Organocatalytic, enantioselective synthesis of benzoxaboroles via Wittig/oxa-Michael reaction Cascade of α-formyl boronic acids

Formulation of benzoxaborole drugs in PLLA: from materials preparation to in vitro release kinetics and cellular assays

(2016) Saad Sene et al.   Journal of Materials Chemistry B

Organocatalytic enantio- and diastereoselective synthesis of highly substituted δ-lactones via a Michael-cyclization cascade

(2015) Santosh Agrawal et al.   CHEMICAL COMMUNICATIONS

A Cu(ii)-based strategy for catalytic enantioselective β-borylation of α,β-unsaturated acceptors

(2015) Lei Zhu et al.   CHEMICAL COMMUNICATIONS

Recent Developments in the Chemistry and Biological Applications of Benzoxaboroles

(2015) Agnieszka Adamczyk-Woźniak et al.   CHEMICAL REVIEWS

Intercalation of Benzoxaborolate Anions in Layered Double Hydroxides: Toward Hybrid Formulations for Benzoxaborole Drugs

(2015) Saad Sene et al.   CHEMISTRY OF MATERIALS

Benzoxaborole Antimalarial Agents. Part 4. Discovery of Potent 6-(2-(Alkoxycarbonyl)pyrazinyl-5-oxy)-1,3-dihydro-1-hydroxy-2,1-benzoxaboroles

(2015) Yong-Kang Zhang et al.   JOURNAL OF MEDICINAL CHEMISTRY

Organocatalytic, Enantioselective Synthesis of 1- and 3-Substituted Isochromans via Intramolecular Oxa-Michael Reaction of Alkoxyboronate: Synthesis of (+)-Sonepiprazole

(2015) Barnala Ravindra et al.   JOURNAL OF ORGANIC CHEMISTRY

Chiral Brønsted Acid as a True Catalyst: Asymmetric Mukaiyama Aldol and Hosomi–Sakurai Allylation Reactions

(2015) Masahiro Sai et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Highly enantioselective synthesis of naphthoquinones and pyranonaphthoquinones catalyzed by bifunctional chiral bis-squaramides

(2015) Nagaraju Molleti et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Catalytic Aldol–Cyclization Cascade of 3-Isothiocyanato Oxindoles with α-Ketophosphonates for the Enantioselective Synthesis of β-Amino-α-hydroxyphosphonates

(2015) Satavisha Kayal et al.   ORGANIC LETTERS

Inhibiting the β-Lactamase of Mycobacterium tuberculosis (Mtb) with Novel Boronic Acid Transition-State Inhibitors (BATSIs)

(2015) Sebastian G. Kurz et al.   ACS Infectious Diseases

4,5-Disubstituted 6-Aryloxy-1,3-dihydrobenzo[c][1,2]oxaboroles Are Broad-Spectrum Serine β-Lactamase Inhibitors

(2015) David C. McKinney et al.   ACS Infectious Diseases

ansa-Ruthenium(II) Complexes of DPEN-SO2N(Me)(CH2)n(η6-aryl) Conjugate Ligands for Asymmetric Transfer Hydrogenation of Aryl Ketones

(2014) Andrea Kišić et al.   ADVANCED SYNTHESIS & CATALYSIS

The unique chemistry of benzoxaboroles: Current and emerging applications in biotechnology and therapeutic treatments

(2014) C. Tony Liu et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Electrochemical displacement sensor based on ferrocene boronic acid tracer and immobilized glycan for saccharide binding proteins and E. coli

(2014) Decha Dechtrirat et al.   BIOSENSORS & BIOELECTRONICS

Organocatalytic, Enantioselective, Intramolecular Oxa-Michael Reaction of Alkoxyboronate: A New Strategy for Enantioenriched 1-Substituted 1,3-Dihydroisobenzofurans

(2014) Barnala Ravindra et al.   ORGANIC LETTERS

Structure–activity relationships of 6-(aminomethylphenoxy)-benzoxaborole derivatives as anti-inflammatory agent

(2013) Tsutomu Akama et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Biomolecular robotics for chemomechanically driven guest delivery fuelled by intracellular ATP

(2013) Shuvendu Biswas et al.   Nature Chemistry

Asymmetric chroman synthesis via an intramolecular oxy-Michael addition by bifunctional organocatalysts

(2013) Ryota Miyaji et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Benzoboroxole-Functionalized Magnetic Core/Shell Microspheres for Highly Specific Enrichment of Glycoproteins under Physiological Conditions

(2013) Yuting Zhang et al.   Small

Temperature, pH, and Glucose Responsive Gels via Simple Mixing of Boroxole- and Glyco-Based Polymers

(2013) Yohei Kotsuchibashi et al.   ACS Macro Letters

Asymmetric Boron Conjugate Additions to Enones in Water Catalyzed by Copper(0)

(2013) Taku Kitanosono et al.   Asian Journal of Organic Chemistry

Boron-based phosphodiesterase inhibitors show novel binding of boron to PDE4 bimetal center

