminothiazolidinone benzenesulfonamides as potent carbonic anhydrase II and IX inhibitors
- (2018) Shams-ul Mahmood et al. BIOORGANIC CHEMISTRY
- Design and synthesis of novel 1,3-diaryltriazene-substituted sulfonamides as potent and selective carbonic anhydrase II inhibitors
- (2018) Nabih Lolak et al. BIOORGANIC CHEMISTRY
- Synthesis of N ′-phenyl- N -hydroxyureas and investigation of their inhibitory activities on human carbonic anhydrases
- (2018) Murat Bozdag et al. BIOORGANIC CHEMISTRY
- Synthesis and Biological Evaluation of 4-Sulfamoylphenyl/Sulfocoumarin Carboxamides as Selective Inhibitors of Carbonic Anhydrase Isoforms hCA II, IX, and XII
- (2018) Srinivas Angapelly et al. ChemMedChem
- Inhibitory effects and structural insights for a novel series of coumarin-based compounds that selectively target human CA IX and CA XII carbonic anhydrases
- (2018) Laura De Luca et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Dual-tail arylsulfone-based benzenesulfonamides differently match the hydrophobic and hydrophilic halves of human carbonic anhydrases active sites: Selective inhibitors for the tumor-associated hCA IX isoform
- (2018) Hany S. Ibrahim et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- 2-Benzylpiperazine: A new scaffold for potent human carbonic anhydrase inhibitors. Synthesis, enzyme inhibition, enantioselectivity, computational and crystallographic studies and in vivo activity for a new class of intraocular pressure lowering agents
- (2018) Niccolò Chiaramonte et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Synthesis of novel 4-functionalized 1,5-diaryl-1,2,3-triazoles containing benzenesulfonamide moiety as carbonic anhydrase I, II, IV and IX inhibitors
- (2018) Lalit Vats et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Discovery of potent anti-convulsant carbonic anhydrase inhibitors: Design, synthesis, in vitro and in vivo appraisal
- (2018) Chandra Bhushan Mishra et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Structural investigations on coumarins leading to chromeno[4,3-c]pyrazol-4-ones and pyrano[4,3-c]pyrazol-4-ones: New scaffolds for the design of the tumor-associated carbonic anhydrase isoforms IX and XII
- (2018) Alessandro Bonardi et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Novel 2-(2-arylmethylthio-4-chloro-5-methylbenzenesulfonyl)-1-(1,3,5-triazin-2-ylamino)guanidine derivatives: Inhibition of human carbonic anhydrase cytosolic isozymes I and II and the transmembrane tumor-associated isozymes IX and XII, anticancer activity, and molecular modeling studies
- (2018) Beata Żołnowska et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Acetazolamide Reduces Blood Pressure and Sleep-Disordered Breathing in Patients With Hypertension and Obstructive Sleep Apnea: A Randomized Controlled Trial
- (2018) Davoud Eskandari et al. Journal of Clinical Sleep Medicine
- Inhibition studies on a panel of human carbonic anhydrases with N1-substituted secondary sulfonamides incorporating thiazolinone or imidazolone-indole tails
- (2018) Fadi M. Awadallah et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- Selective inhibition of carbonic anhydrase-IX by sulphonamide derivatives induces pH and reactive oxygen species-mediated apoptosis in cervical cancer HeLa cells
- (2018) Ismail Koyuncu et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- Discovery of Benzenesulfonamide Derivatives as Carbonic Anhydrase Inhibitors with Effective Anticonvulsant Action: Design, Synthesis, and Pharmacological Evaluation
- (2018) Chandra Bhushan Mishra et al. JOURNAL OF MEDICINAL CHEMISTRY
- Discovery of Novel Nonsteroidal Anti-Inflammatory Drugs and Carbonic Anhydrase Inhibitors Hybrids (NSAIDs–CAIs) for the Management of Rheumatoid Arthritis
- (2018) Ozlem Akgul et al. JOURNAL OF MEDICINAL CHEMISTRY
- Discovery of β-Adrenergic Receptors Blocker–Carbonic Anhydrase Inhibitor Hybrids for Multitargeted Antiglaucoma Therapy
- (2018) Alessio Nocentini et al. JOURNAL OF MEDICINAL CHEMISTRY
- 4-Substituted Benzenesulfonamides Incorporating Bi/Tricyclic Moieties Act as Potent and Isoform-Selective Carbonic Anhydrase II/IX Inhibitors
- (2018) Silvia Salerno et al. JOURNAL OF MEDICINAL CHEMISTRY
- Discovery of 4-Hydroxy-3-(3-(phenylureido)benzenesulfonamides as SLC-0111 Analogues for the Treatment of Hypoxic Tumors Overexpressing Carbonic Anhydrase IX
- (2018) Murat Bozdag et al. JOURNAL OF MEDICINAL CHEMISTRY
- Inhibition of carbonic anhydrase IX targets primary tumors, metastases, and cancer stem cells: Three for the price of one
- (2018) Claudiu T. Supuran et al. MEDICINAL RESEARCH REVIEWS
- Novel 6- and 7-Substituted Coumarins with Inhibitory Action against Lipoxygenase and Tumor-Associated Carbonic Anhydrase IX
- (2018) Aikaterini Peperidou et al. MOLECULES
- Cancer Drug Development of Carbonic Anhydrase Inhibitors beyond the Active Site
- (2018) Srishti Singh et al. MOLECULES
- Design, Synthesis, and X-ray of Selenides as New Class of Agents for Prevention of Diabetic Cerebrovascular Pathology
- (2018) Andrea Angeli et al. ACS Medicinal Chemistry Letters
- Targeting Tumor Associated Carbonic Anhydrases IX and XII: Highly Isozyme Selective Coumarin and Psoralen Inhibitors
- (2018) Claudia Melis et al. ACS Medicinal Chemistry Letters
- pH regulators to target the tumor immune microenvironment in human hepatocellular carcinoma
- (2018) Olga Kuchuk et al. OncoImmunology
- Carbonic anhydrase inhibitors as antitumor/antimetastatic agents: a patent review (2008–2018)
- (2018) Alessio Nocentini et al. EXPERT OPINION ON THERAPEUTIC PATENTS
- Applications of carbonic anhydrases inhibitors in renal and central nervous system diseases
- (2018) Claudiu T. Supuran EXPERT OPINION ON THERAPEUTIC PATENTS
- Carbonic anhydrase inhibitors as emerging agents for the treatment and imaging of hypoxic tumors
- (2018) Claudiu T. Supuran EXPERT OPINION ON INVESTIGATIONAL DRUGS
- Discovery of curcumin inspired sulfonamide derivatives as a new class of carbonic anhydrase isoforms I, II, IX, and XII inhibitors
- (2017) P. V. Sri Ramya et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- Synthesis, biological activity and multiscale molecular modeling studies for coumaryl-carboxamide derivatives as selective carbonic anhydrase IX inhibitors
- (2017) Belma Zengin Kurt et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- Carbonic anhydrase inhibitory properties of some uracil derivatives
- (2017) Emir Alper Türkoğlu et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- Synthesis of an acridine orange sulfonamide derivative with potent carbonic anhydrase IX inhibitory action
- (2017) Marco Bragagni et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- Design and Synthesis of Novel Nonsteroidal Anti-Inflammatory Drugs and Carbonic Anhydrase Inhibitors Hybrids (NSAIDs–CAIs) for the Treatment of Rheumatoid Arthritis
- (2017) Silvia Bua et al. JOURNAL OF MEDICINAL CHEMISTRY
- Discovery of Benzenesulfonamides with Potent Human Carbonic Anhydrase Inhibitory and Effective Anticonvulsant Action: Design, Synthesis, and Pharmacological Assessment
- (2017) Chandra Bhushan Mishra et al. JOURNAL OF MEDICINAL CHEMISTRY
- Lead Development of Thiazolylsulfonamides with Carbonic Anhydrase Inhibitory Action
- (2017) Fabrizio Carta et al. JOURNAL OF MEDICINAL CHEMISTRY
- 3-Hydroxy-1H-quinazoline-2,4-dione as a New Scaffold To Develop Potent and Selective Inhibitors of the Tumor-Associated Carbonic Anhydrases IX and XII
- (2017) Matteo Falsini et al. JOURNAL OF MEDICINAL CHEMISTRY
- Probing Molecular Interactions between Human Carbonic Anhydrases (hCAs) and a Novel Class of Benzenesulfonamides
- (2017) Elvira Bruno et al. JOURNAL OF MEDICINAL CHEMISTRY
- Novel Sulfamide-Containing Compounds as Selective Carbonic Anhydrase I Inhibitors
- (2017) Emanuela Berrino et al. MOLECULES
- Design and Comparative Evaluation of the Anticonvulsant Profile, Carbonic-Anhydrate Inhibition and Teratogenicity of Novel Carbamate Derivatives of Branched Aliphatic Carboxylic Acids with 4-Aminobenzensulfonamide
- (2017) David Bibi et al. NEUROCHEMICAL RESEARCH
- Lucky Switcheroo: Dramatic Potency and Selectivity Improvement of Imidazoline Inhibitors of Human Carbonic Anhydrase VII
- (2017) Stanislav Kalinin et al. ACS Medicinal Chemistry Letters
- Synthesis of Novel Selenides Bearing Benzenesulfonamide Moieties as Carbonic Anhydrase I, II, IV, VII, and IX Inhibitors
- (2017) Andrea Angeli et al. ACS Medicinal Chemistry Letters
- Discovery of New Sulfonamide Carbonic Anhydrase IX Inhibitors Incorporating Nitrogenous Bases
- (2017) Alessio Nocentini et al. ACS Medicinal Chemistry Letters
- Sulfamide derivatives with selective carbonic anhydrase VII inhibitory action
- (2016) Maria Luisa Villalba et al. BIOORGANIC & MEDICINAL CHEMISTRY
- A novel library of saccharin and acesulfame derivatives as potent and selective inhibitors of carbonic anhydrase IX and XII isoforms
- (2016) Simone Carradori et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Development of 3-(4-aminosulphonyl)-phenyl-2-mercapto-3H-quinazolin-4-ones as inhibitors of carbonic anhydrase isoforms involved in tumorigenesis and glaucoma
- (2016) Ahmed M. Alafeefy et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Microwave assisted synthesis of novel acridine–acetazolamide conjugates and investigation of their inhibition effects on human carbonic anhydrase isoforms hCA I, II, IV and VII
- (2016) Ramazan Ulus et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Synthesis of 4-(thiazol-2-ylamino)-benzenesulfonamides with carbonic anhydrase I, II and IX inhibitory activity and cytotoxic effects against breast cancer cell lines
- (2016) Nagwa M. Abdel Gawad et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Synthesis of 4-sulfamoylphenyl-benzylamine derivatives with inhibitory activity against human carbonic anhydrase isoforms I, II, IX and XII
- (2016) Mustafa Durgun et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Inhibition of carbonic anhydrase isoforms I, II, IV, VII and XII with carboxylates and sulfonamides incorporating phthalimide/phthalic anhydride scaffolds
- (2016) Adel S. El-Azab et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Synthesis and carbonic anhydrase inhibitory effects of new N-glycosylsulfonamides incorporating the phenol moiety
- (2016) Leonardo E. Riafrecha et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Synthesis and carbonic anhydrase inhibitory properties of novel chalcone substituted benzenesulfonamides
- (2016) Tayfun Arslan et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Carbonic anhydrase inhibitors reduce cardiac dysfunction after sustained coronary artery ligation in rats
- (2016) Lorena A. Vargas et al. CARDIOVASCULAR PATHOLOGY
- The Emerging Hallmarks of Cancer Metabolism
- (2016) Natalya N. Pavlova et al. Cell Metabolism
- Polypharmacological Drugs in the Treatment of Epilepsy: The Comprehensive Review of Marketed and New Emerging Molecules
- (2016) Shikha Kumari et al. CURRENT PHARMACEUTICAL DESIGN
- Advances in structure-based drug discovery of carbonic anhydrase inhibitors
- (2016) Claudiu T. Supuran Expert Opinion on Drug Discovery
- Overexpression of the transmembrane carbonic anhydrase isoforms IX and XII in the inflamed synovium
- (2016) Francesca Margheri et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- Design, synthesis and biological evaluation of N-(5-methyl-isoxazol-3-yl/1,3,4-thiadiazol-2-yl)-4-(3-substitutedphenylureido) benzenesulfonamides as human carbonic anhydrase isoenzymes I, II, VII and XII inhibitors
- (2016) Chandra Bhushan Mishra et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- Open saccharin-based secondary sulfonamides as potent and selective inhibitors of cancer-related carbonic anhydrase IX and XII isoforms
- (2016) Melissa D’Ascenzio et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- 4-Arylbenzenesulfonamides as Human Carbonic Anhydrase Inhibitors (hCAIs): Synthesis by Pd Nanocatalyst-Mediated Suzuki–Miyaura Reaction, Enzyme Inhibition, and X-ray Crystallographic Studies
- (2016) Benedetta Cornelio et al. JOURNAL OF MEDICINAL CHEMISTRY
- Monothiocarbamates Strongly Inhibit Carbonic Anhydrases in Vitro and Possess Intraocular Pressure Lowering Activity in an Animal Model of Glaucoma
- (2016) Daniela Vullo et al. JOURNAL OF MEDICINAL CHEMISTRY
- PEGylated Bis-Sulfonamide Carbonic Anhydrase Inhibitors Can Efficiently Control the Growth of Several Carbonic Anhydrase IX-Expressing Carcinomas
- (2016) Suleyman Akocak et al. JOURNAL OF MEDICINAL CHEMISTRY
- 1,2-Benzisothiazole Derivatives Bearing 4-, 5-, or 6-Alkyl/arylcarboxamide Moieties Inhibit Carbonic Anhydrase Isoform IX (CAIX) and Cell Proliferation under Hypoxic Conditions
- (2016) Vito Coviello et al. JOURNAL OF MEDICINAL CHEMISTRY
- Central Neuropathic Pain Syndromes
- (2016) James C. Watson et al. MAYO CLINIC PROCEEDINGS
- Core Management Principles in Rheumatoid Arthritis to Help Guide Managed Care Professionals
- (2016) Sandeep K. Agarwal JOURNAL OF MANAGED CARE PHARMACY
- New natural product carbonic anhydrase inhibitors incorporating phenol moieties
- (2015) Anastasia Karioti et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Cyclodextrin complexation highly enhances efficacy of arylsulfonylureido benzenesulfonamide carbonic anhydrase inhibitors as a topical antiglaucoma agents
- (2015) Marco Bragagni et al. BIOORGANIC & MEDICINAL CHEMISTRY
- New approaches to the synthesis of sildenafil analogues and their enzyme inhibitory activity
- (2015) Mariusz Mojzych et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Synthesis of a new series of dithiocarbamates with effective human carbonic anhydrase inhibitory activity and antiglaucoma action
- (2015) Murat Bozdag et al. BIOORGANIC & MEDICINAL CHEMISTRY
- New pyrazolo[4,3- e ][1,2,4]triazine sulfonamides as carbonic anhydrase inhibitors
- (2015) Mariusz Mojzych et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Click-tailed coumarins with potent and selective inhibitory action against the tumor-associated carbonic anhydrases IX and XII
- (2015) Alessio Nocentini et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Synthesis of 6-aryl-substituted sulfocoumarins and investigation of their carbonic anhydrase inhibitory action
- (2015) Aiga Grandane et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Benzenesulfonamides incorporating bulky aromatic/heterocyclic tails with potent carbonic anhydrase inhibitory activity
- (2015) Murat Bozdag et al. BIOORGANIC & MEDICINAL CHEMISTRY
- A class of sulfonamide carbonic anhydrase inhibitors with neuropathic pain modulating effects
- (2015) Fabrizio Carta et al. BIOORGANIC & MEDICINAL CHEMISTRY
- New amide derivatives of Probenecid as selective inhibitors of carbonic anhydrase IX and XII: Biological evaluation and molecular modelling studies
