Sortase ligation enables homogeneous GPCR phosphorylation to reveal diversity in β-arrestin coupling

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Distinct conformations of GPCR–β-arrestin complexes mediate desensitization, signaling, and endocytosis

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Internalized TSH receptors en route to the TGN induce local Gs-protein signaling and gene transcription

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Identification of key phosphorylation sites in PTH1R that determine arrestin3 binding and fine-tune receptor signaling

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The β-Arrestins: Multifunctional Regulators of G Protein-coupled Receptors

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Functional competence of a partially engaged GPCR–β-arrestin complex

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Nanodiscs for structural and functional studies of membrane proteins

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Structural insights into µ-opioid receptor activation

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A Brief History of G-Protein Coupled Receptors (Nobel Lecture)

(2013) Robert J. Lefkowitz   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Structure of active β-arrestin-1 bound to a G-protein-coupled receptor phosphopeptide

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Activation and allosteric modulation of a muscarinic acetylcholine receptor

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Conformational biosensors reveal GPCR signalling from endosomes

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Noncanonical GPCR signaling arising from a PTH receptor–arrestin–Gβγ complex

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Molecular Mechanism of β-Arrestin-Biased Agonism at Seven-Transmembrane Receptors

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Distinct Phosphorylation Sites on the  2-Adrenergic Receptor Establish a Barcode That Encodes Differential Functions of  -Arrestin

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β-arrestin-mediated receptor trafficking and signal transduction

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Differential G-protein-coupled Receptor Phosphorylation Provides Evidence for a Signaling Bar Code

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The effect of ligand efficacy on the formation and stability of a GPCR-G protein complex

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Peptide−Sugar Ligation Catalyzed by Transpeptidase Sortase:  A Facile Approach to Neoglycoconjugate Synthesis

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Lipid Modification of Proteins through Sortase-Catalyzed Transpeptidation

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Structural diversity of G protein-coupled receptors and significance for drug discovery

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