(2012) Yvonne R. Freund et al.   FEBS LETTERS

Boronate-Mediated Biologic Delivery

(2012) Gregory A. Ellis et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Monosaccharide-Responsive Release of Insulin from Polymersomes of Polyboroxole Block Copolymers at Neutral pH

(2012) Hyunkyu Kim et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

pH-Independent Transfer Hydrogenation in Water: Catalytic, Enantioselective Reduction of β-Keto Esters

(2012) Martin A. Ariger et al.   ORGANIC LETTERS

Application of a novel 1,3-diol with a benzyl backbone as chiral ligand for asymmetric oxidation of sulfides to sulfoxides

(2012) Paramartha Gogoi et al.   TETRAHEDRON LETTERS

Directed ortho,ortho'-dimetalation of hydrobenzoin: Rapid access to hydrobenzoin derivatives useful for asymmetric synthesis

(2011) Inhee Cho et al.   Beilstein Journal of Organic Chemistry

Synthesis and SAR of acyclic HCV NS3 protease inhibitors with novel P4-benzoxaborole moieties

(2011) Xianfeng Li et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis and SAR of novel benzoxaboroles as a new class of β-lactamase inhibitors

(2011) Yi Xia et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Boron-containing inhibitors of synthetases

(2011) Stephen J. Baker et al.   CHEMICAL SOCIETY REVIEWS

Enantioselective Double Aldol Reaction Catalyzed by Chiral Phosphine Oxide

(2011) Yasushi Shimoda et al.   CHEMISTRY-A EUROPEAN JOURNAL

Benzoxaboroles: a new class of potential drugs for human African trypanosomiasis

(2011) Robert T Jacobs et al.   Future Medicinal Chemistry

Asymmetric Catalytic Cycloetherification Mediated by Bifunctional Organocatalysts

(2011) Keisuke Asano et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

SCYX-7158, an Orally-Active Benzoxaborole for the Treatment of Stage 2 Human African Trypanosomiasis

(2011) Robert T. Jacobs et al.   PLoS Neglected Tropical Diseases

Boronic Acid-Based Lectin Mimics (Boronolectins) That Can Recognize Cancer Biomarker, the Thomsen-Friedenrich Antigen

(2010) Sarah Burroughs et al.   CHEMBIOCHEM

Developing High-Affinity Boron-Based Receptors for Cell-Surface Carbohydrates

(2010) Todd A. Houston   CHEMBIOCHEM

Enhanced gene transfection capability of polyethylenimine by incorporating boronic acid groups

(2010) Qi Peng et al.   CHEMICAL COMMUNICATIONS

Privileged scaffolds for library design and drug discovery

(2010) Matthew E Welsch et al.   CURRENT OPINION IN CHEMICAL BIOLOGY

Influence of the Substituents on the Structure and Properties of Benzoxaboroles

(2010) Agnieszka Adamczyk-Woźniak et al.   JOURNAL OF PHYSICAL CHEMISTRY A

The stereodivergent asymmetric synthesis of a range of 2-(1′-hydroxyalkyl)phenols

(2010) Stephen G. Davies et al.   TETRAHEDRON

Discovery and structure–activity study of a novel benzoxaborole anti-inflammatory agent (AN2728) for the potential topical treatment of psoriasis and atopic dermatitis

(2009) Tsutomu Akama et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Direct Catalytic Asymmetric Synthesis of Highly Functionalized 2-Methylchroman-2,4-diols via Barbas-List Aldol Reaction

(2009) Dhevalapally B. Ramachary et al.   CHEMISTRY-A EUROPEAN JOURNAL

Crystal Structures of the Human and Fungal Cytosolic Leucyl-tRNA Synthetase Editing Domains: A Structural Basis for the Rational Design of Antifungal Benzoxaboroles

(2009) Elena Seiradake et al.   JOURNAL OF MOLECULAR BIOLOGY

Benzoxaboroles – Old compounds with new applications

(2009) Agnieszka Adamczyk-Woźniak et al.   JOURNAL OF ORGANOMETALLIC CHEMISTRY

Noninvasive Sialic Acid Detection at Cell Membrane by Using Phenylboronic Acid Modified Self-Assembled Monolayer Gold Electrode

(2009) Akira Matsumoto et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Bidirectional Metalation of Hydrobenzoin: Direct Access to New Chiral Ligands and Auxiliaries

(2009) Inhee Cho et al.   ORGANIC LETTERS

Benzoboroxoles as Efficient Glycopyranoside-Binding Agents in Physiological Conditions: Structure and Selectivity of Complex Formation

(2008) Marie Bérubé et al.   JOURNAL OF ORGANIC CHEMISTRY

Chiral Squaramide Derivatives are Excellent Hydrogen Bond Donor Catalysts

(2008) Jeremiah P. Malerich et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Enantioselective, Organocatalytic Oxy-Michael Addition to γ/δ-Hydroxy-α,β-enones:  Boronate-Amine Complexes as Chiral Hydroxide Synthons

(2007) De Run Li et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY