Synthesis, larvicidal efficiency and molecular docking studies of novel annulated pyrano[2,3-c]pyrazoles against Culex pipiens L. and Musca domestica L. larvae

Design and Synthesis of New Quinoline Linked to Pyranotriazolopyrimidines Conjugates as Novel Targets to Discover Promising Anti-SARS-COV-2

(2022) Hichem Ben Jannet et al.   HETEROCYCLES

The Binary Mixtures of Lambda-Cyhalothrin, Chlorfenapyr, and Abamectin, against the House Fly Larvae, Musca domestica L.

(2022) Doaa F. El Sherif et al.   MOLECULES

A Practical Insecticide Resistance Monitoring Bioassay for Orally Ingested Dinotefuran in Anopheles Malaria Vectors

(2022) George John Ian Parsons et al.   Insects

Larvicidal Activity of Pentagalloyl Glucose and Mangiferin Isolated from the Waste of Mango Kernel Against Culex pipiens L.

(2021) Mahmoud Emam et al.   Waste and Biomass Valorization

Design, Synthesis, and Biological Evaluation of Densely Substituted Dihydropyrano[2,3-c]pyrazoles via a Taurine-Catalyzed Green Multicomponent Approach

(2021) Ghanshyam Mali et al.   ACS Omega

1,2,4-Triazolo[1,5-a]pyrimidines as a Novel Class of Inhibitors of the HIV-1 Reverse Transcriptase-Associated Ribonuclease H Activity

(2020) Jenny Desantis et al.   MOLECULES

Design, synthesis, anti-proliferative activity, and molecular docking studies of novel benzo[f]chromene, chromeno [2,3-d]pyrimidines and chromenotriazolo[1,5-c]pyrimidines

(2020) Fatma S. M. Abu El-Azm et al.   SYNTHETIC COMMUNICATIONS

Novel Anticancer Fused Pyrazole Derivatives as EGFR and VEGFR-2 Dual TK Inhibitors

(2020) Nashwa M. Saleh et al.   Frontiers in Chemistry

Design, synthesis, and biological evaluation of piperidinyl‐substituted [1,2,4]triazolo[1,5‐a]pyrimidine derivatives as potential anti‐HIV‐1 agents with reduced cytotoxicity

(2020) Boshi Huang et al.   Chemical Biology & Drug Design

Synthesis and Antimicrobial Evaluation of Some Novel Pyrimidine, Pyrazole, Chromene and Tetrahydrobenzo[b]thiophene Derivatives Bearing Pyrimidinthione Moiety

(2020) Mohamed Ahmed Mahmoud Abdel Reheim et al.   CURRENT ORGANIC SYNTHESIS

Utilization of cyanoacetohydrazide and 2-(1,3-dioxoisoindolin-2-yl) acetyl chloride in the synthesis of some novel anti-proliferative heterocyclic compounds

(2020) Mohamed H. Hekal et al.   SYNTHETIC COMMUNICATIONS

Binding properties to nicotinic acetylcholine receptors can explain differential toxicity of neonicotinoid insecticides in Chironomidae

(2020) E.M. Maloney et al.   AQUATIC TOXICOLOGY

Using targeted next-generation sequencing to characterize genetic differences associated with insecticide resistance in Culex quinquefasciatus populations from the southern U.S.

(2019) Linda Kothera et al.   PLoS One

Ecofriendly and highly efficient microwave-induced synthesis of novel quinazolinone-undecyl hybrids with in vitro antitumor activity

(2019) Mohamed H. Hekal et al.   SYNTHETIC COMMUNICATIONS

Identification of Novel 3-Hydroxy-pyran-4-One Derivatives as Potent HIV-1 Integrase Inhibitors Using in silico Structure-Based Combinatorial Library Design Approach

(2019) Hajar Sirous et al.   Frontiers in Chemistry

Efficacy and repellency of some essential oils and their blends against larval and adult house flies, Musca domestica L. (Diptera: Muscidae)

(2019) Hanem F. Khater et al.   JOURNAL OF VECTOR ECOLOGY

A cascade synthesis, in vitro cholinesterases inhibitory activity and docking studies of novel Tacrine-pyranopyrazole derivatives

(2018) Chamseddine Derabli et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Synthesis, Anticancer Screening and Molecular Docking Studies of New Heterocycles with Trimethoxyphenyl Scaffold as Combretastatin Analogues

(2018) Korany A. Ali et al.   MINI-REVIEWS IN MEDICINAL CHEMISTRY

Synthesis and antitumor evaluation of novel tetrahydrobenzo[4′,5′]thieno[3′,2′:5,6]pyrimido[1,2-b]isoquinoline derivatives

(2018) Mahmoud R. Mahmoud et al.   SYNTHETIC COMMUNICATIONS

Host Selection by Culex pipiens Mosquitoes and West Nile Virus Amplification

(2018) Gabriel L. Hamer et al.   AMERICAN JOURNAL OF TROPICAL MEDICINE AND HYGIENE

Pyranopyrazoles as efficient antimicrobial agents: Green, one pot and multicomponent approach

(2018) Guda Mallikarjuna Reddy et al.   BIOORGANIC CHEMISTRY

An efficient and green approach: One pot, multi component, reusable catalyzed synthesis of pyranopyrazoles and investigation of biological assays

(2018) Guda Mallikarjuna Reddy et al.   Journal of Saudi Chemical Society

Rift Valley fever virus and European mosquitoes: vector competence of Culex pipiens and Stegomyia albopicta (= Aedes albopictus )

(2017) M. BRUSTOLIN et al.   MEDICAL AND VETERINARY ENTOMOLOGY

Design of New Benzo[h]chromene Derivatives: Antitumor Activities and Structure-Activity Relationships of the 2,3-Positions and Fused Rings at the 2,3-Positions

(2017) Rawda Okasha et al.   MOLECULES

Synthesis and antimicrobial evaluation of some novel dithiolane, thiophene, coumarin, and 2-pyridone derivatives

(2017) Mahmoud R. Mahmoud et al.   SYNTHETIC COMMUNICATIONS

Uncatalyzed four-component synthesis of pyrazolopyranopyrimidine derivatives and their antituberculosis activities

(2016) Kirti T. Patil et al.   SYNTHETIC COMMUNICATIONS

Synthesis of functionalized pyrazolopyran derivatives: comparison of two-step vs. one-step vs. microwave-assisted protocol and X-ray crystallographic analysis of 6-amino-1,4-dihydro-3-methyl-4-phenylpyrano[2,3-c]pyrazole-5-carbonitrile

(2015) PARITOSH SHUKLA et al.   BULLETIN OF MATERIALS SCIENCE

Efficacy of granular applications of clothianidin and nitenpyram against Aphis gossypii (Glover) and Apolygus lucorum (Meyer-Dür) in cotton fields in China

(2015) Peng Zhang et al.   CROP PROTECTION

Synthesis and Insecticidal Efficacy of Novel Bis Quinazolinone Derivatives

(2015) Manal M. Elshahawi et al.   JOURNAL OF HETEROCYCLIC CHEMISTRY

Xenomonitoring of Different Filarial Nematodes Using Single and Multiplex PCR in Mosquitoes from Assiut Governorate, Egypt

(2015) Ahmed Kamal Dyab et al.   KOREAN JOURNAL OF PARASITOLOGY

4-([1,2,4]Triazolo[1,5-a]pyridin-6-yl)-5(3)-(6-methylpyridin-2-yl)imidazole and -pyrazole derivatives as potent and selective inhibitors of transforming growth factor-β type I receptor kinase

(2014) Cheng Hua Jin et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis, in vitro antimicrobial and cytotoxic activities of novel pyrimidine–benzimidazol combinations

(2014) Peng-Ju Chen et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Initial Synthesis of Diastereomeric Pyran Spirooxoindolinones Based on (–)-Carvone and (+)-3-Carene

(2014) F. Z. Macaev et al.   CHEMISTRY OF NATURAL COMPOUNDS

Design, synthesis and bioevaluation of N-trisubstituted pyrimidine derivatives as potent aurora A kinase inhibitors

(2014) Yu Luo et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Design, synthesis and molecular modeling of pyrazole–quinoline–pyridine hybrids as a new class of antimicrobial and anticancer agents

(2014) Chetan B. Sangani et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Structure Based Design, Synthesis, Pharmacophore Modeling, Virtual Screening, and Molecular Docking Studies for Identification of Novel Cyclophilin D Inhibitors

(2014) Koteswara Rao Valasani et al.   Journal of Chemical Information and Modeling

An efficient and eco-friendly synthesis and evaluation of antibactrial activity of pyrano[2,3-c]pyrazole derivatives

(2014) Manouchehr Mamaghani et al.   MEDICINAL CHEMISTRY RESEARCH

A synthetic compound, 4-acetyl-3-methyl-6-(3,4,5-trimethoxyphenyl)pyrano[3,4-c]pyran-1,8-dione, ameliorates ovalbumin-induced asthma

(2013) Hwan-Suck Chung et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis and Biological Activities of Some New Annulated Pyrazolopyranopyrimidines and Their Derivatives Containing Indole Nucleus

(2013) Anand R. Saundane et al.   JOURNAL OF HETEROCYCLIC CHEMISTRY

Antiplatelet therapy: new pharmacological agents and changing paradigms

(2013) D. Capodanno et al.   JOURNAL OF THROMBOSIS AND HAEMOSTASIS

Insecticide Mixtures Could Enhance the Toxicity of Insecticides in a Resistant Dairy Population of Musca domestica L

(2013) Hafiz Azhar Ali Khan et al.   PLoS One

Synthesis and potential biological activity of some novel 3-[(N-substituted indol-3-yl)methyleneamino]-6-amino-4-aryl-pyrano(2,3-c)pyrazole-5-carbonitriles and 3,6-diamino-4-(N-substituted indol-3-yl)pyrano(2,3-c)pyrazole-5-carbonitriles

(2012) Adel Mandour et al.   ACTA PHARMACEUTICA

Eco-friendly synthesis and biological evaluation of substituted pyrano[2,3-c]pyrazoles

(2012) Santhosh Reddy Mandha et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Variability in docking success rates due to dataset preparation

(2012) Christopher R. Corbeil et al.   JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN

Trifluoroacetyl Neonicotinoid Insecticides with Enhanced Hydrophobicity and Effectiveness

(2010) Ikuya Ohno et al.   JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY

Computer-Aided Drug Design of Pyranopyrazoles and Related Compounds for Checkpoint Kinase-1

(2009) Rahul Ramtekkar et al.   Letters in Drug Design & Discovery

Crystal structures of Lymnaea stagnalis AChBP in complex with neonicotinoid insecticides imidacloprid and clothianidin

(2008) Makoto Ihara et al.   INVERTEBRATE NEUROSCIENCE

Neonicotinoids-from zero to hero in insecticide chemistry

(2008) Peter Jeschke et al.   PEST MANAGEMENT SCIENCE

Flea blood feeding patterns in cats treated with oral nitenpyram and the topical insecticides imidacloprid, fipronil and selamectin

(2008) C. McCoy et al.   VETERINARY PARASITOLOGY