Concatenated γ-aminobutyric acid type A receptors revisited: Finding order in chaos

Galantamine is not a positive allosteric modulator of human α4β2 or α7 nicotinic acetylcholine receptors

(2018) Natalia M Kowal et al.   BRITISH JOURNAL OF PHARMACOLOGY

Concatenated nicotinic acetylcholine receptors: A gift or a curse?

(2018) Philip Kiær Ahring et al.   JOURNAL OF GENERAL PHYSIOLOGY

Probing the molecular basis for affinity/potency- and efficacy-based subtype-selectivity exhibited by benzodiazepine-site modulators at GABAA receptors

(2018) Pella Cecilia Söderhielm et al.   BIOCHEMICAL PHARMACOLOGY

Structure of a human synaptic GABAA receptor

(2018) Shaotong Zhu et al.   NATURE

Low Expression in Xenopus Oocytes and Unusual Functional Properties of α1β2γ2 GABAA Receptors with Non-Conventional Subunit Arrangement

(2017) Roland Baur et al.   PLoS One

α subunits in GABAA receptors are dispensable for GABA and diazepam action

(2017) Nisa Wongsamitkul et al.   Scientific Reports

High and low GABA sensitivity α4β2δ GABAA receptors are expressed in Xenopus laevis oocytes with divergent stoichiometries

(2016) Leonny Y. Hartiadi et al.   BIOCHEMICAL PHARMACOLOGY

A pharmacological characterization of GABA, THIP and DS2 at binary α4β3 and β3δ receptors: GABA activates β3δ receptors via the β3(+)δ(−) interface

(2016) H.J. Lee et al.   BRAIN RESEARCH

Comparison of γ-Aminobutyric Acid, Type A (GABAA), Receptor αβγ and αβδ Expression Using Flow Cytometry and Electrophysiology

(2016) Emmanuel J. Botzolakis et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

A pharmacological assessment of agonists and modulators at α4β2γ2 and α4β2δ GABA A receptors: The challenge in comparing apples with oranges

(2016) Philip K. Ahring et al.   PHARMACOLOGICAL RESEARCH

Zolpidem is a potent stoichiometry-selective modulator of α1β3 GABAA receptors: evidence of a novel benzodiazepine site in the α1-α1 interface

(2016) Ahmad Tarmizi Che Has et al.   Scientific Reports

The Direct Actions of GABA, 2’-Methoxy-6-Methylflavone and General Anaesthetics at β3γ2L GABAA Receptors: Evidence for Receptors with Different Subunit Stoichiometries

(2015) Han Chow Chua et al.   PLoS One

Crystal structure of a human GABAA receptor

(2014) Paul S. Miller et al.   NATURE

A Unified Model of the GABAA Receptor Comprising Agonist and Benzodiazepine Binding Sites

(2013) Rikke Bergmann et al.   PLoS One

Characteristics of concatemeric GABAA receptors containing α4/δ subunits expressed in Xenopus oocytes

(2011) Hong-Jin Shu et al.   BRITISH JOURNAL OF PHARMACOLOGY

Three Arginines in the GABAA Receptor Binding Pocket Have Distinct Roles in the Formation and Stability of Agonist- versus Antagonist-Bound Complexes

(2011) M. P. Goldschen-Ohm et al.   MOLECULAR PHARMACOLOGY

Diversity of Structure and Function of α1α6β3δ GABAAReceptors

(2010) Roland Baur et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Expression of Functional Human  6 2 3* Acetylcholine Receptors in Xenopus laevis Oocytes Achieved through Subunit Chimeras and Concatamers

(2010) A. Kuryatov et al.   MOLECULAR PHARMACOLOGY

Use of concatamers to study GABAAreceptor architecture and function: application to δ-subunit-containing receptors and possible pitfalls

(2009) Erwin Sigel et al.   BIOCHEMICAL SOCIETY TRANSACTIONS

Pentameric concatenated (α4)2(β2)3 and (α4)3(β2)2 nicotinic acetylcholine receptors: subunit arrangement determines functional expression

(2009) A-L Carbone et al.   BRITISH JOURNAL OF PHARMACOLOGY

Unanticipated Structural and Functional Properties of δ-Subunit-containing GABAAReceptors

(2009) Kuldeep H. Kaur et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Structure of α6β3δ GABAAreceptors and their lack of ethanol sensitivity

(2009) Roland Baur et al.   JOURNAL OF NEUROCHEMISTRY

Steroid Interaction with a Single Potentiating Site Is Sufficient to Modulate GABA-A Receptor Function

(2009) J. R. Bracamontes et al.   MOLECULAR PHARMACOLOGY

NS11394 [3'-[5-(1-Hydroxy-1-methyl-ethyl)-benzoimidazol-1-yl]-biphenyl-2-carbonitrile], a Unique Subtype-Selective GABAA Receptor Positive Allosteric Modulator: In Vitro Actions, Pharmacokinetic Properties and in Vivo Anxiolytic Efficacy

(2008) N. R. Mirza et al.   JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS

International Union of Pharmacology. LXX. Subtypes of  -Aminobutyric AcidA Receptors: Classification on the Basis of Subunit Composition, Pharmacology, and Function. Update

(2008) R. W. Olsen et al.   PHARMACOLOGICAL REVIEWS