De Novo Construction of Chiral Aminoindolines by Cu-Catalyzed Asymmetric Cyclization and Subsequent Discovery of an Unexpected Sulfonyl Migration

Synthesis of Chiral Endocyclic Allenes by Palladium‐Catalyzed Asymmetric Annulation Followed by Cope Rearrangement

(2022) Bin Shi et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Propargylic Amination Enabled the Access to Enantioenriched Acyclic α-Quaternary α-Amino Ketones

(2021) Wusheng Guo et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Silver‐Catalyzed Asymmetric Dearomatization of Electron‐Deficient Heteroarenes via Interrupted Barton–Zard Reaction

(2021) Qian Wan et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

How do we address neglected sulfur pharmacophores in drug discovery?

(2021) Michael J. Tilby et al.   Expert Opinion on Drug Discovery

Synthesis and Pharmacological Evaluation of Tetrahydro-γ-carboline Derivatives as Potent Anti-inflammatory Agents Targeting Cyclic GMP–AMP Synthase

(2021) Jing Tan et al.   JOURNAL OF MEDICINAL CHEMISTRY

Electrooxidation enables selective dehydrogenative [4+2] annulation between indole derivatives

(2020) Chunlan Song et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Palladium‐Catalyzed Asymmetric [8+2] Dipolar Cycloadditions of Vinyl Carbamates and Photogenerated Ketenes

(2020) Liang-Qiu Lu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Asymmetric Coupling of Carbon‐Centered Radical Adjacent to Nitrogen: Copper‐Catalyzed Cyanation and Etherification of Enamides

(2020) Guosheng Liu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Electrochemical Dearomative 2,3-Difunctionalization of Indoles

(2019) Ju Wu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Enantioselective A3-Coupling Reaction Employing Chiral CuI-iPrpyboxdiPh/N-Boc-(l)-Proline Complex under Cooperative Catalysis: Application in the Synthesis of (Indol-2-yl)methanamines

(2019) Sivasankaran Dhanasekaran et al.   JOURNAL OF ORGANIC CHEMISTRY

Transition Metal Vinylidene- and Allenylidene-Mediated Catalysis in Organic Synthesis

(2019) Sang Weon Roh et al.   CHEMICAL REVIEWS

Phosphine-Catalyzed Enantioselective Dearomative [3+2]-Cycloaddition of 3-Nitroindoles and 2-Nitrobenzofurans

(2019) Huamin Wang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Dearomatization of 3-Nitroindoles by a Phosphine-Catalyzed Enantioselective [3+2] Annulation Reaction

(2019) Kaizhi Li et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Indole Alkaloid Synthesis Facilitated by Photoredox Catalytic Radical Cascade Reactions

(2019) Xiao-Yu Liu et al.   ACCOUNTS OF CHEMICAL RESEARCH

Exploration of Novel Chiral Cobalt Catalyst for Visible-Light-Induced Enantioselective Radical Conjugate Addition

(2019) Wen-Jing Xiao et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Organocatalytic Asymmetric Synthesis of Indole-Based Chiral Heterocycles: Strategies, Reactions, and Outreach

(2019) Yu-Chen Zhang et al.   ACCOUNTS OF CHEMICAL RESEARCH

Stereodivergent Synthesis of Tetrahydrofuroindoles through Pd-Catalyzed Asymmetric Dearomative Formal [3+2] Cycloaddition

(2018) Qiang Cheng et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Transition-Metal-Free Decarboxylative Propargylic Substitution/Cyclization with either Azolium Enolates or Acyl Anions

(2018) Shenci Lu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Polycyclic Indoline-Benzodiazepines through Electrophilic Additions of α-Imino Carbenes to Tröger Bases

(2018) Alessandro Bosmani et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Manganese(I)-Catalyzed C−H (2-Indolyl)methylation: Expedient Access to Diheteroarylmethanes

(2018) Qingquan Lu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Divergent Strategy in Natural Product Total Synthesis

(2018) Lei Li et al.   CHEMICAL REVIEWS

Recent advances in spirocyclization of indole derivatives

(2018) Jitender Bariwal et al.   CHEMICAL SOCIETY REVIEWS

Catalytic Asymmetric Dearomative [3 + 2] Cycloaddition of Electron-Deficient Indoles with All-Carbon 1,3-Dipoles

(2018) Meng Sun et al.   JOURNAL OF ORGANIC CHEMISTRY

Pd-Catalyzed Asymmetric Dearomative Cycloaddition for Construction of Optically Active Pyrroloindoline and Cyclopentaindoline Derivatives: Access to 3a-Aminopyrroloindolines

(2018) Jun-Qi Zhang et al.   JOURNAL OF ORGANIC CHEMISTRY

Metamorphosis of cycloalkenes for the divergent total synthesis of polycyclic indole alkaloids

(2018) Zhengren Xu et al.   CHEMICAL SOCIETY REVIEWS

Stereocontrolled Synthesis of 1,4-Dicarbonyl Compounds by Photochemical Organocatalytic Acyl Radical Addition to Enals

(2018) Giulio Goti et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Enantioselective Trapping of Pd-Containing 1,5-Dipoles by Photogenerated Ketenes: Access to 7-Membered Lactones Bearing Chiral Quaternary Stereocenters

(2018) Yi Wei et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Sequential Visible-Light Photoactivation and Palladium Catalysis Enabling Enantioselective [4+2] Cycloadditions

(2017) Miao-Miao Li et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

N- to C-sulfonyl photoisomerisation of dihydropyridinones: a synthetic and mechanistic study

(2017) Pei-Pei Yeh et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Incorporation of Axial Chirality into Phosphino-Imidazoline Ligands for Enantioselective Catalysis

(2017) Paulo H. S. Paioti et al.   ACS Catalysis

Catalytic Enantioselective Synthesis of Amino Skipped Diynes

(2016) Paulo H. S. Paioti et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Catalytic Asymmetric [4 + 1] Annulation of Sulfur Ylides with Copper–Allenylidene Intermediates

(2016) Qiang Wang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Enantioselective dearomative [3 + 2] cycloadditions of indoles with azomethine ylides derived from alanine imino esters

(2016) Anthony L. Gerten et al.   Organic Chemistry Frontiers

Intramolecular Dearomative Oxidative Coupling of Indoles: A Unified Strategy for the Total Synthesis of Indoline Alkaloids

(2015) Weiwei Zi et al.   ACCOUNTS OF CHEMICAL RESEARCH

Asymmetric Brønsted Acid Catalyzed Synthesis of Triarylmethanes-Construction of Communesin and Spiroindoline Scaffolds

(2015) Hsuan-Hung Liao et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Gold-Catalyzed Cascade Cyclization of 2-Alkynyl-N-Propargylanilines by Rearrangement of a Propargyl Group

(2015) Yusuke Tokimizu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Asymmetric Michael/Cyclization Cascade Reaction of 3-Isothiocyanato Oxindoles and 3-Nitroindoles with Amino-Thiocarbamate Catalysts: Enantioselective Synthesis of Polycyclic Spirooxindoles

(2015) Jian-Qiang Zhao et al.   ORGANIC LETTERS

PyBidine/Copper Catalyst: Asymmetricexo′-Selective [3+2] Cycloaddition using Imino Ester and Electrophilic Indole

(2014) Atsuko Awata et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Palladium-Catalyzed Dearomative Trimethylenemethane Cycloaddition Reactions

(2014) Barry M. Trost et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Copper-Catalyzed Oxoazidation and Alkoxyazidation of Indoles

(2014) Hang Yin et al.   ORGANIC LETTERS

Iron(II)-Catalyzed Asymmetric Intramolecular Aminohydroxylation of Indoles

(2013) Yong-Qiang Zhang et al.   ORGANIC LETTERS

Synthetic Studies on Chartelline C: Stereoselective Construction of the Core Skeleton

(2012) Kotaro Iwasaki et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Efficient and General Synthesis of 3-Aminoindolines and 3-Aminoindoles via Copper-Catalyzed Three-Component Coupling Reaction

(2010) Dmitri Chernyak et al.   ADVANCED SYNTHESIS & CATALYSIS

Oxaziridine-Mediated Oxyamination of Indoles: An Approach to 3-Aminoindoles and Enantiomerically Enriched 3-Aminopyrroloindolines

(2010) Tamas Benkovics et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Total Synthesis of (−)-Mersicarpine

(2010) Rie Nakajima et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Highly enantioselective intramolecular aza-spiroannulation onto indoles using chiral rhodium catalysis: asymmetric entry to the spiro-β-lactam core of chartellines

(2009) Shigeki Sato et al.   CHEMICAL COMMUNICATIONS

Advances in Solution- and Solid-Phase Synthesis toward the Generation of Natural Product-like Libraries

(2009) Jyoti P. Nandy et al.   CHEMICAL REVIEWS

Discovery of Indoline-Based, Natural-Product-like Compounds as Probes of Focal Adhesion Kinase Signaling Pathways

(2009) Rajamohan R. Poondra et al.   JOURNAL OF COMBINATORIAL CHEMISTRY

An Expedient Route to a Potent Gastrin/CCK-B Receptor Antagonist (+)-AG-041R

(2009) Shigeki Sato et al.   JOURNAL OF ORGANIC CHEMISTRY

Enantiospecific Total Syntheses of Kapakahines B and F

(2009) Timothy Newhouse et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Enantioselective Copper-Catalyzed Propargylic Amination

(2008) Remko J. Detz et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Copper-Catalyzed Asymmetric Propargylic Substitution Reactions of Propargylic Acetates with Amines

(2008) Gaku Hattori et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

An Expeditious Synthesis of C(3)−N(1′) Heterodimeric Indolines

(2008) Vinson R. Espejo et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Total Synthesis of (±)-Psychotrimine

(2008) Timothy Newhouse et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Total Synthesis of (±)-Mersicarpine

(2008) Jakob Magolan et al.   ORGANIC LETTERS