Metal-, Photocatalyst-, and Light-Free Minisci C–H Acetylation of N-Heteroarenes with Vinyl Ethers

Photoredox‐Catalyzed Redox‐Neutral Minisci C−H Formylation of N ‐Heteroarenes

(2020) Jianyang Dong et al.   ADVANCED SYNTHESIS & CATALYSIS

Iron-catalyzed Minisci acylation of N-heteroarenes with α-keto acids

(2019) Xiu-Zhi Wang et al.   TETRAHEDRON

Iron-Catalyzed Minisci Type Acetylation of N -Heteroarenes Mediated by CH(OEt)3 /TBHP

(2019) A. Srinivasulu et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Recent Advances in Minisci-Type Reactions

(2019) Rupert S. J. Proctor et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Visible-Light-Mediated Direct Decarboxylative Acylation of Electron-Deficient Heteroarenes Using α-Ketoacids

(2019) Sabyasachi Manna et al.   JOURNAL OF ORGANIC CHEMISTRY

Metal-, Photocatalyst-, and Light-Free Minisci C–H Alkylation of N-Heteroarenes with Oxalates

(2019) Jianyang Dong et al.   JOURNAL OF ORGANIC CHEMISTRY

Visible-Light-Induced Copper-Catalyzed Decarboxylative Coupling of Redox-Active Esters with N-Heteroarenes

(2019) Xue-Li Lyu et al.   ORGANIC LETTERS

Ketones and aldehydes as alkyl radical equivalents for C─H functionalization of heteroarenes

(2019) Jianyang Dong et al.   Science Advances

The synergistic effect of self-assembly and visible-light induced the oxidative C–H acylation of N-heterocyclic aromatic compounds with aldehydes

(2018) Lingling Zhang et al.   CHEMICAL COMMUNICATIONS

Drugs in Development for Malaria

(2018) Elizabeth A. Ashley et al.   DRUGS

Visible-Light-Initiated, Photocatalyst-Free Decarboxylative Coupling of Carboxylic Acids with N-Heterocycles

(2018) Xiao-Yu Zhang et al.   ORGANIC LETTERS

Photoredox-Mediated Direct Cross-Dehydrogenative Coupling of Heteroarenes and Amines

(2018) Jianyang Dong et al.   ORGANIC LETTERS

Metal-, Photocatalyst-, and Light-Free, Late-Stage C–H Alkylation of Heteroarenes and 1,4-Quinones Using Carboxylic Acids

(2018) Daniel R. Sutherland et al.   ORGANIC LETTERS

Construction and Functionalization of Heteroarenes by Use of Photoredox Catalysis

(2017) Oualid Boubertakh et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Intramolecular Minisci acylation under silver-free neutral conditions for the synthesis of azafluorenones and fluorenones

(2017) Joydev K. Laha et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Electrocatalytic Minisci Acylation Reaction of N-Heteroarenes Mediated by NH4I

(2017) Qing-Qing Wang et al.   ORGANIC LETTERS

Recent Advances in Direct C–H Functionalization of Pyrimidines

(2017) Egor Verbitskiy et al.   SYNTHESIS-STUTTGART

Visible Light Mediated Photoredox Catalytic Arylation Reactions

(2016) Indrajit Ghosh et al.   ACCOUNTS OF CHEMICAL RESEARCH

Transition metal-free Minisci reaction promoted by NCS, and TBHP: acylation of heteroarenes

(2016) Yogesh Siddaraju et al.   TETRAHEDRON

Recent developments in intermolecular radical arylations of arenes and heteroarenes

(2016) Josefa Hofmann et al.   TETRAHEDRON LETTERS

Recent developments for the photoinduced Ar–X bond dissociation reaction

(2016) Guanyinsheng Qiu et al.   Organic Chemistry Frontiers

Regiospecific Benzoylation of Electron-Deficient N-Heterocycles with Methylbenzenes via a Minisci-Type Reaction

(2015) Wajid Ali et al.   JOURNAL OF ORGANIC CHEMISTRY

TBHP/TFA mediated oxidative cross-dehydrogenative coupling of N-heterocycles with aldehydes

(2015) Jiayu Chen et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Transition Metal-Mediated Direct CH Arylation of Heteroarenes Involving Aryl Radicals

(2014) Hélène Bonin et al.   ADVANCED SYNTHESIS & CATALYSIS

Single Electron Transfer in Radical Ion and Radical-Mediated Organic, Materials and Polymer Synthesis

(2014) Na Zhang et al.   CHEMICAL REVIEWS

Transition-Metal-Free Coupling Reactions

(2014) Chang-Liang Sun et al.   CHEMICAL REVIEWS

Analysis of the Structural Diversity, Substitution Patterns, and Frequency of Nitrogen Heterocycles among U.S. FDA Approved Pharmaceuticals

(2014) Edon Vitaku et al.   JOURNAL OF MEDICINAL CHEMISTRY

A Transition Metal-Free Minisci Reaction: Acylation of Isoquinolines, Quinolines, and Quinoxaline

(2014) Yogesh Siddaraju et al.   JOURNAL OF ORGANIC CHEMISTRY

Radical Addition to Iminium Ions and Cationic Heterocycles

(2014) Johannes Tauber et al.   MOLECULES

Amine α-heteroarylation via photoredox catalysis: a homolytic aromatic substitution pathway

(2014) Christopher K. Prier et al.   Chemical Science

Metal-Free Cross-Dehydrogenative Coupling of Heterocycles with Aldehydes

(2013) Kiran Matcha et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Palladium-catalyzed ortho-acylation of 2-aryl pyridine derivatives using arylmethyl amines as new acyl sources

(2013) Qian Zhang et al.   CHEMICAL COMMUNICATIONS

A Radical Process towards the Development of Transition-Metal-Free Aromatic CarbonCarbon Bond-Forming Reactions

(2013) Tek Long Chan et al.   CHEMISTRY-A EUROPEAN JOURNAL

C–H bond activation enables the rapid construction and late-stage diversification of functional molecules

(2013) Joanna Wencel-Delord et al.   Nature Chemistry

Photoredox Activation for the Direct  -Arylation of Ketones and Aldehydes

(2013) M. T. Pirnot et al.   SCIENCE

Methyl Effects on Protein–Ligand Binding

(2012) Cheryl S. Leung et al.   JOURNAL OF MEDICINAL CHEMISTRY

Innate and Guided C–H Functionalization Logic

(2011) Tobias Brückl et al.   ACCOUNTS OF CHEMICAL RESEARCH

Organocatalysis and CH Activation Meet Radical- and Electron-Transfer Reactions

(2011) Armido Studer et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Discovery of an  -Amino C-H Arylation Reaction Using the Strategy of Accelerated Serendipity

(2011) A. McNally et al.   SCIENCE

Minisci reactions: Versatile CH-functionalizations for medicinal chemists

(2011) Matthew A. J. Duncton   MedChemComm

Privileged scaffolds for library design and drug discovery

(2010) Matthew E Welsch et al.   CURRENT OPINION IN CHEMICAL BIOLOGY

Transition-Metal-Catalyzed Direct Arylation of (Hetero)Arenes by CH Bond Cleavage

(2009) Lutz Ackermann et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION