A2A Adenosine Receptor Partial Agonism Related to Structural Rearrangements in an Activation Microswitch
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Title
A2A Adenosine Receptor Partial Agonism Related to Structural Rearrangements in an Activation Microswitch
Authors
Keywords
NMR spectroscopy, G protein-coupled receptors, partial agonists, drug efficacy
Journal
STRUCTURE
Volume 29, Issue 2, Pages 170-176.e3
Publisher
Elsevier BV
Online
2020-11-24
DOI
10.1016/j.str.2020.11.005
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