Synthesis and Structural Characteristics of all Mono- and Difluorinated 4,6-Dideoxy-d-xylo-hexopyranoses

Polyfluoroglycoside Synthesis via Simple Alkylation of an Anomeric Hydroxyl Group: Access to Fluoroetoposide Analogues

(2021) Thomas Tremblay et al.   JOURNAL OF ORGANIC CHEMISTRY

General Method for the Synthesis of α- or β-Deoxyaminoglycosides Bearing Basic Nitrogen

(2021) Kevin M. Hoang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

TBAF Effects 3,6-Anhydro Formation from 6-O-Tosyl Pyranosides

(2020) Zachary A. Morrison et al.   ORGANIC LETTERS

Sugar-Pirating as an Enabling Platform for the Synthesis of 4,6-Dideoxyhexoses

(2020) Yinan Zhang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Reagent-Controlled α-Selective Dehydrative Glycosylation of 2,6-Dideoxy Sugars: Construction of the Arugomycin Tetrasaccharide

(2020) Joseph R. Romeo et al.   ORGANIC LETTERS

Addressing the structural complexity of fluorinated glucose analogues: Insight into lipophilicities and solvation effects

(2020) Jacob St-Gelais et al.   CHEMISTRY-A EUROPEAN JOURNAL

Synthetic Fluorinated l-Fucose Analogs Inhibit Proliferation of Cancer Cells and Primary Endothelial Cells

(2020) Yuanwei Dai et al.   ACS Chemical Biology

Catalytic Activation of Cis-Vicinal Diols by Boronic Acids: Site-Selective Acylation of Carbohydrates

(2019) Naoyuki Shimada et al.   ORGANIC LETTERS

Molecular Insights into DC-SIGN Binding to Self-Antigens: The Interaction with the Blood Group A/B Antigens

(2019) Pablo Valverde et al.   ACS Chemical Biology

Synthesis and Lipophilicity of Trifluorinated Analogues of Glucose

(2019) Jacob St-Gelais et al.   JOURNAL OF ORGANIC CHEMISTRY

Rapid de Novo Preparation of 2,6-Dideoxy Sugar Libraries through Gold-Catalyzed Homopropargyl Orthoester Cyclization

(2019) Subbarao Yalamanchili et al.   ORGANIC LETTERS

Flexible Total Synthesis of 11-Deoxylandomycins and Their Non-Natural Analogues by Way of Asymmetric Metal Catalysis

(2019) Juyeol Lee et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Isolation and characterisation of an unexpected byproduct in the regioselective butane diacetal protection of α-methyl galactopyranoside

(2018) Clément Q. Fontenelle et al.   CARBOHYDRATE RESEARCH

The recognition of glycans by protein receptors. Insights from NMR spectroscopy

(2018) Ana Ardá et al.   CHEMICAL COMMUNICATIONS

Synthesis of Conformationally-Locked cis- and trans-Bicyclo[4.4.0] Mono-, Di-, and Trioxadecane Modifications of Galacto- and Glucopyranose; Experimental Limiting 3JH,H Coupling Constants for the Estimation of Carbohydrate Side Chain Populations and Beyond

(2018) Harsha Amarasekara et al.   JOURNAL OF ORGANIC CHEMISTRY

Anomer Preferences for Glucuronic and Galacturonic Acid and Derivatives and Influence of Electron-Withdrawing Substituents

(2018) Louise Kerins et al.   JOURNAL OF ORGANIC CHEMISTRY

Probing deoxysugar conformational preference: A comprehensive computational study investigating the effects of deoxygenation

(2018) Alison E. Vickman et al.   CARBOHYDRATE RESEARCH

A Chiron approach towards the stereoselective synthesis of polyfluorinated carbohydrates

(2018) Vincent Denavit et al.   Nature Communications

Facile Modulation of Antibody Fucosylation with Small Molecule Fucostatin Inhibitors and Cocrystal Structure with GDP-Mannose 4,6-Dehydratase

(2016) John G. Allen et al.   ACS Chemical Biology

Reagent-Controlled α-Selective Dehydrative Glycosylation of 2,6-Dideoxy- and 2,3,6-Trideoxy Sugars

(2016) Jason M. Nogueira et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Next Generation of Fluorine-Containing Pharmaceuticals, Compounds Currently in Phase II–III Clinical Trials of Major Pharmaceutical Companies: New Structural Trends and Therapeutic Areas

(2016) Yu Zhou et al.   CHEMICAL REVIEWS

Triacetonide of Glucoheptonic Acid in the Scalable Syntheses of d-Gulose, 6-Deoxy-d-gulose, l-Glucose, 6-Deoxy-l-glucose, and Related Sugars

(2016) Zilei Liu et al.   ORGANIC LETTERS

Synthesis of D -Desosamine and Analogs by Rapid Assembly of 3-Amino Sugars

(2015) Ziyang Zhang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Investigating the Influence of (Deoxy)fluorination on the Lipophilicity of Non-UV-Active Fluorinated Alkanols and Carbohydrates by a New log P Determination Method

(2015) Bruno Linclau et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Applications of Fluorine in Medicinal Chemistry

(2015) Eric P. Gillis et al.   JOURNAL OF MEDICINAL CHEMISTRY

Structural Basis of Ligand Binding to UDP-Galactopyranose Mutase from Mycobacterium tuberculosis Using Substrate and Tetrafluorinated Substrate Analogues

(2015) Karin E. van Straaten et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

New fluorinated fructose analogs as selective probes of the hexose transporter protein GLUT5

(2015) Olivier-Mohamad Soueidan et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

A thorough experimental study of CH/π interactions in water: quantitative structure–stability relationships for carbohydrate/aromatic complexes

(2015) Ester Jiménez-Moreno et al.   Chemical Science

Fluorinated Mechanism-Based Inhibitors: Common Themes and Recent Developments

(2014) Christina Tysoe et al.   CURRENT TOPICS IN MEDICINAL CHEMISTRY

BFMP: A Method for Discretizing and Visualizing Pyranose Conformations

(2014) Spandana Makeneni et al.   Journal of Chemical Information and Modeling

Immunogenicity Study of Globo H Analogues with Modification at the Reducing or Nonreducing End of the Tumor Antigen

(2014) Hsin-Yu Lee et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

l-Fucose from Vitamin C with Only Acetonide Protection

(2014) Zilei Liu et al.   ORGANIC LETTERS

Fluorine in Pharmaceutical Industry: Fluorine-Containing Drugs Introduced to the Market in the Last Decade (2001–2011)

(2013) Jiang Wang et al.   CHEMICAL REVIEWS

Tetrafluorination of Sugars as Strategy for Enhancing Protein-Carbohydrate Affinity: Application to UDP-GalpMutase Inhibition

(2013) Inès N'Go et al.   CHEMISTRY-A EUROPEAN JOURNAL

Carbohydrate-Based Molecules for Molecular Imaging in Nuclear Medicine

(2013) Goreti Ribeiro Morais et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

A Dynamic Combinatorial Approach for the Analysis of Weak Carbohydrate/Aromatic Complexes: Dissecting Facial Selectivity in CH/π Stacking Interactions

(2013) Andrés G. Santana et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Broadening the scope of glycosyltransferase-catalyzed sugar nucleotide synthesis

(2013) R. W. Gantt et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

Easy Access toL-Mannosides andL-Galactosides by Using CH Activation of the Corresponding 6-Deoxysugars

(2012) Tobias Gylling Frihed et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis and glycosidase inhibitory profiles of functionalised morpholines and oxazepanes

(2011) Peter A. Burland et al.   BIOORGANIC & MEDICINAL CHEMISTRY

De novo synthesis of deoxy sugar via a Wharton rearrangement

(2011) Hua-Yu Leo Wang et al.   CHEMICAL COMMUNICATIONS

Structure of the Major O-Specific Polysaccharide from the Lipopolysaccharide ofPseudomonas fluorescensBIM B-582: Identification of 4-Deoxy-d-xylo-hexose As a Component of Bacterial Polysaccharides

(2011) Olga A. Valueva et al.   JOURNAL OF NATURAL PRODUCTS

Radiopharmacological evaluation of 6-deoxy-6-[18F]fluoro-d-fructose as a radiotracer for PET imaging of GLUT5 in breast cancer

(2011) Melinda Wuest et al.   NUCLEAR MEDICINE AND BIOLOGY

Crystal structure of the synergistic antibiotic pair, lankamycin and lankacidin, in complex with the large ribosomal subunit

(2011) M. J. Belousoff et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

Fluorosugars: synthesis of the 2,3,4-trideoxy-2,3,4-trifluoro hexose analogues of d-glucose and d-altrose and assessment of their erythrocyte transmembrane transport

(2010) Stefano Bresciani et al.   CHEMICAL COMMUNICATIONS

Potassium carbonate–silica: a highly effective stationary phase for the chromatographic removal of organotin impurities

(2010) David C. Harrowven et al.   CHEMICAL COMMUNICATIONS

Fluorinated Glycosyl Amino Acids for Mucin-Like Glycopeptide Antigen Analogues

(2010) Sarah Wagner et al.   CHEMISTRY-A EUROPEAN JOURNAL

Synthesis and Structure Elucidation of Benzoylated Deoxyfluoropyranosides

(2010) Aslan M. Esmurziev et al.   JOURNAL OF CARBOHYDRATE CHEMISTRY

Stereochemical Survey of Digitoxin Monosaccharides

(2010) Hua-Yu Leo Wang et al.   ACS Medicinal Chemistry Letters

Recent advances in the synthesis of 2-deoxy-glycosides

(2009) Dianjie Hou et al.   CARBOHYDRATE RESEARCH

Natural-Product Sugar Biosynthesis and Enzymatic Glycodiversification

(2008) Christopher J. Thibodeaux et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis ofD-Trigalacturonic Acid Methylglycoside and Conformational Comparison with Its Sulfur Analogue

(2008) Kazunori YAMAMOTO et al.   BIOSCIENCE BIOTECHNOLOGY AND BIOCHEMISTRY

Acyl Group Migration and Cleavage in Selectively Protected β-d-Galactopyranosides as Studied by NMR Spectroscopy and Kinetic Calculations

(2008) Mattias U. Roslund et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Concise syntheses of d-desosamine, 2-thiopyrimidinyl desosamine donors, and methyl desosaminide analogues from d-glucose

(2007) Venkata Velvadapu et al.   CARBOHYDRATE RESEARCH