Transition Metal-Free De Novo Synthesis of Sulfonated Pyrazoles from Sulfonyl Hydrazides, 1,3-Diketones, and Sodium Sulfinates at Room Temperature

Fluorinated Pyrazoles: From Synthesis to Applications

(2021) Pavel K. Mykhailiuk   CHEMICAL REVIEWS

Transition Metal‐free C‐H Sulfonylation and Pyrazole Annulation Cascade for the Synthesis of 4‐Sulfonyl Pyrazoles

(2020) Lihong Tian et al.   ChemCatChem

Copper-Catalyzed Aminoboration from Hydrazones To Generate Borylated Pyrazoles

(2019) Kim N. Tu et al.   ORGANIC LETTERS

Domino C-H Sulfonylation and Pyrazole Annulation for Fully Substituted Pyrazole Synthesis in Water Using Hydrophilic Enaminones

(2019) Yanhui Guo et al.   JOURNAL OF ORGANIC CHEMISTRY

Aerobic Oxidative Sulfenylation of Pyrazolones and Pyrazoles Catalyzed by Metal-Free Flavin–Iodine Catalysis

(2019) Kazumasa Tanimoto et al.   JOURNAL OF ORGANIC CHEMISTRY

Green approach for the synthesis of thiophenyl pyrazoles and isoxazoles by adopting 1,3-dipolar cycloaddition methodology and their antimicrobial activity

(2018) D.V. Sowmya et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

In Situ Generation of Nitrilimines from Aryldiazonium Salts and Diazo Esters: Synthesis of Fully Substituted Pyrazoles under Room Temperature

(2018) Ying Shao et al.   ORGANIC LETTERS

Copper Catalyzed Regioselective N - Alkynylation of Pyrazoles and Evaluation of the Anticancer Activity of Ethynyl- Pyrazoles

(2018) Mohan Chandra Sau et al.   ChemistrySelect

Synthesis of 5-Aryl-3(2H)-furanones Using Intramolecular Cyclization of Sulfonium Salts

(2018) Sho Inagaki et al.   JOURNAL OF ORGANIC CHEMISTRY

Facile and efficient access to Androsten-17-(1′,3′,4′)-pyrazoles and Androst-17β-(1′,3′,4′)-pyrazoles via Vilsmeier reagents, and their antiproliferative activity evaluation in vitro

(2017) Jian Li et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Recent advances of pyrazole-containing derivatives as anti-tubercular agents

(2017) Zhi Xu et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Review: biologically active pyrazole derivatives

(2017) Anam Ansari et al.   NEW JOURNAL OF CHEMISTRY

Copper-Mediated Domino Cyclization/Trifluoromethylation/Deprotection with TMSCF3: Synthesis of 4-(Trifluoromethyl)pyrazoles

(2017) Quande Wang et al.   ORGANIC LETTERS

Metal-free molecular iodine-catalyzed direct sulfonylation of pyrazolones with sodium sulfinates leading to sulfonated pyrazoles at room temperature

(2017) Wei Wei et al.   Organic Chemistry Frontiers

The therapeutic voyage of pyrazole and its analogs: A review

(2016) Mohemmed Faraz Khan et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Metal-Free Direct Construction of SulfonamidesviaIodine- Mediated Coupling Reaction of Sodium Sulfinates and Amines at Room Temperature

(2015) Wei Wei et al.   ADVANCED SYNTHESIS & CATALYSIS

Recent advances in bioactive pyrazoles

(2015) Ş.Güniz Küçükgüzel et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Metal-Free Iodine-Catalyzed Synthesis of Fully Substituted Pyrazoles and Its Sulphenylation

(2015) Jun Sun et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-catalyzed oxidative cyclization of arylamides and β-diketones: new synthesis of 2,4,5-trisubstituted oxazoles

(2015) Yang Bai et al.   RSC Advances

Copper-mediated pyrazole synthesis from 2,3-allenoates or 2-alkynoates, amines and nitriles

(2014) Bo Chen et al.   CHEMICAL COMMUNICATIONS

Regioselective C2 Sulfonylation of Indoles Mediated by Molecular Iodine

(2014) Praewpan Katrun et al.   JOURNAL OF ORGANIC CHEMISTRY

Dual Roles of Sulfonyl Hydrazides: A Three-Component Reaction To Construct Fully Substituted Pyrazoles Using TBAI/TBHP

(2014) Jie Zhang et al.   ORGANIC LETTERS

Disposition of fipronil in rats

(2013) J.P. Cravedi et al.   CHEMOSPHERE

Synthesis and antioxidant activity of amido-linked benzoxazolyl/benzothiazolyl/benzimidazolyl-pyrroles and pyrazoles

(2013) Suram Durgamma et al.   MEDICINAL CHEMISTRY RESEARCH

Lewis Base Catalyzed Synthesis of Multisubstituted 4-Sulfonyl-1H-Pyrazole Involving a Novel 1,3-Sulfonyl Shift

(2013) Yu Zhu et al.   ORGANIC LETTERS

A molecular dynamics investigation on the crizotinib resistance mechanism of C1156Y mutation in ALK

(2012) Hui-Yong Sun et al.   BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS

Oxidative Mizoroki-Heck-Type Reaction of Arylsulfonyl Hydrazides for a Highly Regio- and Stereoselective Synthesis of Polysubstituted Alkenes

(2012) Fu-Lai Yang et al.   CHEMISTRY-A EUROPEAN JOURNAL

Pyrazoles as Promising Scaffold for the Synthesis of Anti-Inflammatory and/or Antimicrobial Agent: A Review

(2012) Adnan A. Bekhit et al.   MINI-REVIEWS IN MEDICINAL CHEMISTRY

One-Pot, Two-Step Conversion of Aldehydes to Phosphonyl- and Sulfonylpyrazoles Using Bestmann–Ohira Reagent

(2012) Rahul Kumar et al.   ORGANIC LETTERS

Regioselective Synthesis of Sulfonylpyrazoles via Base Mediated Reaction of Diazosulfones with Nitroalkenes and a Facile Entry into Withasomnine‡

(2011) Rahul Kumar et al.   ORGANIC LETTERS

Efficient Synthesis of Pyrazoles: Oxidative CC/NN Bond-Formation Cascade

(2010) Julia J. Neumann et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Design and Synthesis of Benzosultine-sulfone as ao-Xylylene Precursor via Cross-enyne Metathesis and Rongalite: Further Expansion to Polycyclics via Regioselective Diels−Alder Reaction

(2010) Sambasivarao Kotha et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of Fully Substituted Pyrazoles via Regio- and Chemoselective Metalations

(2009) Christina Despotopoulou et al.   ORGANIC LETTERS

Development of Peptidomimetics with a Vinyl Sulfone Warhead as Irreversible Falcipain-2 Inhibitors

(2008) Roberta Ettari et al.   JOURNAL OF MEDICINAL CHEMISTRY

1,3-Dipolar Cycloadditions of Acetylenic Sulfones in Solution and on Solid Supports

(2008) Detian Gao et al.   JOURNAL OF ORGANIC CHEMISTRY