Design, synthesis, and biological activity of novel dithiocarbamate‐methylsulfonyl hybrids as carbonic anhydrase inhibitors
Published 2022 View Full Article
- Home
- Publications
- Publication Search
- Publication Details
Title
Design, synthesis, and biological activity of novel dithiocarbamate‐methylsulfonyl hybrids as carbonic anhydrase inhibitors
Authors
Keywords
-
Journal
ARCHIV DER PHARMAZIE
Volume -, Issue -, Pages -
Publisher
Wiley
Online
2022-05-03
DOI
10.1002/ardp.202200132
References
Ask authors/readers for more resources
Related references
Note: Only part of the references are listed.- Discovery of a novel series of indolylchalcone-benzenesulfonamide hybrids acting as selective carbonic anhydrase II inhibitors
- (2021) Priti Singh et al. BIOORGANIC CHEMISTRY
- Comprehensive research on potent and selective carbonic anhydrase inhibitors: Synthesis, bioactivities and molecular modelling studies of 4-(3-(2-arylidenehydrazine-1-carbonyl)-5-(thiophen-2-yl)-1H-pyrazole-1-yl) benzenesulfonamides
- (2021) Cem Yamali et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Design and synthesis of benzenesulfonamide‐linked imidazo[2,1‐ b ][1,3,4]thiadiazole derivatives as carbonic anhydrase I and II inhibitors
- (2021) Baijayantimala Swain et al. ARCHIV DER PHARMAZIE
- Quinoline-sulfamoyl carbamates/sulfamide derivatives: Synthesis, cytotoxicity, carbonic anhydrase activity, and molecular modelling studies
- (2021) Elmas Begum Cakmak et al. BIOORGANIC CHEMISTRY
- Novel inhibitors with sulfamethazine backbone: synthesis and biological study of multi-target cholinesterases and α-glucosidase inhibitors
- (2021) Cüneyt Türkeş et al. JOURNAL OF BIOMOLECULAR STRUCTURE & DYNAMICS
- Developments of small molecules as inhibitors for carbonic anhydrase isoforms
- (2021) Emmanuel Ramsey Buabeng et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Novel triazole-sulfonamide bearing pyrimidine moieties with carbonic anhydrase inhibitory action: Design, synthesis, computational and enzyme inhibition studies
- (2021) Shoaib Manzoor et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Design, synthesis, characterization, in vitro and in silico evaluation of novel imidazo[2,1-b][1,3,4]thiadiazoles as highly potent acetylcholinesterase and non-classical carbonic anhydrase inhibitors
- (2021) Sercan Askin et al. BIOORGANIC CHEMISTRY
- Inhibition studies on carbonic anhydrase isoforms I, II, IV and IX with N-arylsubstituted secondary sulfonamides featuring a bicyclic tetrahydroindazole scaffold
- (2021) Silvia Salerno et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Transition‐Metal Complexes of Bidentate Schiff‐Base Ligands: In Vitro and In Silico Evaluation as Non‐Classical Carbonic Anhydrase and Potential Acetylcholinesterase Inhibitors
- (2021) Ümit Yaşar et al. ChemistrySelect
- Synthesis and Human Carbonic Anhydrase I, II, IX, and XII Inhibition Studies of Sulphonamides Incorporating Mono-, Bi- and Tricyclic Imide Moieties
- (2021) Kalyan Sethi et al. Pharmaceuticals
- Novel benzenesulfonamides aryl and arylsulfone conjugates adopting tail/dual tail approaches: Synthesis, carbonic anhydrase inhibitory activity and molecular modeling studies
- (2021) Assem H. Eldeeb et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Calcium Channel Blockers: Molecular Docking and Inhibition Studies on Carbonic Anhydrase I and II Isoenzymes
- (2020) Cüneyt Türkeş et al. JOURNAL OF BIOMOLECULAR STRUCTURE & DYNAMICS
- Sulfonamides incorporating ketene N,S -acetal bioisosteres as potent carbonic anhydrase and acetylcholinesterase inhibitors
- (2020) Qëndresa Istrefi et al. ARCHIV DER PHARMAZIE
- Naphthoquinones, benzoquinones, and anthraquinones: Molecular docking, ADME and inhibition studies on human serum paraoxonase-1 associated with cardiovascular diseases
- (2020) Yeliz Demir DRUG DEVELOPMENT RESEARCH
- Synthesis, characterization, biological evaluation, and in silico studies of novel 1,3‐diaryltriazene‐substituted sulfathiazole derivatives
- (2020) Mesut Işık et al. ARCHIV DER PHARMAZIE
- Synthesis and carbonic anhydrase inhibition studies of sulfonamide based indole-1,2,3-triazole chalcone hybrids
- (2020) Priti Singh et al. BIOORGANIC CHEMISTRY
- Synthesis, characterization, inhibition effects, and molecular docking studies as acetylcholinesterase, α-glycosidase, and carbonic anhydrase inhibitors of novel benzenesulfonamides incorporating 1,3,5-triazine structural motifs
- (2020) Nebih Lolak et al. BIOORGANIC CHEMISTRY
- New chalcone derivatives having pyrazole and sulfonamide pharmacophores as carbonic anhydrase inhibitors
- (2020) Mehtap Tugrak et al. Letters in Drug Design & Discovery
- 3-Methylthiazolo[3,2-a]benzimidazole-benzenesulfonamide conjugates as novel carbonic anhydrase inhibitors endowed with anticancer activity: Design, synthesis, biological and molecular modeling studies
- (2020) Abdulsalam A.M. Alkhaldi et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Gadolinium-based contrast agents: in vitro paraoxonase 1 inhibition, in silico studies
- (2019) Şükrü Beydemir et al. DRUG AND CHEMICAL TOXICOLOGY
- A potential risk factor for paraoxonase 1: in silico and in‐vitro analysis of the biological activity of proton‐pump inhibitors
- (2019) Cüneyt Türkeş JOURNAL OF PHARMACY AND PHARMACOLOGY
- Synthesis, biological evaluation and in silico studies of novel N-substituted phthalazine sulfonamide compounds as potent carbonic anhydrase and acetylcholinesterase inhibitors
- (2019) Cüneyt Türkeş et al. BIOORGANIC CHEMISTRY
- Synthesis and evaluation of 4-(1,3,4-oxadiazol-2-yl)-benzenesulfonamides as potent carbonic anhydrase inhibitors
- (2019) Chaofu Yang et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Synthesis of coumarin-sulfonamide derivatives and determination of their cytotoxicity, carbonic anhydrase inhibitory and molecular docking studies
- (2019) Belma Zengin Kurt et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- New Isoindole‐1,3‐dione Substituted Sulfonamides as Potent Inhibitors of Carbonic Anhydrase and Acetylcholinesterase: Design, Synthesis, and Biological Evaluation
- (2019) Saliha Gündoğdu et al. ChemistrySelect
- Dithiocarbamates with potent inhibitory activity against theSaccharomyces cerevisiaeβ-carbonic anhydrase
- (2015) Murat Bozdag et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- In silico applications of bioisosterism in contemporary medicinal chemistry practice
- (2013) George Papadatos et al. Wiley Interdisciplinary Reviews-Computational Molecular Science
- More effective dithiocarbamate derivatives inhibiting carbonic anhydrases, generated by QSAR and computational design
- (2012) Speranta Avram et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- Dithiocarbamates Strongly Inhibit Carbonic Anhydrases and Show Antiglaucoma Action in Vivo
- (2012) Fabrizio Carta et al. JOURNAL OF MEDICINAL CHEMISTRY
- Dithiocarbamates are strong inhibitors of the beta-class fungal carbonic anhydrases from Cryptococcus neoformans, Candida albicans and Candida glabrata
- (2011) Simona Maria Monti et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Dithiocarbamates: a new class of carbonic anhydrase inhibitors. Crystallographic and kinetic investigations
- (2011) Fabrizio Carta et al. CHEMICAL COMMUNICATIONS
- Dithiocarbamates strongly inhibit the β-class carbonic anhydrases fromMycobacterium tuberculosis
- (2011) Alfonso Maresca et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- Carbonic anhydrase inhibitors. Inhibition of transmembrane isoforms IX, XII, and XIV with less investigated anions including trithiocarbonate and dithiocarbamate
- (2010) Alessio Innocenti et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Potent inhibitory effects of benzyl andp-xylidine-bis dithiocarbamate sodium salts on activities of mushroom tyrosinase
- (2010) E. Amin et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
- High-resolution structure of human carbonic anhydrase II complexed with acetazolamide reveals insights into inhibitor drug design
- (2009) Katherine H. Sippel et al. Acta Crystallographica Section F-Structural Biology and Crystallization Communications
Publish scientific posters with Peeref
Peeref publishes scientific posters from all research disciplines. Our Diamond Open Access policy means free access to content and no publication fees for authors.
Learn MoreCreate your own webinar
Interested in hosting your own webinar? Check the schedule and propose your idea to the Peeref Content Team.
Create Now