Chalcone hybrids as potential anticancer agents: Current development, mechanism of action, and structure‐activity relationship
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Title
Chalcone hybrids as potential anticancer agents: Current development, mechanism of action, and structure‐activity relationship
Authors
Keywords
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Journal
MEDICINAL RESEARCH REVIEWS
Volume 40, Issue 5, Pages 2049-2084
Publisher
Wiley
Online
2020-06-11
DOI
10.1002/med.21698
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- Design and Synthesis of C3-Pyrazole/Chalcone-Linked Beta-Carboline Hybrids: Antitopoisomerase I, DNA-Interactive, and Apoptosis-Inducing Anticancer Agents
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- Synthesis, biological evaluation and molecular docking of novel chalcone–coumarin hybrids as anticancer and antimalarial agents
- (2014) Ratchanok Pingaew et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Antiobesity, antioxidant and cytotoxicity activities of newly synthesized chalcone derivatives and their metal complexes
- (2014) Mohamed Ramadan El Sayed Aly et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
- Synthesis, characterization of new imidazoquinonyl chalcones and pyrazolines as potential anticancer and antioxidant agents
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- Synthesis, in-vitro screening, and docking analysis of novel pyrrolidine and piperidine-substituted ethoxy chalcone as anticancer agents
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- Advances in Chalcones with Anticancer Activities
- (2014) Chandrabose Karthikeyan et al. Recent Patents on Anti-Cancer Drug Discovery
- Anticancer Activity of Pyrazole via Different Biological Mechanisms
- (2014) Simpal Chauhan et al. SYNTHETIC COMMUNICATIONS
- Synthesis of imidazo[2,1-b][1,3,4]thiadiazole–chalcones as apoptosis inducing anticancer agents
- (2014) Ahmed Kamal et al. MedChemComm
- Synthesis and anticancer activity evaluation of resveratrol–chalcone conjugates
- (2014) Deepak Kumar et al. MedChemComm
- Synthesis and Antitumor Activity of Novel Nitrogen Mustard-Linked Chalcones
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- Chromenylchalcones showing cytotoxicity on human colon cancer cell lines and in silico docking with aurora kinases
- (2013) Soon Young Shin et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Design, synthesis and biological evaluation of millepachine derivatives as a new class of tubulin polymerization inhibitors
- (2013) Guangcheng Wang et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Chalcones, inhibitors for topoisomerase I and cathepsin B and L, as potential anti-cancer agents
- (2013) Seok-Ho Kim et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Novel anthraquinone based chalcone analogues containing an imine fragment: Synthesis, cytotoxicity and anti-angiogenic activity
- (2013) Branka Kolundžija et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Synthesis and antiproliferative and c-Src kinase inhibitory activities of cinnamoyl- and pyranochromen-2-one derivatives
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- Adamantyl Arotinoids That Inhibit IκB Kinase α and IκB Kinase β
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- Synthesis and evaluation of novel marine bromopyrrole alkaloid-based hybrids as anticancer agents
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- Chalcone derivatives from the fern Cyclosorus parasiticus and their anti-proliferative activity
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- Triazole-linked Chalcone and Flavone Hybrid Compounds Based on AZT Exhibiting In Vitro Anti-Cancer Activity
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- Synthesis and anticancer activity of some new s-triazine derivatives
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- A New Age for Iron: Antitumoral Ferrocenes
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- New chalcone dimers from Caesalpinia ferrea Mart act as potent inhibitors of DNA topoisomerase II
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- Cytotoxic activity evaluation and QSAR study of chromene-based chalcones
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- Anti-breast cancer activity of heteroaryl chalcone derivatives
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- Synthesis and biological evaluation of bifendate–chalcone hybrids as a new class of potential P-glycoprotein inhibitors
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- Cytotoxic and apoptotic effects of chalcone derivatives of 2-acetyl thiophene on human colon adenocarcinoma cells
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- Design, synthesis and biological evaluation of novel (E)-α-benzylsulfonyl chalcone derivatives as potential BRAF inhibitors
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- Synthesis of novel quinoline-2-one based chalcones of potential anti-tumor activity
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- Synthesis and cytotoxicity evaluation of biaryl-based chalcones and their potential in TNFα-induced nuclear factor-κB activation inhibition
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- Design, synthesis and anticancer activity of nitric oxide donating/chalcone hybrids
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- Synthesis and antiproliferative evaluation of 3-phenylquinolinylchalcone derivatives against non-small cell lung cancers and breast cancers
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- Indole molecules as inhibitors of tubulin polymerization: potential new anticancer agents
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- Synthesis of Some Coumarinyl Chalcones and their Antiproliferative Activity Against Breast Cancer Cell Lines
- (2012) Kuldeep Patel et al. Letters in Drug Design & Discovery
- Synthesis and biologic activities of some novel heterocyclic chalcone derivatives
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- Anti-Tumor Activity of New Artemisinin-Chalcone Hybrids
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- Chalcone-imidazolone conjugates induce apoptosis through DNA damage pathway by affecting telomeres
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- Design, Synthesis and Antitumor Activity of Novel Artemisinin Derivatives Using Hybrid Approach
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- A chalcone-related small molecule that induces methuosis, a novel form of non-apoptotic cell death, in glioblastoma cells
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- Design, synthesis and antiproliferative activity of urocanic-chalcone hybrid derivatives
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- Synthesis and antitumor activity of novel chalcone derivatives
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- Identification of chalcones as in vivo liver monofunctional phase II enzymes inducers
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- Synthesis and biological evaluation of 2′,5′-dimethoxychalcone derivatives as microtubule-targeted anticancer agents
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- Synthesis, molecular modeling and biological evaluation of guanidine derivatives as novel antitubulin agents
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- Synthesis and biological evaluation of novel coumarin-based inhibitors of Cdc25 phosphatases
- (2010) Sergio Valente et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Synthesis and anti-cancer activity of chalcone linked imidazolones
- (2010) Ahmed Kamal et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Synthesis and biological evaluation of indolyl chalcones as antitumor agents
- (2010) Dalip Kumar et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Synthesis and in vitro evaluation of novel coumarin–chalcone hybrids as potential anticancer agents
- (2010) Koneni V. Sashidhara et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Synthesis of Imidazothiazole-Chalcone Derivatives as Anticancer and Apoptosis Inducing Agents
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- New 4-Maleamic Acid and 4-Maleamide Peptidyl Chalcones as Potential Multitarget Drugs for Human Prostate Cancer
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- A boronic acid chalcone analog of combretastatin A-4 as a potent anti-proliferation agent
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- Synthesis, characterization, electrochemical studies and antitumor activity of some new chalcone analogues containing ferrocenyl pyrazole moiety
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- Hybrid Molecules with a Dual Mode of Action: Dream or Reality?†
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