- (2015) Simone Carradori et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Synthesis of sulfonamides incorporating piperazinyl-ureido moieties and their carbonic anhydrase I, II, IX and XII inhibitory activity
- (2015) Cenzo Congiu et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Synthesis of 4-[2-(3,4-dimethoxybenzyl)cyclopentyl]-1,2-dimethoxybenzene Derivatives and Evaluations of Their Carbonic Anhydrase Isoenzymes Inhibitory Effects
- (2015) Tekin Artunç et al. Chemical Biology & Drug Design
- X-ray crystallography-promoted drug design of carbonic anhydrase inhibitors
- (2015) Jekaterina Ivanova et al. CHEMICAL COMMUNICATIONS
- Synthesis, carbonic anhydrase inhibition and cytotoxic activity of novel chromone-based sulfonamide derivatives
- (2015) Fadi M. Awadallah et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Probing the ‘bipolar’ nature of the carbonic anhydrase active site: Aromatic sulfonamides containing 1,3-oxazol-5-yl moiety as picomolar inhibitors of cytosolic CA I and CA II isoforms
- (2015) Mikhail Krasavin et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Discovery of novel inhibitors for the treatment of glaucoma
- (2015) Kishore Cholkar et al. Expert Opinion on Drug Discovery
- 7-Amino-3,4-dihydro-1H-quinolin-2-one, a compound similar to the substituted coumarins, inhibitsα-carbonic anhydrases without hydrolysis of the lactam ring
- (2015) Daniela Vullo et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- 7-Aryl-triazolyl-substituted sulfocoumarins are potent, selective inhibitors of the tumor-associated carbonic anhydrase IX and XII
- (2015) Alessio Nocentini et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- Carbonic anhydrase inhibition for the management of cerebral ischemia: in vivo evaluation of sulfonamide and coumarin inhibitors
- (2015) Lorenzo Di Cesare Mannelli et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- Inhibition of carbonic anhydrase isoforms I, II, IX and XII with Schiff’s bases incorporating iminoureido moieties
- (2015) Namrata Singasane et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- The history and rationale of using carbonic anhydrase inhibitors in the treatment of peptic ulcers. In memoriam Ioan Puşcaş (1932–2015)
- (2015) György M. Buzás et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- Synthesis of 4-(2-substituted hydrazinyl)benzenesulfonamides and their carbonic anhydrase inhibitory effects
- (2015) Halise Inci Gul et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- Carbonic Anhydrase Inhibitors with Dual-Tail Moieties To Match the Hydrophobic and Hydrophilic Halves of the Carbonic Anhydrase Active Site
- (2015) Rajendra P. Tanpure et al. JOURNAL OF MEDICINAL CHEMISTRY
- 6-Substituted Sulfocoumarins Are Selective Carbonic Anhdydrase IX and XII Inhibitors with Significant Cytotoxicity against Colorectal Cancer Cells
- (2015) Aiga Grandane et al. JOURNAL OF MEDICINAL CHEMISTRY
- Nitric Oxide Donors and Selective Carbonic Anhydrase Inhibitors: A Dual Pharmacological Approach for the Treatment of Glaucoma, Cancer and Osteoporosis
- (2015) Simone Carradori et al. MOLECULES
- Targeting Carbonic Anhydrase IX Activity and Expression
- (2015) Brian Mahon et al. MOLECULES
- Eriocitrin and Apigenin as New Carbonic Anhydrase VA Inhibitors from a Virtual Screening of Calabrian Natural Products
- (2015) Maria Gidaro et al. PLANTA MEDICA
- New ways to image and target tumour hypoxia and its molecular responses
- (2015) Ludwig J. Dubois et al. RADIOTHERAPY AND ONCOLOGY
- Increased Carbonic Anhydrase Activity is Associated with Sleep Apnea Severity and Related Hypoxemia
- (2015) Tengyu Wang et al. SLEEP
- Carbonic Anhydrase Glycoinhibitors belonging to the Aminoxysulfonamide Series
- (2015) Joanna Ombouma et al. ACS Medicinal Chemistry Letters
- Carbonic anhydrase XII is a new therapeutic target to overcome chemoresistance in cancer cells
- (2015) Joanna Kopecka et al. Oncotarget
- Increased Carbonic Anhydrase Activity is Associated with Sleep Apnea Severity and Related Hypoxemia
- (2015) Tengyu Wang et al. SLEEP
- Recent Developments in Targeting Carbonic Anhydrase IX for Cancer Therapeutics
- (2015) Paul C. McDonald et al. Oncotarget
- Carbonic anhydrase inhibitors: Synthesis, molecular docking, cytotoxic and inhibition of the human carbonic anhydrase isoforms I, II, IX, XII with novel benzenesulfonamides incorporating pyrrole, pyrrolopyrimidine and fused pyrrolopyrimidine moieties
- (2014) Mostafa M. Ghorab et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Ferrier sulfamidoglycosylation of glycals catalyzed by nitrosonium tetrafluoroborate: Towards new carbonic anhydrase glycoinhibitors
- (2014) Joanna Ombouma et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Inhibition studies of new ureido-substituted sulfonamides incorporating a GABA moiety against human carbonic anhydrase isoforms I–XIV
- (2014) Mariangela Ceruso et al. BIOORGANIC & MEDICINAL CHEMISTRY
- 4-Functionalized 1,3-diarylpyrazoles bearing 6-aminosulfonylbenzothiazole moiety as potent inhibitors of carbonic anhydrase isoforms hCA I, II, IX and XII
