Recent advances in indole syntheses: New routes for a classic target

Rhodium-Catalyzed Synthesis of 2,3-Disubstituted Indoles from β,β-Disubstituted Stryryl Azides

(2011) Ke Sun et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Microwave-Assisted Synthesis of Medicinally Relevant Indoles

(2011) S. A. Patil et al.   CURRENT MEDICINAL CHEMISTRY

Synthesis ofN-(2-Pyridyl)indoles via Pd(II)-Catalyzed Oxidative Coupling

(2011) Jinlei Chen et al.   JOURNAL OF ORGANIC CHEMISTRY

Distribution of the Cationic State over the Chlorophyll Pair of the Photosystem II Reaction Center

(2011) Keisuke Saito et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Rh2(II)-Catalyzed Nitro-Group Migration Reactions: Selective Synthesis of 3-Nitroindoles from β-Nitro Styryl Azides

(2011) Benjamin J. Stokes et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Palladium-Catalyzed Intramolecular Trapping of the Blaise Reaction Intermediate for Tandem One-Pot Synthesis of Indole Derivatives

(2011) Ju Hyun Kim et al.   ORGANIC LETTERS

Nickel-Catalyzed Cycloaddition of Anthranilic Acid Derivatives to Alkynes

(2011) Nobuyoshi Maizuru et al.   ORGANIC LETTERS

Palladium-Catalyzed Selective Heck-Type Diarylation of Allylic Esters with Aryl Halides Involving a β-OAc Elimination Process

(2011) Yan Liu et al.   ORGANIC LETTERS

A Facile Route to Polysubstituted Indoles via Three-Component Reaction of 2-Ethynylaniline, Sulfonyl Azide, and Nitroolefin

(2011) Zhiyuan Chen et al.   ORGANIC LETTERS

CuBr-Catalyzed Coupling ofN-Tosylhydrazones and Terminal Alkynes: Synthesis of Benzofurans and Indoles

(2011) Lei Zhou et al.   ORGANIC LETTERS

Iron(II) Triflate as a Catalyst for the Synthesis of Indoles by Intramolecular C−H Amination

(2011) Julien Bonnamour et al.   ORGANIC LETTERS

A Novel One-Pot, Two-Step Synthesis of Polycyclic Indoles via Tandem Intramolecular Hydroamidation/Palladium-Catalyzed Annulation

(2010) Jianxiu Liu et al.   ADVANCED SYNTHESIS & CATALYSIS

Sulfur-Assisted and 1,8-Diazabicyclo[5.4.0]undec-7-ene (DBU)-Catalyzed Cyclization of 2-Alkynylanilines for the Metal-Free Synthesis of Indole Derivatives

(2010) Hongwei Zhou et al.   ADVANCED SYNTHESIS & CATALYSIS

Cascade Palladium-Catalyzed Direct Intramolecular Arylation/Alkene Isomerization Sequences: Synthesis of Indoles and Benzofurans

(2010) Myriam Yagoubi et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Fischer Indole Synthesis with Organozinc Reagents

(2010) Benjamin A. Haag et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Gold-Catalyzed Cycloisomerization Reactions of 2-Tosylaminophenylprop-1-yn-3-ols as a Versatile Approach for Indole Synthesis

(2010) Prasath Kothandaraman et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Preparation of indoles via iron catalyzed direct oxidative coupling

(2010) Zheng-Hui Guan et al.   CHEMICAL COMMUNICATIONS

[Fe(F20TPP)Cl] catalyzed intramolecular C–N bond formation for alkaloid synthesis using aryl azides as nitrogen source

(2010) Yungen Liu et al.   CHEMICAL COMMUNICATIONS

A two step route to indoles from haloarenes—a versatile variation on the Fischer indole synthesis

(2010) Martyn Inman et al.   CHEMICAL COMMUNICATIONS

A general and mild domino approach to substituted 1-aminoindoles

(2010) Nis Halland et al.   CHEMICAL COMMUNICATIONS

Continuous flow thermolysis of azidoacrylates for the synthesis of heterocycles and pharmaceutical intermediates

(2010) Alexander G. O'Brien et al.   CHEMICAL COMMUNICATIONS

Synthesis of Indoles by Conjugate Addition and Ligand-Free Copper-Catalyzed Intramolecular Arylation of Activated Acetylenes with o-Haloanilines

(2010) Detian Gao et al.   CHEMISTRY-A EUROPEAN JOURNAL

“On-Water,” Microwave-Assisted, Pd-Catalyzed Synthesis of Indoles from Imines and o-Difunctionalized Arenes

(2010) José Barluenga et al.   CHEMISTRY-A EUROPEAN JOURNAL

A General Synthesis of Alkenyl-Substituted Benzofurans, Indoles, and Isoquinolones by Cascade Palladium-Catalyzed Heterocyclization/Oxidative Heck Coupling

(2010) Rosana Álvarez et al.   CHEMISTRY-A EUROPEAN JOURNAL

Synthesis of Indole Derivatives with Biological Activity by Reactions Between Unsaturated Hydrocarbons and N-Aromatic Precursors

(2010) Giovanni Palmisano et al.   CURRENT ORGANIC CHEMISTRY

Mechanistic Dichotomy with Alkynes in the Formal Hydrohydrazination/Fischer Indolization Tandem Reaction Catalyzed by a Ph3PAuNTf2/pTSA Binary System

(2010) Nitin T. Patil et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Synthesis of Substituted Indole from 2-Aminobenzaldehyde through [1,2]-Aryl Shift

(2010) Patrick Levesque et al.   JOURNAL OF ORGANIC CHEMISTRY

Platinum-Catalyzed, One-Pot Tandem Synthesis of Indoles and Isoquinolines via Sequential Rearrangement of Amides and Aminocyclization

(2010) Noriko Okamoto et al.   JOURNAL OF ORGANIC CHEMISTRY

Nickel-catalyzed, base-mediated amination/hydroamination reaction sequence for a modular synthesis of indoles

(2010) Lutz Ackermann et al.   JOURNAL OF ORGANOMETALLIC CHEMISTRY

Total Synthesis of Complestatin: Development of a Pd(0)-Mediated Indole Annulation for Macrocyclization

(2010) Hiroyuki Shimamura et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

The Role of Reversible Oxidative Addition in Selective Palladium(0)-Catalyzed Intramolecular Cross-Couplings of Polyhalogenated Substrates: Synthesis of Brominated Indoles

(2010) Stephen G. Newman et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Palladium-Catalyzed Amination of Aromatic C−H Bonds with Oxime Esters

(2010) Yichen Tan et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Domino Process in Silver-Catalyzed Reactions ofN-Arylformimidates and Active Methylene Compounds Involving Cycloisomerization and 1,3-Alkenyl Shift

(2010) Chang Ho Oh et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Rhodium(III)-Catalyzed Arene and Alkene C−H Bond Functionalization Leading to Indoles and Pyrroles

(2010) David R. Stuart et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Copper catalysis in the construction of indole and benzo[b]furan rings

(2010) Sandro Cacchi et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Multicatalytic One-Pot Reaction of 1-(2-Alkynylphenyl)ketoximes for Generation of Indole Derivatives

(2010) Guanyinsheng Qiu et al.   ORGANIC LETTERS

Fe(II)-Catalyzed Amination of Aromatic C−H Bonds via Ring Opening of 2H-Azirines: Synthesis of 2,3-Disubstituted Indoles

(2010) Samaresh Jana et al.   ORGANIC LETTERS

A Novel Approach to 3-Methylindoles by a Heck/Cyclization/Isomerization Process

(2010) Carl A. Baxter et al.   ORGANIC LETTERS

Cationic Pd(II)-Catalyzed Tandem Reaction of 2-Arylethynylanilines and Aldehydes: An Efficient Synthesis of Substituted 3-Hydroxymethyl Indoles

(2010) Xiuling Han et al.   ORGANIC LETTERS

2,3-Disubstituted Indoles via Palladium-Catalyzed Reaction of 2-Alkynyltrifluoroacetanilides with Arenediazonium Tetrafluoroborates

(2010) Sandro Cacchi et al.   ORGANIC LETTERS

Rh(III)-Catalyzed Oxidative Coupling ofN-Aryl-2-aminopyridine with Alkynes and Alkenes

(2010) Jinlei Chen et al.   ORGANIC LETTERS

Exploiting the Chemistry of Strained Rings: Synthesis of Indoles via Domino Reaction of Aryl Iodides with 2H-Azirines

(2010) David A. Candito et al.   ORGANIC LETTERS

Palladium catalyzed tandem alkenyl- and aryl-C–N bond formation: a cascade N-annulation route to 4-, 5-, 6- and 7-chloroindoles

(2010) Luke C. Henderson et al.   TETRAHEDRON

Cupric Halide-Mediated Intramolecular Halocyclization of N-Electron-Withdrawing Group-Substituted 2-Alkynylanilines for the Synthesis of 3-Haloindoles

(2009) Zengming Shen et al.   ADVANCED SYNTHESIS & CATALYSIS

Copper-CatalyzedN-Arylation/Hydroamin(d)ation Domino Synthesis of Indoles and its Application to the Preparation of a Chek1/KDR Kinase Inhibitor Pharmacophore

(2009) Lutz Ackermann et al.   ADVANCED SYNTHESIS & CATALYSIS

Enantioselective Gold-Catalyzed Allylic Alkylation of Indoles with Alcohols: An Efficient Route to Functionalized Tetrahydrocarbazoles

(2009) Marco Bandini et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Metal-Ion Selectivity of Chemically Modified Uracil Pairs in DNA Duplexes

(2009) Itaru Okamoto et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Copper-Catalyzed CC Bond Formation through CH Functionalization: Synthesis of Multisubstituted Indoles fromN-Aryl Enaminones

(2009) Roberta Bernini et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Indoles from Simple Anilines and Alkynes: Palladium-Catalyzed CH Activation Using Dioxygen as the Oxidant

(2009) Zhuangzhi Shi et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Assembly of indole-2-carboxylic acid esters through a ligand-free copper-catalysed cascade process

(2009) Qian Cai et al.   CHEMICAL COMMUNICATIONS

Recent Advances in the Synthesis of Indole and Quinoline Derivatives through Cascade Reactions

(2009) José Barluenga et al.   Chemistry-An Asian Journal

Examination of the Mechanism of Rh2(II)-Catalyzed Carbazole Formation Using Intramolecular Competition Experiments

(2009) Benjamin J. Stokes et al.   JOURNAL OF ORGANIC CHEMISTRY

Construction of Nitrogen Heterocycles Bearing an Aminomethyl Group by Copper-Catalyzed Domino Three-Component Coupling−Cyclization

(2009) Yusuke Ohta et al.   JOURNAL OF ORGANIC CHEMISTRY

Total Synthesis of Chloropeptin II (Complestatin) and Chloropeptin I

(2009) Joie Garfunkle et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Modular Synthesis of Indoles from Imines ando-Dihaloarenes oro-Chlorosulfonates by a Pd-Catalyzed Cascade Process

(2009) José Barluenga et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Palladium-Catalyzed Domino C,N-Coupling/Carbonylation/Suzuki Coupling Reaction: An Efficient Synthesis of 2-Aroyl-/Heteroaroylindoles

(2009) Martin Arthuis et al.   ORGANIC LETTERS

Rhodium(I)-Catalyzed Cyclization Reaction ofo-Alkynyl Phenols and Anilines. Domino Approach to 2,3-Disubstituted Benzofurans and Indoles

(2009) Naohiro Isono et al.   ORGANIC LETTERS

PIDA-Mediated Oxidative C−C Bond Formation: Novel Synthesis of Indoles fromN-Aryl Enamines

(2009) Wenquan Yu et al.   ORGANIC LETTERS

Simple Conversion of Enamines to 2H-Azirines and Their Rearrangements under Thermal Conditions

(2009) Xiaoxun Li et al.   ORGANIC LETTERS

Facile Synthesis of 1,2,3,4-Tetrahydro-β-carbolines by One-Pot Domino Three-Component Indole Formation and Nucleophilic Cyclization

(2009) Yusuke Ohta et al.   ORGANIC LETTERS

Palladium-Catalyzed Indolization ofN-Aroylbenzotriazoles with Disubstituted Alkynes

(2009) Itaru Nakamura et al.   ORGANIC LETTERS

Thieme Chemistry Journal Awardees - Where Are They Now? Palladium-Catalyzed N-Arylation-Hydroamination Sequence for the Synthesis of Indoles with Sterically Demanding N-Substituents

(2009) Lutz Ackermann et al.   SYNLETT

Palladium-catalyzed sequential indole synthesis using sterically hindered amines

(2009) Lutz Ackermann et al.   TETRAHEDRON

Catalytic Synthesis of Indoles from Alkynes

(2008) Karolin Krüger (née Alex) et al.   ADVANCED SYNTHESIS & CATALYSIS

Synthesis of N-Fused Tricyclic Indoles by a Tandem [1,2] Stevens-Type Rearrangement/1,2-Alkyl Migration of Metal-Containing Ammonium Ylides

(2008) Jun Takaya et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Expanding the [1,2]-Aryl Migration to the Synthesis of Substituted Indoles

(2008) Tao Pei et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Zinc-Promoted Hydrohydrazination of Terminal Alkynes: An Efficient Domino Synthesis of Indoles

(2008) Karolin Alex et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Palladium-Catalyzed Oxidative Cyclization ofN-Aryl Enamines: From Anilines to Indoles

(2008) Sebastian Würtz et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Dirhodium(II)-Catalyzed Intramolecular CH Amination of Aryl Azides

(2008) Meihua Shen et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Coinage Metal-Assisted Synthesis of Heterocycles

(2008) Nitin T. Patil et al.   CHEMICAL REVIEWS

Synthesis of Indoles via Domino Reaction ofN-Aryl Amides and Ethyl Diazoacetate

(2008) Sun-Liang Cui et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Indole Synthesis via Rhodium Catalyzed Oxidative Coupling of Acetanilides and Internal Alkynes

(2008) David R. Stuart et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Tandem copper-catalysed aryl and alkenyl amination reactions: the synthesis of N-functionalised indoles

(2008) Roy C. Hodgkinson et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Alternating Iodonium-Mediated Reaction Cascades Giving Indole- And Quinoline-Containing Polycycles

(2008) Rosliana Halim et al.   ORGANIC LETTERS

Silver-Promoted Domino Pd-Catalyzed Amination/Direct Arylation: Access to Polycyclic Heteroaromatics

(2008) Christopher S. Bryan et al.   ORGANIC LETTERS

Tandem Palladium-Catalyzed N,C-Coupling/Carbonylation Sequence for the Synthesis of 2-Carboxyindoles

(2008) Tiago O. Vieira et al.   ORGANIC LETTERS

Titanium-Catalyzed Hydrohydrazination with Monosubstituted Hydrazines: Catalyst Design, Synthesis, and Reactivity

(2008) Sanjukta Banerjee et al.   ORGANOMETALLICS

Palladium-Catalyzed Aryl Amination–Heck Cyclization Cascade: A One-Flask Approach to 3-Substituted Indoles

(2007) Thomas Jensen et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Platinum-Catalyzed Formation of Cyclic-Ketone-Fused Indoles fromN-(2-Alkynylphenyl)lactams

(2007) Guotao Li et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

One-Pot Multicomponent Synthesis of Indoles from 2-Iodobenzoic Acid

(2007) Olivier Leogane et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Pd PEPPSI-IPr-Mediated Reactions in Metal-Coated Capillaries Under MACOS: The Synthesis of Indoles by Sequential Aryl Amination/ Heck Coupling

(2007) Gjergji Shore et al.   CHEMISTRY-A EUROPEAN JOURNAL

A Highly Selective Tandem Cross-Coupling ofgem-Dihaloolefins for a Modular, Efficient Synthesis of Highly Functionalized Indoles

(2007) Yuan-Qing Fang et al.   JOURNAL OF ORGANIC CHEMISTRY

Preparation of Fully Substituted Anilines for the Synthesis of Functionalized Indoles

(2007) Armin H. Stoll et al.   ORGANIC LETTERS

Annulation of internal alkynes through a hydroamination/aza-Heck reaction sequence for the regioselective synthesis of indoles

(2007) Lutz Ackermann et al.   TETRAHEDRON