Diastereoselective Synthesis of Tetrahydrospiro[carbazole-1,3′-indolines] via an InBr3-Catalyzed Domino Diels–Alder Reaction

Enantioselective synthesis of tetrahydrocarbazoles via trienamine catalysis and their anxiolytic-like activity

(2020) Tushar Janardan Pawar et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Lipid‐Embedded Molecular Dynamics Simulation Model for Exploring the Reverse Prostaglandin D2 Agonism of CT‐133 towards CRTH2 in the Treatment of Type‐2 Inflammation Dependent Diseases

(2020) Abdul Rashid Issahaku et al.   CHEMISTRY & BIODIVERSITY

Rh(III)-Catalyzed Hydroarylation of Alkyne MIDA Boronates via C–H Activation of Indole Derivatives

(2019) Xiao Fei et al.   JOURNAL OF ORGANIC CHEMISTRY

Metal-Free Double Csp2–H Bond Functionalization: Strategy for Synthesizing Benzo[a]carbazoles from 2-Arylindoles and Acetophenones/Alkynes

(2019) Penghui Ni et al.   ORGANIC LETTERS

Construction of Spiro[indoline-3,3′-pyridazines] and Spiro[indene-2,3′-pyridazines] via TEMPO-Mediated Oxidative Aza-Diels-Alder Reactions

(2019) Rong Ye et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Catalytic asymmetric synthesis of spirooxindoles: recent developments

(2018) Guang-Jian Mei et al.   CHEMICAL COMMUNICATIONS

Selective Synthesis of 3-(9H-Carbazol-2-yl)indolin-2-ones and Spiro[tetrahydrocarbazole-3,3′-oxindoles] via a HOTf Catalyzed Three-Component Reaction

(2018) Ren-Yin Yang et al.   JOURNAL OF ORGANIC CHEMISTRY

Remote Control of Axial Chirality: Synthesis of Spirooxindole–Urazoles via Desymmetrization of ATAD

(2018) Lin-Lin Zhang et al.   ORGANIC LETTERS

Stereoselective Construction of Complex Spirooxindoles via Bisthiourea Catalyzed Three-Component Reactions

(2018) Lin-Lin Zhang et al.   CHINESE JOURNAL OF CHEMISTRY

Organocatalytic Asymmetric Synthesis of Spiro-Bridged and Spiro-Fused Heterocyclic Compounds Containing Chromane, Indole, and Oxindole Moieties

(2018) Zhi-Hao You et al.   ORGANIC LETTERS

2- and 3-Vinylindoles as 4π Components in Cycloaddition Reactions

(2017) Elisabetta Rossi et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

TfOH-Catalyzed One-Pot Domino Reaction for Diastereoselective Synthesis of Polysubstituted Tetrahydrospiro[carbazole-1,3′-indoline]s

(2017) Ren-Yin Yang et al.   JOURNAL OF ORGANIC CHEMISTRY

One-Pot Cascade Synthesis of Substituted Carbazoles from Indoles, Ketones, and Alkenes Using Oxygen as the Oxidant

(2017) Shanping Chen et al.   JOURNAL OF ORGANIC CHEMISTRY

L-Pyroglutamic Sulphonamide as Hydrogen-Bonding Organocatalyst: Enantioselective Diels–Alder Cyclization to Construct Carbazolespirooxindoles

(2017) Ji-Wei Ren et al.   JOURNAL OF ORGANIC CHEMISTRY

A Novel Synthesis of Aryl- and Heteroaryl - Annulated Carbazoles: Newly Synthesized Pyrido-, Benzo[a ]- and Spirooxindolinebenzo[a ]-carbazols

(2017) Karunanidhi Murali et al.   ChemistrySelect

Easy Access to a Library of Alkylindoles: Reductive Alkylation of Indoles with Carbonyl Compounds and Hydrosilanes under Indium Catalysis

(2016) Shota Nomiyama et al.   ADVANCED SYNTHESIS & CATALYSIS

Synthesis of benzo[a]carbazole derivatives from 3-ethylindoles by exploiting the dual character of benzoquinone as an oxidizing agent and dienophile

(2016) Chun-Wei Kuo et al.   CHEMICAL COMMUNICATIONS

An unprecedented benzannulation of oxindoles with enalcarbenoids: a regioselective approach to functionalized carbazoles

(2016) Kuldeep Singh Rathore et al.   CHEMICAL COMMUNICATIONS

Acid-Relayed Organocatalyticexo-Diels-Alder Cycloaddition of Cyclic Enones with 2-Vinyl-1H-indoles

(2016) Ji-Wei Ren et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Development and Scope of the Arene-Fused Domino Michael/Mannich Reaction: Application to the Total Syntheses of Aspidosperma Alkaloids (−)-Aspidospermidine, (−)-Tabersonine, and (−)-Vincadifformine