- (2014) SitaRam et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Pyrazolo[4,3-e][1,2,4]triazine sulfonamides as carbonic anhydrase inhibitors with antitumor activity
- (2014) Mariusz Mojzych et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Synthesis of 6-tetrazolyl-substituted sulfocoumarins acting as highly potent and selective inhibitors of the tumor-associated carbonic anhydrase isoforms IX and XII
- (2014) Aiga Grandane et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Carbonic anhydrase inhibitors: Synthesis and inhibition of the human carbonic anhydrase isoforms I, II, IX and XII with benzene sulfonamides incorporating 4- and 3-nitrophthalimide moieties
- (2014) Kalyan K. Sethi et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Dual carbonic anhydrase/matrix metalloproteinase inhibitors incorporating bisphosphonic acid moieties targeting bone tumors
- (2014) Marilena Tauro et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Carbonic anhydrase inhibitory activity of sulfonamides and carboxylic acids incorporating cyclic imide scaffolds
- (2014) Alaa A.-M. Abdel-Aziz et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Synthesis and carbonic anhydrase I, II, IX and XII inhibition studies of 4-N,N-disubstituted sulfanilamides incorporating 4,4,4-trifluoro-3-oxo-but-1-enyl, phenacylthiourea and imidazol-2(3H)-one/thione moieties
- (2014) Cenzo Congiu et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- 6-Triazolyl-substituted sulfocoumarins are potent, selective inhibitors of the tumor-associated carbonic anhydrases IX and XII
- (2014) Aiga Grandane et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Novel sulfonamides bearing pyrrole and pyrrolopyrimidine moieties as carbonic anhydrase inhibitors: Synthesis, cytotoxic activity and molecular modeling
- (2014) Mostafa M. Ghorab et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Cyclic tertiary sulfamates: Selective inhibition of the tumor-associated carbonic anhydrases IX and XII by N- and O-substituted acesulfame derivatives
- (2014) Celeste De Monte et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Zonisamide reduces obstructive sleep apnoea: a randomised placebo-controlled study
- (2014) D. Eskandari et al. EUROPEAN RESPIRATORY JOURNAL
- Inhibition of human carbonic anhydrase isozymes I, II, IX and XII with a new series of sulfonamides incorporating aroylhydrazone-, [1,2,4]triazolo[3,4-b][1,3,4]thiadiazinyl- or 2-(cyanophenylmethylene)-1,3,4-thiadiazol-3(2H)-yl moieties
- (2014) Ahmed M. Alafeefy et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- Computational investigation of the selectivity of salen and tetrahydrosalen compounds towards the tumor-associated hCA XII isozyme
- (2014) Atilla Akdemir et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- Synthesis and biological activity of novel thiourea derivatives as carbonic anhydrase inhibitors
- (2014) Neslihan Korkmaz et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- Structural Insights on Carbonic Anhydrase Inhibitory Action, Isoform Selectivity, and Potency of Sulfonamides and Coumarins Incorporating Arylsulfonylureido Groups
- (2014) Murat Bozdag et al. JOURNAL OF MEDICINAL CHEMISTRY
- Structural Insights into Carbonic Anhydrase IX Isoform Specificity of Carbohydrate-Based Sulfamates
- (2014) Janina Moeker et al. JOURNAL OF MEDICINAL CHEMISTRY
- Cyclic Secondary Sulfonamides: Unusually Good Inhibitors of Cancer-Related Carbonic Anhydrase Enzymes
- (2014) Janina Moeker et al. JOURNAL OF MEDICINAL CHEMISTRY
- Inhibition of Carbonic Anhydrase Augments GABAA Receptor-Mediated Analgesia via a Spinal Mechanism of Action
- (2014) Marina N. Asiedu et al. JOURNAL OF PAIN
- Defining Phenotypic Causes of Obstructive Sleep Apnea. Identification of Novel Therapeutic Targets
- (2013) Danny J. Eckert et al. AMERICAN JOURNAL OF RESPIRATORY AND CRITICAL CARE MEDICINE
- Carbonic anhydrase inhibitors: Synthesis and inhibition of the human carbonic anhydrase isoforms I, II, VII, IX and XII with benzene sulfonamides incorporating 4,5,6,7-tetrabromophthalimide moiety
- (2013) Kalyan K. Sethi et al. BIOORGANIC & MEDICINAL CHEMISTRY
- 7-Substituted-sulfocoumarins are isoform-selective, potent carbonic anhydrase II inhibitors
- (2013) Muhammet Tanc et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Natural product hybrid and its superacid synthesized analogues: Dodoneine and its derivatives show selective inhibition of carbonic anhydrase isoforms I, III, XIII and XIV
- (2013) Hélène Carreyre et al. BIOORGANIC & MEDICINAL CHEMISTRY
- 5-Substituted-(1,2,3-triazol-4-yl)thiophene-2-sulfonamides strongly inhibit human carbonic anhydrases I, II, IX and XII: Solution and X-ray crystallographic studies
- (2013) Janis Leitans et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Synthesis and carbonic anhydrase inhibitory properties of sulfamides structurally related to dopamine
- (2013) Kadir Aksu et al. BIOORGANIC & MEDICINAL CHEMISTRY
