Valdecoxib vs. borazavaldecoxib: isoxazole BN/CC isosterism as a case study in designing and stabilizing boron heterocycles

The State of the Art in Azaborine Chemistry: New Synthetic Methods and Applications

(2018) Zachary X. Giustra et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Structural basis for selective inhibition of Cyclooxygenase-1 (COX-1) by diarylisoxazoles mofezolac and 3-(5-chlorofuran-2-yl)-5-methyl-4-phenylisoxazole (P6)

(2017) Gino Cingolani et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synergic “Click” Boronate/Thiosemicarbazone System for Fast and Irreversible Bioorthogonal Conjugation in Live Cells

(2017) Burcin Akgun et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Fast and Tight Boronate Formation for Click Bioorthogonal Conjugation

(2016) Burcin Akgun et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Chemical philanthropy: a path forward for antibiotic discovery?

(2016) Karl A Hansford et al.   Future Medicinal Chemistry

A Study of Boratriazaroles: An Underdeveloped Class of Heterocycles

(2016) Sean K. Liew et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis, characterization, antimicrobial activity, and QSAR studies on substituted oxadiazaboroles

(2016) Meryem Pir et al.   MEDICINAL CHEMISTRY RESEARCH

Characterization of the Dynamic Equilibrium between Closed and Open Forms of the Benzoxaborole Pharmacophore

(2016) Sergey Vshyvenko et al.   ACS Medicinal Chemistry Letters

A Four-Component Reaction for the Synthesis of Dioxadiazaborocines

(2015) Thomas Flagstad et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Recent Developments in the Chemistry and Biological Applications of Benzoxaboroles

(2015) Agnieszka Adamczyk-Woźniak et al.   CHEMICAL REVIEWS

General role of the amino and methylsulfamoyl groups in selective cyclooxygenase(COX)-1 inhibition by 1,4-diaryl-1,2,3-triazoles and validation of a predictive pharmacometric PLS model

(2015) Maria Grazia Perrone et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Condensation-Driven Assembly of Boron-Containing Bis(Heteroaryl) Motifs Using a Linchpin Approach

(2015) Shinya Adachi et al.   ORGANIC LETTERS

Helping Chemists Discover New Antibiotics

(2015) Mark A. T. Blaskovich et al.   ACS Infectious Diseases

The unique chemistry of benzoxaboroles: Current and emerging applications in biotechnology and therapeutic treatments

(2014) C. Tony Liu et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis and Stability of Boratriazaroles

(2014) Didier Zurwerra et al.   ORGANIC LETTERS

Selection of boron reagents for Suzuki–Miyaura coupling

(2013) Alastair J. J. Lennox et al.   CHEMICAL SOCIETY REVIEWS

Discovery of new heterocycles with activity against human neutrophile elastase based on a boron promoted one-pot assembly reaction

(2013) Francesco Montalbano et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Orthogonal aerobic conversion of N-benzyl amidoximes to 1,2,4-oxadiazoles or quinazolinones

(2013) Feng-Lian Zhang et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

The synthesis of benzoxaboroles and their applications in medicinal chemistry

(2013) Jiong Zhang et al.   Science China-Chemistry

Recent Advances in Azaborine Chemistry

(2012) Patrick G. Campbell et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

UV-Photoelectron Spectroscopy of 1,2- and 1,3-Azaborines: A Combined Experimental and Computational Electronic Structure Analysis

(2012) Anna Chrostowska et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Boron-containing inhibitors of synthetases

(2011) Stephen J. Baker et al.   CHEMICAL SOCIETY REVIEWS

Development of novel drugs for human African trypanosomiasis

(2011) Reto Brun et al.   Future Microbiology

Enantioselective preparation and chemoselective cross-coupling of 1,1-diboron compounds

(2011) Jack Chang Hung Lee et al.   Nature Chemistry

Synthesis of Benzisoxazoles by the [3 + 2] Cycloaddition ofin situGenerated Nitrile Oxides and Arynes

(2010) Anton V. Dubrovskiy et al.   ORGANIC LETTERS

A Hybrid Organic/Inorganic Benzene

(2008) Adam J. V. Marwitz et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Crystal Clear Structural Evidence for Electron Delocalization in 1,2-Dihydro-1,2-azaborines

(2008) Eric R. Abbey et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthesis of new thiophene, furan and pyridine substituted 1,2,4,5-oxadiazaboroles

(2008) Yaşar Dürüst et al.   POLYHEDRON

Cyclic Triolborates: Air- and Water-Stable Ate Complexes of Organoboronic Acids

(2007) Yasunori Yamamoto et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Simple, Efficient, and Modular Syntheses of Polyene Natural Products via Iterative Cross-Coupling

(2007) Suk Joong Lee et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY