TBHP as Methyl Source under Metal-Free Aerobic Conditions To Synthesize Quinazolin-4(3H )-ones and Quinazolines by Oxidative Amination of C(sp3 )-H Bond

Synthesis of Quinazolines via an Iron-Catalyzed Oxidative Amination of N–H Ketimines

(2018) Cheng-yi Chen et al.   JOURNAL OF ORGANIC CHEMISTRY

Quinazoline derivatives as selective CYP1B1 inhibitors

(2017) Mohd Usman Mohd Siddique et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Metal-free radical C–H methylation of pyrimidinones and pyridinones with dicumyl peroxide

(2017) Pei-Zhi Zhang et al.   GREEN CHEMISTRY

Copper-catalyzed S-methylation of sulfonyl hydrazides with TBHP for the synthesis of methyl sulfones in water

(2017) Yu Yang et al.   GREEN CHEMISTRY

Approach to the Synthesis of 2,3-Disubstituted-3H-quinazolin-4-ones Mediated by Ph3P–I2

(2017) Wong Phakhodee et al.   JOURNAL OF ORGANIC CHEMISTRY

Intramolecular functionalization of C(sp 3 ) H bonds adjacent to an amide nitrogen atom: Metal-free synthesis of 2-hydroxy-benzoxazinone derivatives

(2017) Biao Gao et al.   TETRAHEDRON

Copper-catalyzed methylation of 1,3-diketones with tert -butyl peroxybenzoate

(2017) Zhi-Hao Zhou et al.   TETRAHEDRON

Identification of potent cholecystokinin-B receptor antagonists: synthesis, molecular modeling and anti-cancer activity against pancreatic cancer cells

(2017) Saroj Kumari et al.   MedChemComm

Synthesis of 3-Substituted Quinazolinones via C-N and C-C bond Cleavage of Enaminone

(2017) Sethurajan Ambethkar et al.   ChemistrySelect

Iron(III)-Catalyzed Peroxide-Mediated C-3 Functionalization of Flavones

(2016) Bilal Ahmad Mir et al.   ADVANCED SYNTHESIS & CATALYSIS

Quinazolines and quinazolinones as ubiquitous structural fragments in medicinal chemistry: An update on the development of synthetic methods and pharmacological diversification

(2016) Imtiaz Khan et al.   BIOORGANIC & MEDICINAL CHEMISTRY

2-(3-Methoxyphenyl)quinazoline Derivatives: A New Class of Direct Constitutive Androstane Receptor (CAR) Agonists

(2016) Tomas Smutny et al.   JOURNAL OF MEDICINAL CHEMISTRY

One-pot three-component synthesis of quinazolines via a copper-catalysed oxidative amination reaction

(2016) Tiantian Duan et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Recent developments in transition metal catalysis for quinazolinone synthesis

(2016) T. M. M. Maiden et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Acceptorless Dehydrogenative Coupling of o-Aminobenzamides with the Activation of Methanol as a C1 Source for the Construction of Quinazolinones

(2016) Feng Li et al.   ORGANIC LETTERS

Quinazoline Synthesis via Rh(III)-Catalyzed Intermolecular C–H Functionalization of Benzimidates with Dioxazolones

(2016) Jie Wang et al.   ORGANIC LETTERS

Metal-Free Oxidative 1,2-Arylmethylation Cascades of N-(Arylsulfonyl)acrylamides Using Peroxides as the Methyl Resource

(2016) Fang-Lin Tan et al.   ORGANIC LETTERS

Divergent Synthesis of Quinazolin-4(3H)-ones and Tryptanthrins Enabled by a tert-Butyl Hydroperoxide/K3PO4-Promoted Oxidative Cyclization of Isatins at Room Temperature

(2016) Feng-Cheng Jia et al.   ORGANIC LETTERS

Concise SAR Exploration Based on the “Head-to-Tail” Approach: Discovery of PI4KIIIα Inhibitors Bearing Diverse Scaffolds

(2016) Satoru Noji et al.   ACS Medicinal Chemistry Letters

Iodine-Catalyzed Oxidative Benzylic C−H Bond Amination of Azaarenes: Practical Synthesis of Quinazolin-4(3 H )-ones

(2016) Luo Yang et al.   Asian Journal of Organic Chemistry

Direct and metal-free oxidative amination of sp3 C–H bonds for the construction of 2-hetarylquinazolin-4(3H)-ones

(2016) Huanhuan Liu et al.   Organic Chemistry Frontiers

The cascade synthesis of quinazolinones and quinazolines using an α-MnO2 catalyst and tert-butyl hydroperoxide (TBHP) as an oxidant

(2015) Zhe Zhang et al.   CHEMICAL COMMUNICATIONS

Synthetic approaches, functionalization and therapeutic potential of quinazoline and quinazolinone skeletons: The advances continue

(2015) Imtiaz Khan et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Sulfate Radical Anion (SO4•–) Mediated C(sp3)–H Nitrogenation/Oxygenation in N-Aryl Benzylic Amines Expanded the Scope for the Synthesis of Benzamidine/Oxazine Heterocycles

(2015) Joydev K. Laha et al.   JOURNAL OF ORGANIC CHEMISTRY

I2-Catalyzed Aerobic Oxidative C(sp3)–H Amination/C–N Cleavage of Tertiary Amine: Synthesis of Quinazolines and Quinazolinones

(2015) Yizhe Yan et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-Catalyzed Radical Methylation/C–H Amination/Oxidation Cascade for the Synthesis of Quinazolinones

(2015) Yajie Bao et al.   JOURNAL OF ORGANIC CHEMISTRY

Metal- and Oxidant-Free Synthesis of Quinazolinones from β-Ketoesters with o-Aminobenzamides via Phosphorous Acid-Catalyzed Cyclocondensation and Selective C–C Bond Cleavage

(2015) Zhongwen Li et al.   JOURNAL OF ORGANIC CHEMISTRY

Iodine Catalyzed Oxidative Synthesis of Quinazolin-4(3H)-ones and Pyrazolo[4,3-d]pyrimidin-7(6H)-ones via Amination of sp3 C–H Bond

(2015) Shabber Mohammed et al.   JOURNAL OF ORGANIC CHEMISTRY

Recent developments in the chemistry of quinazolinone alkaloids

(2015) U. A. Kshirsagar   ORGANIC & BIOMOLECULAR CHEMISTRY

Cleavage of the C–C triple bond of ketoalkynes: synthesis of 4(3H)-quinazolinones

(2015) Xifa Yang et al.   Organic Chemistry Frontiers

Potassium Iodide-Catalyzed Three-Component Synthesis of 2-ArylquinazolinesviaAmination of Benzylic CH Bonds of Methylarenes

(2014) Dan Zhao et al.   ADVANCED SYNTHESIS & CATALYSIS

Di-tertButyl Peroxide-Promoted Sequential Methylation and Intramolecular Aromatization of Isonitriles

(2014) Qiang Dai et al.   ADVANCED SYNTHESIS & CATALYSIS

Metal-free oxidative synthesis of quinazolinones via dual amination of sp3 C–H bonds

(2014) Dan Zhao et al.   CHEMICAL COMMUNICATIONS

Mechanistic Study of a Complementary Reaction System that Easily Affords Quinazoline and Perimidine Derivatives

(2014) Zerong Daniel Wang et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

A convenient palladium-catalyzed carbonylative synthesis of 4(3H)-quinazolinones from 2-bromoformanilides and organo nitros with Mo(CO)6 as a multiple promoter

(2014) Lin He et al.   GREEN CHEMISTRY

Palladium-Catalyzed One-Pot Synthesis of Quinazolinones via tert-Butyl Isocyanide Insertion

(2014) Xiao Jiang et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis, Anti-microbial and Molecular Docking Studies of Quinazolin-4(3H)-one Derivatives

(2014) Yahia Mabkhot et al.   MOLECULES

Metal-free aerobic oxidative C–N bond cleavage of tertiary amines for the synthesis of N-heterocycles with high atom efficiency

(2014) Xiuling Chen et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Copper-Catalyzed Aerobic Oxidative Amination of sp3C–H Bonds: Efficient Synthesis of 2-Hetarylquinazolin-4(3H)-ones

(2014) Qiang Li et al.   ORGANIC LETTERS

Asymmetric Henry Reaction Catalyzed by a Chiral Dinuclear Nickel Complex

(2014) Hui Zhou et al.   SYNLETT

Iron-catalyzed decarboxylative methylation of α,β-unsaturated acids under ligand-free conditions

(2014) Guangwei Rong et al.   TETRAHEDRON

Synthesis of quinazolinones from anthranilamides and aldehydes via metal-free aerobic oxidation in DMSO

(2014) Na Yeun Kim et al.   TETRAHEDRON LETTERS

Copper-catalyzed tandem N-arylation/condensation: synthesis of quinazolin-4(3H)-ones from 2-halobenzonitriles and amides

(2014) Hongxin Chai et al.   RSC Advances

Palladium-Catalyzed Carbonylative Synthesis of Quinazolinones from 2-Aminobenzamide and Aryl Bromides

(2013) Xiao-Feng Wu et al.   CHEMISTRY-A EUROPEAN JOURNAL

Copper-Catalyzed Methyl Esterification Reactions via C–C Bond Cleavage

(2013) Yan Zhu et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-catalyzed methyl esterification of aromatic aldehydes and benzoic alcohols by TBHP as both oxidant and methyl source

(2013) Pan Li et al.   TETRAHEDRON LETTERS

Selective Iodine-Catalyzed Intermolecular Oxidative Amination of C(sp3)H Bonds with ortho-Carbonyl-Substituted Anilines to Give Quinazolines

(2012) Yizhe Yan et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

High-Temperature Measurements of the Reactions of OH with Small Methyl Esters: Methyl Formate, Methyl Acetate, Methyl Propanoate, and Methyl Butanoate

(2012) King-Yiu Lam et al.   JOURNAL OF PHYSICAL CHEMISTRY A

An efficient, greener, and solvent-free one-pot multicomponent synthesis of 3-substituted quinazolin-4(3H)ones and thienopyrimidin-4(3H)ones

(2012) Hitesh B. Jalani et al.   TETRAHEDRON LETTERS

Metal-free intramolecular oxidative decarboxylative amination of primary α-amino acids with product selectivity

(2011) Yizhe Yan et al.   CHEMICAL COMMUNICATIONS

Iodine Catalyzed One-pot Synthesis of 3,4-Dihydroquinazolin-4-ones from Anthranilic Acids, Ortho Esters and Amines under Solvent-free Conditions

(2008) Hong-She WANG et al.   CHINESE JOURNAL OF CHEMISTRY

Quinoline, quinazoline and acridonealkaloids

(2007) Joseph P. Michael   NATURAL PRODUCT REPORTS