- New superacid synthesized (fluorinated) tertiary benzenesulfonamides acting as selective hCA IX inhibitors: toward a new mode of carbonic anhydrase inhibition by sulfonamides
- (2013) Benoît Métayer et al. CHEMICAL COMMUNICATIONS
- Thiol–ene click chemistry for the synthesis of highly effective glycosyl sulfonamide carbonic anhydrase inhibitors
- (2013) Mohamed-Chiheb Saada et al. CHEMICAL COMMUNICATIONS
- Neuronal carbonic anhydrase VII provides GABAergic excitatory drive to exacerbate febrile seizures
- (2013) Eva Ruusuvuori et al. EMBO JOURNAL
- Carbonic anhydrase inhibitors. Synthesis of heterocyclic 4-substituted pyridine-3-sulfonamide derivatives and their inhibition of the human cytosolic isozymes I and II and transmembrane tumor-associated isozymes IX and XII
- (2013) Jarosław Sławiński et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Application of Monoclonal Antibody G250 Recognizing Carbonic Anhydrase IX in Renal Cell Carcinoma
- (2013) Jeannette Oosterwijk-Wakka et al. INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES
- Carbonic anhydrases: from biomedical applications of the inhibitors and activators to biotechnological use for CO2 capture
- (2013) Claudiu T. Supuran JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- Xanthates and Trithiocarbonates Strongly Inhibit Carbonic Anhydrases and Show Antiglaucoma Effects in Vivo
- (2013) Fabrizio Carta et al. JOURNAL OF MEDICINAL CHEMISTRY
- Hypoxia-Targeting Carbonic Anhydrase IX Inhibitors by a New Series of Nitroimidazole-Sulfonamides/Sulfamides/Sulfamates
- (2013) Marouan Rami et al. JOURNAL OF MEDICINAL CHEMISTRY
- Breathing and sleep at high altitude
- (2013) Philip N. Ainslie et al. RESPIRATORY PHYSIOLOGY & NEUROBIOLOGY
- New selective carbonic anhydrase IX inhibitors: Synthesis and pharmacological evaluation of diarylpyrazole-benzenesulfonamides
- (2012) Tiphaine Rogez-Florent et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Carbonic anhydrase inhibitors: Benzenesulfonamides incorporating cyanoacrylamide moieties are low nanomolar/subnanomolar inhibitors of the tumor-associated isoforms IX and XII
- (2012) Ahmed M. Alafeefy et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Ureido-substituted sulfamates show potent carbonic anhydrase IX inhibitory and antiproliferative activities against breast cancer cell lines
- (2012) Jean-Yves Winum et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Inhibition of α-class cytosolic human carbonic anhydrases I, II, IX and XII, and β-class fungal enzymes by carboxylic acids and their derivatives: New isoform-I selective nanomolar inhibitors
- (2012) Mario Sechi et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Transgenic mice over-expressing carbonic anhydrase I showed aggravated joint inflammation and tissue destruction
- (2012) Yabing Zheng et al. BMC MUSCULOSKELETAL DISORDERS
- Multiple Binding Modes of Inhibitors to Carbonic Anhydrases: How to Design Specific Drugs Targeting 15 Different Isoforms?
- (2012) Vincenzo Alterio et al. CHEMICAL REVIEWS
- Carbonic Anhydrase IX as a Target for Designing Novel Anticancer Drugs
- (2012) S. M. Monti et al. CURRENT MEDICINAL CHEMISTRY
- Ocular perfusion pressure and ocular blood flow in glaucoma
- (2012) A Popa Cherecheanu et al. CURRENT OPINION IN PHARMACOLOGY
- Effects of acetazolamide on central blood pressure, peripheral blood pressure, and arterial distensibility at acute high altitude exposure
- (2012) Gianfranco Parati et al. EUROPEAN HEART JOURNAL
- Update on carbonic anhydrase inhibitors: a patent review (2008 – 2011)
- (2012) Mayank Aggarwal et al. EXPERT OPINION ON THERAPEUTIC PATENTS
- Structure-based drug discovery of carbonic anhydrase inhibitors
- (2012) Claudiu T. Supuran JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- Inhibition of the alpha- and beta-carbonic anhydrases from the gastric pathogenHelycobacter pyloriwith anions
- (2012) Alfonso Maresca et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- Tricyclic Sulfonamides Incorporating Benzothiopyrano[4,3-c]pyrazole and Pyridothiopyrano[4,3-c]pyrazole Effectively Inhibit α- and β-Carbonic Anhydrase: X-ray Crystallography and Solution Investigations on 15 Isoforms
- (2012) Anna M. Marini et al. JOURNAL OF MEDICINAL CHEMISTRY
- Antimetastatic Effect of Sulfamate Carbonic Anhydrase IX Inhibitors in Breast Carcinoma Xenografts
- (2012) Roben G. Gieling et al. JOURNAL OF MEDICINAL CHEMISTRY
- Metallocene-Based Inhibitors of Cancer-Associated Carbonic Anhydrase Enzymes IX and XII
- (2012) Adam J. Salmon et al. JOURNAL OF MEDICINAL CHEMISTRY
- Dithiocarbamates Strongly Inhibit Carbonic Anhydrases and Show Antiglaucoma Action in Vivo
- (2012) Fabrizio Carta et al. JOURNAL OF MEDICINAL CHEMISTRY
- Acetazolamide improves loop gain but not the other physiological traits causing obstructive sleep apnoea
- (2012) Bradley A. Edwards et al. JOURNAL OF PHYSIOLOGY-LONDON