(2016) Senzhi Zhao et al.   JOURNAL OF ORGANIC CHEMISTRY

Cascade Reactions of Nitrones and Allenes for the Synthesis of Indole Derivatives

(2016) Laura L. Anderson et al.   JOURNAL OF ORGANIC CHEMISTRY

Hexadehydro-Diels–Alder (HDDA)-Enabled Carbazolyne Chemistry: Single Step, de Novo Construction of the Pyranocarbazole Core of Alkaloids of the Murraya koenigii (Curry Tree) Family

(2016) Tao Wang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Enantioselective Construction of Functionalized Tetrahydrocarbazoles Enabled by Asymmetric Relay Catalysis of Gold Complex and Chiral Brønsted Acid

(2016) Feng Zhao et al.   ORGANIC LETTERS

Indole-to-Carbazole Strategy for the Synthesis of Substituted Carbazoles under Metal-Free Conditions

(2016) Shanping Chen et al.   ORGANIC LETTERS

Synthesis of pentacyclic pyrrolo[3,4- a ]carbazole-1,3(2 H )-diones via an intermolecular Diels–Alder, intramolecular carbonyl-ene reaction strategy

(2016) Matokah Abualnaja et al.   TETRAHEDRON

Silver(i)-catalysed domino alkyne-annulation/Diels–Alder reaction: a mild synthetic approach to tetrahydrospiro[carbazole-4,3′-indoline] scaffolds

(2016) Pankaj Sharma et al.   Organic Chemistry Frontiers

Organocatalytic Diels-Alder Reaction of 2-Vinylindoles with Methyleneindolinones: An Efficient Approach to Functionalized Carbazolespirooxindoles

(2015) Lin-Jie Huang et al.   ADVANCED SYNTHESIS & CATALYSIS

Synthesis of Carbazole Alkaloids by Ring-Closing Metathesis and Ring Rearrangement-Aromatization

(2015) Kalyan Dhara et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Metal-Free Dehydrogenative Diels-Alder Reactions of 2-Methyl-3-Alkylindoles with Dienophiles: Rapid Access to Tetrahydrocarbazoles, Carbazoles, and Heteroacenes

(2015) Liejin Zhou et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis and biological evaluation of spiro[cyclopropane-1,3′-indolin]-2′-ones as potential anticancer agents

(2015) Chada Narsimha Reddy et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Multi-site cyclization via initial C–H activation using a rhodium(iii) catalyst: rapid assembly of frameworks containing indoles and indolines

(2015) Ji-Rong Huang et al.   CHEMICAL COMMUNICATIONS

Brønsted Acid Catalyzed Asymmetric Diels–Alder Reactions: Stereoselective Construction of Spiro[tetrahydrocarbazole-3,3′-oxindole] Framework

(2015) Yang Wang et al.   JOURNAL OF ORGANIC CHEMISTRY

Construction of Benzo[c]carbazoles and Their Antitumor Derivatives through the Diels–Alder Reaction of 2-Alkenylindoles and Arynes

(2015) Feng Sha et al.   JOURNAL OF ORGANIC CHEMISTRY

Application of 3-Methyl-2-vinylindoles in Catalytic Asymmetric Povarov Reaction: Diastereo- and Enantioselective Synthesis of Indole-Derived Tetrahydroquinolines

(2015) Wei Dai et al.   JOURNAL OF ORGANIC CHEMISTRY

Diastereoselective synthesis of functionalised carbazoles via a sequential Diels–Alder/ene reaction strategy

(2015) Joseph Cowell et al.   RSC Advances

Construction of benzo[a]carbazole derivatives via Diels–Alder reaction of arynes with vinylindoles

(2015) Lijun Wu et al.   RSC Advances

Rapid Synthesis of Fused N-Heterocycles by Transition-Metal-Free Electrophilic Amination of Arene CH Bonds

(2014) Hongyin Gao et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Efficient synthesis of carbazolespirooxindole skeletons via asymmetric Diels–Alder reaction of 3-vinylindoles and methyleneindolinones

(2014) Haifeng Zheng et al.   CHEMICAL COMMUNICATIONS

Synthetic Approaches to 3-(2-Nitroalkyl) Indoles and Their Use to Access Tryptamines and Related Bioactive Compounds

(2014) Stefano Lancianesi et al.   CHEMICAL REVIEWS

Organocatalytic Asymmetric Synthesis of 1,1-Diarylethanes by Transfer Hydrogenation

(2014) Zhaobin Wang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Catalytic asymmetric Povarov reaction of isatin-derived 2-azadienes with 3-vinylindoles

(2014) Hong-Hao Zhang et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Studies on the stereochemical assignment of 3-acylidene 2-oxindoles

(2014) Steven J. Edeson et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Some electrophilic reactivity studies of di-(2-indolyl)dibenzofurans and di-(2-indolyl)carbazoles

(2014) Ibrahim F. Sengul et al.   TETRAHEDRON

Catalytic asymmetric synthesis of 3,3-disubstituted oxindoles: diazooxindole joins the field

(2014) Zhong-Yan Cao et al.   TETRAHEDRON LETTERS

Organocatalytic Asymmetric Assembly Reactions: Synthesis of Spirooxindoles via Organocascade Strategies

(2014) Daojuan Cheng et al.   ACS Catalysis

Direct Assembly of Benzo[a]carbazole-5-carboxylates via a Diels-Alder Reaction with Arynes and 3-Alkenylindoles

(2014) Yuan Tao et al.   Asian Journal of Organic Chemistry

Recent Advances in Asymmetric Organocatalytic Construction of 3,3′-Spirocyclic Oxindoles

(2013) Liang Hong et al.   ADVANCED SYNTHESIS & CATALYSIS

A Visible-Light-Mediated Synthesis of Carbazoles

(2013) Augusto C. Hernandez-Perez et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Total Synthesis of the Biscarbazole Alkaloids Murrafoline A-D by a Domino Sonogashira Coupling/Claisen Rearrangement/Electrocyclization Reaction

(2013) V. Pavan Kumar et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Domino Michael/Mannich/N-Alkylation Route to the Tetrahydrocarbazole Framework of Aspidosperma Alkaloids: Concise Total Syntheses of (−)-Aspidospermidine, (−)-Tabersonine, and (−)-Vincadifformine

(2013) Senzhi Zhao et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Mild, efficient Fischer indole synthesis using 2,4,6-trichloro-1,3,5-triazine (TCT)

(2013) Eranna Siddalingamurthy et al.   TETRAHEDRON LETTERS

Occurrence, Biogenesis, and Synthesis of Biologically Active Carbazole Alkaloids

(2012) Arndt W. Schmidt et al.   CHEMICAL REVIEWS

Isatins As Privileged Molecules in Design and Synthesis of Spiro-Fused Cyclic Frameworks

(2012) Girija S. Singh et al.   CHEMICAL REVIEWS

Enantioselective [4+2] Cycloadditions of 2-Vinyl-1 H-indoles with 3-Nitro-2 H-chromenes Catalyzed by a Zn(OTf)2/Bis(oxazoline) Complex: An Efficient Approach to Fused Heterocycles with a Quaternary Stereocenter

(2012) Fen Tan et al.   Chemistry-An Asian Journal

Intramolecular Oxidative C−N Bond Formation for the Synthesis of Carbazoles: Comparison of Reactivity between the Copper-Catalyzed and Metal-Free Conditions

(2011) Seung Hwan Cho et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Highly Efficient Hydrogen-Bonding Catalysis of the Diels–Alder Reaction of 3-Vinylindoles and Methyleneindolinones Provides Carbazolespirooxindole Skeletons

(2011) Bin Tan et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Asymmetric Catalysis of Diels–Alder Reactions with in Situ Generated Heterocyclicortho-Quinodimethanes

(2011) Yankai Liu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Reductive Alkylation of Indoles with Alkynes and Hydrosilanes under Indium Catalysis

(2011) Teruhisa Tsuchimoto et al.   ORGANIC LETTERS

An Enantioselective Approach to Highly Substituted Tetrahydrocarbazoles through Hydrogen Bonding-Catalyzed Cascade Reactions

(2010) Xu-Fan Wang et al.   ORGANIC LETTERS

Indium(III) bromide-catalyzed hydroarylation of alkynes with indoles

(2010) G. Bhaskar et al.   TETRAHEDRON LETTERS

Antifungal Carbazoles

(2009) Karin Thevissen et al.   CURRENT MEDICINAL CHEMISTRY

Brønsted Acid Mediated Tandem Diels−Alder/Aromatization Reactions of Vinylindoles

(2009) Cai-Bao Chen et al.   JOURNAL OF ORGANIC CHEMISTRY

Organocatalytic Asymmetric Diels-Alder Reactions of 3-Vinylindoles

(2008) Claudio Gioia et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Indium-Catalyzed Annulation of 2-Aryl- and 2-Heteroarylindoles with Propargyl Ethers: Concise Synthesis and Photophysical Properties of Diverse Aryl- and Heteroaryl-Annulated[a]carbazoles

(2008) Teruhisa Tsuchimoto et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Transition metals in organic synthesis - Part 83#: Synthesis and pharmacological potential of carbazoles

(2008) Taylor A. Choi et al.   MEDICINAL CHEMISTRY RESEARCH