- Characterization of Carbonic Anhydrase IX Interactome Reveals Proteins Assisting Its Nuclear Localization in Hypoxic Cells
- (2012) Pasquale Buanne et al. JOURNAL OF PROTEOME RESEARCH
- Multimodal Imaging and Detection Strategy With 124 I-Labeled Chimeric Monoclonal Antibody cG250 for Accurate Localization and Confirmation of Extent of Disease During Laparoscopic and Open Surgical Resection of Clear Cell Renal Cell Carcinoma
- (2012) Stephen P. Povoski et al. Surgical Innovation
- Carbonic anhydrase I (CA1) is involved in the process of bone formation and is susceptible to ankylosing spondylitis
- (2012) Xiaotian Chang et al. ARTHRITIS RESEARCH & THERAPY
- Kinetic and docking studies of phenol-based inhibitors of carbonic anhydrase isoforms I, II, IX and XII evidence a new binding mode within the enzyme active site
- (2011) Serdar Durdagi et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Sulfonamides incorporating 1,3,5-triazine moieties selectively and potently inhibit carbonic anhydrase transmembrane isoforms IX, XII and XIV over cytosolic isoforms I and II: Solution and X-ray crystallographic studies
- (2011) Fabrizio Carta et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Synthesis of glycoconjugate carbonic anhydrase inhibitors by ruthenium-catalysed azide-alkyne 1,3-dipolar cycloaddition
- (2011) Adam J. Salmon et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Phenylethynylbenzenesulfonamide regioisomers strongly and selectively inhibit the transmembrane, tumor-associated carbonic anhydrase isoforms IX and XII over the cytosolic isoforms I and II
- (2011) Edward E. Knaus et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Virtual screening-driven identification of human carbonic anhydrase inhibitors incorporating an original, new pharmacophore
- (2011) Nicolino Pala et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- (R)-/(S)-10-Camphorsulfonyl-substituted aromatic/heterocyclic sulfonamides selectively inhibit mitochondrial over cytosolic carbonic anhydrases
- (2011) Alfonso Maresca et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- N-β-Glycosyl sulfamides are selective inhibitors of the cancer associated carbonic anhydrase isoforms IX and XII
- (2011) Oscar M. Rodríguez et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- In vitro inhibition of α-carbonic anhydrase isozymes by some phenolic compounds
- (2011) Sevim Beyza Öztürk Sarikaya et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Generation and characterization of the first inhibitory antibody targeting tumour-associated carbonic anhydrase XII
- (2011) Christina Battke et al. CANCER IMMUNOLOGY IMMUNOTHERAPY
- Targeting Tumor Hypoxia: Suppression of Breast Tumor Growth and Metastasis by Novel Carbonic Anhydrase IX Inhibitors
- (2011) Y. Lou et al. CANCER RESEARCH
- Medical Management of Parkinsons Disease: Focus on Neuroprotection
- (2011) Camilo Rios et al. Current Neuropharmacology
- Sulfapyridine-like benzenesulfonamide derivatives as inhibitors of carbonic anhydrase isoenzymes I, II and VI
- (2011) Cemalettin Alp et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- Glycosyl Coumarin Carbonic Anhydrase IX and XII Inhibitors Strongly Attenuate the Growth of Primary Breast Tumors
- (2011) Nadia Touisni et al. JOURNAL OF MEDICINAL CHEMISTRY
- Targeting Hypoxic Tumor Cell Viability with Carbohydrate-Based Carbonic Anhydrase IX and XII Inhibitors
- (2011) Jason C. Morris et al. JOURNAL OF MEDICINAL CHEMISTRY
- Design, Synthesis, and Biological Evaluation of Novel Carbohydrate-Based Sulfamates as Carbonic Anhydrase Inhibitors
- (2011) Marie Lopez et al. JOURNAL OF MEDICINAL CHEMISTRY
- Ureido-Substituted Benzenesulfonamides Potently Inhibit Carbonic Anhydrase IX and Show Antimetastatic Activity in a Model of Breast Cancer Metastasis
- (2011) Fabio Pacchiano et al. JOURNAL OF MEDICINAL CHEMISTRY
- Using Recombinant Tissue Plasminogen Activator to Treat Acute Ischemic Stroke in China
- (2011) Yilong Wang et al. STROKE
- Inhibition of Carbonic Anhydrase Reduces Brain Injury After Intracerebral Hemorrhage
- (2011) Fuyou Guo et al. Translational Stroke Research
- Is the incidence of rheumatoid arthritis rising?: Results from Olmsted County, Minnesota, 1955-2007
- (2010) Elena Myasoedova et al. ARTHRITIS AND RHEUMATISM
- Pteridine–sulfonamide conjugates as dual inhibitors of carbonic anhydrases and dihydrofolate reductase with potential antitumor activity
- (2010) Sérgio M. Marques et al. BIOORGANIC & MEDICINAL CHEMISTRY
- NO-releasing esters show carbonic anhydrase inhibitory action against human isoforms I and II
- (2010) Deniz Ekinci et al. BIOORGANIC & MEDICINAL CHEMISTRY
- 7,8-Disubstituted- but not 6,7-disubstituted coumarins selectively inhibit the transmembrane, tumor-associated carbonic anhydrase isoforms IX and XII over the cytosolic ones I and II in the low nanomolar/subnanomolar range
- (2010) Alfonso Maresca et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Coumarins incorporating hydroxy- and chloro-moieties selectively inhibit the transmembrane, tumor-associated carbonic anhydrase isoforms IX and XII over the cytosolic ones I and II
- (2010) Alfonso Maresca et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Increased expression of carbonic anhydrase I in the synovium of patients with ankylosing spondylitis
- (2010) Xiaotian Chang et al. BMC MUSCULOSKELETAL DISORDERS
- Drug Design Studies of the Novel Antitumor Targets Carbonic Anhydrase IX and XII
- (2010) O. Guler et al. CURRENT MEDICINAL CHEMISTRY
- Carbonic Anhydrase Related Protein VIII and its Role in Neurodegeneration and Cancer
- (2010) Ashok Aspatwar et al. CURRENT PHARMACEUTICAL DESIGN
- Sulfonamide Linked Neoglycoconjugates−A New Class of Inhibitors for Cancer-Associated Carbonic Anhydrases
- (2010) Marie Lopez et al. JOURNAL OF MEDICINAL CHEMISTRY
- Polyamines Inhibit Carbonic Anhydrases by Anchoring to the Zinc-Coordinated Water Molecule
- (2010) Fabrizio Carta et al. JOURNAL OF MEDICINAL CHEMISTRY
- Recommendations for the Pharmacological Management of Neuropathic Pain: An Overview and Literature Update
- (2010) Robert H. Dworkin et al. MAYO CLINIC PROCEEDINGS
- Protein Carbonylation in Skeletal Muscles: Impact on Function
- (2009) Esther Barreiro et al. ANTIOXIDANTS & REDOX SIGNALING
- Carbonic anhydrase III is insufficient in muscles of myasthenia gravis patients
- (2009) Ai-Lian Du et al. AUTOIMMUNITY
- Carbonic anhydrase IX: Biochemical and crystallographic characterization of a novel antitumor target
- (2009) Giuseppina De Simone et al. BIOCHIMICA ET BIOPHYSICA ACTA-PROTEINS AND PROTEOMICS
- Expression of transmembrane carbonic anhydrases, CAIX and CAXII, in human development
- (2009) Shu-Yuan Liao et al. BMC DEVELOPMENTAL BIOLOGY
- Which Carbonic Anhydrases are Targeted by the Antiepileptic Sulfonamides and Sulfamates?
- (2009) Giuseppina De Simone et al. Chemical Biology & Drug Design
- Elevated erythrocyte carbonic anhydrase activity is a novel clinical marker in hyperventilation syndrome
- (2009) Ying-Hock Teng et al. CLINICAL CHEMISTRY AND LABORATORY MEDICINE
- Carbonic Anhydrase Inhibitors. Comparison of Aliphatic Sulfamate/Bis-sulfamate Adducts with Isozymes II and IX as a Platform for Designing Tight-Binding, More Isoform-Selective Inhibitors
- (2009) Rosa Maria Vitale et al. JOURNAL OF MEDICINAL CHEMISTRY
- Deciphering the Mechanism of Carbonic Anhydrase Inhibition with Coumarins and Thiocoumarins
- (2009) Alfonso Maresca et al. JOURNAL OF MEDICINAL CHEMISTRY
- Acetazolamide and midazolam act synergistically to inhibit neuropathic pain
- (2009) Marina Asiedu et al. PAIN
- Pathogenesis of retinitis pigmentosa associated with apoptosis-inducing mutations in carbonic anhydrase IV
- (2009) R. Datta et al. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA
- Crystal structure of the catalytic domain of the tumor-associated human carbonic anhydrase IX
- (2009) V. Alterio et al. PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA
- Bio-sequestration of carbon dioxide using carbonic anhydrase enzyme purified from Citrobacter freundii
- (2009) Rishiram Ramanan et al. WORLD JOURNAL OF MICROBIOLOGY & BIOTECHNOLOGY
- Molecular mechanisms of carbonic anhydrase IX-mediated pH regulation under hypoxia
- (2008) Silvia Pastorekova et al. BJU INTERNATIONAL
- Hypoxia-Inducible Carbonic Anhydrase IX and XII Promote Tumor Cell Growth by Counteracting Acidosis through the Regulation of the Intracellular pH
- (2008) J. Chiche et al. CANCER RESEARCH
- Anticonvulsant Sulfonamides/Sulfamates/Sulfamides with Carbonic Anhydrase Inhibitory Activity: Drug Design and Mechanism of Action
- (2008) Bernard Masereel et al. CURRENT PHARMACEUTICAL DESIGN
- Diuretics: From Classical Carbonic Anhydrase Inhibitors to Novel Applications of the Sulfonamides
- (2008) Claudiu Supuran CURRENT PHARMACEUTICAL DESIGN
- Entrapment of Carbon Dioxide in the Active Site of Carbonic Anhydrase II
- (2008) John F. Domsic et al. JOURNAL OF BIOLOGICAL CHEMISTRY
- Inhibition of Carbonic Anhydrases with Glycosyltriazole Benzene Sulfonamides
- (2008) Brendan L. Wilkinson et al. JOURNAL OF MEDICINAL CHEMISTRY
- Carbonic anhydrases: novel therapeutic applications for inhibitors and activators
- (2008) Claudiu T. Supuran NATURE REVIEWS DRUG DISCOVERY
- Crystal structure of human carbonic anhydrase XIII and its complex with the inhibitor acetazolamide
- (2008) Anna Di Fiore et al. PROTEINS-STRUCTURE FUNCTION AND BIOINFORMATICS
- Antibody therapy in renal cell carcinoma
- (2008) Egbert Oosterwijk et al. WORLD JOURNAL OF UROLOGY
- Prevalence of chronic pain with neuropathic characteristics in the general population
- (2007) Didier Bouhassira et al. PAIN
Find Funding. Review Successful Grants.
Explore over 25,000 new funding opportunities and over 6,000,000 successful grants.
ExplorePublish scientific posters with Peeref
Peeref publishes scientific posters from all research disciplines. Our Diamond Open Access policy means free access to content and no publication fees for authors.
Learn More