Identifying lead hits in catalyst discovery by screening and deconvoluting complex mixtures of catalyst components

Nickel(II)-Catalyzed Direct Arylation of C–H Bonds in Aromatic Amides Containing an 8-Aminoquinoline Moiety as a Directing Group

(2014) Ayana Yokota et al.   JOURNAL OF ORGANIC CHEMISTRY

Nickel-Catalyzed Site-Selective Alkylation of Unactivated C(sp3)–H Bonds

(2014) Xuesong Wu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Contemporary screening approaches to reaction discovery and development

(2014) Karl D. Collins et al.   Nature Chemistry

Breaking the dichotomy of reactivity vs. chemoselectivity in catalytic SN1 reactions of alcohols

(2014) Malik Hellal et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Nanomole-scale high-throughput chemistry for the synthesis of complex molecules

(2014) A. Buitrago Santanilla et al.   SCIENCE

8-Aminoquinoline: A Powerful Directing Group in Metal-Catalyzed Direct Functionalization of CH Bonds

(2013) Matthieu Corbet et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic Functionalization of C(sp2)H and C(sp3)H Bonds by Using Bidentate Directing Groups

(2013) Guy Rouquet et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Scope and Limitations of Auxiliary-Assisted, Palladium-Catalyzed Arylation and Alkylation of sp2 and sp3 C–H Bonds

(2013) Enrico T. Nadres et al.   JOURNAL OF ORGANIC CHEMISTRY

Nickel-Catalyzed Direct Arylation of C(sp3)–H Bonds in Aliphatic Amides via Bidentate-Chelation Assistance

(2013) Yoshinori Aihara et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Organoboron Acids and Their Derivatives as Catalysts for Organic Synthesis

(2013) Elena Dimitrijević et al.   ACS Catalysis

Rapid Catalyst Identification for the Synthesis of the Pyrimidinone Core of HIV Integrase Inhibitors

(2012) Ana Bellomo et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Reaction Discovery by Using a Sandwich Immunoassay

(2012) Julia Quinton et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Boronic Acid Catalysis as a Mild and Versatile Strategy for Direct Carbo- and Heterocyclizations of Free Allylic Alcohols

(2012) Hongchao Zheng et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Ruthenium-catalyzed direct arylation of C–H bonds in aromatic amides containing a bidentate directing group: significant electronic effects on arylation

(2012) Yoshinori Aihara et al.   Chemical Science

Three-component reaction discovery enabled by mass spectrometry of self-assembled monolayers

(2011) Timothy J. Montavon et al.   Nature Chemistry

Discovery of an  -Amino C-H Arylation Reaction Using the Strategy of Accelerated Serendipity

(2011) A. McNally et al.   SCIENCE

A Simple, Multidimensional Approach to High-Throughput Discovery of Catalytic Reactions

(2011) D. W. Robbins et al.   SCIENCE

A review of new developments in the Friedel–Crafts alkylation – From green chemistry to asymmetric catalysis

(2010) Magnus Rueping et al.   Beilstein Journal of Organic Chemistry

Direct Nucleophilic SN1-Type Reactions of Alcohols

(2010) Enrico Emer et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Boronic Acid Catalyzed Friedel−Crafts Reactions of Allylic Alcohols with Electron-Rich Arenes and Heteroarenes.

(2010) J. Adam McCubbin et al.   JOURNAL OF ORGANIC CHEMISTRY

Tandem Processes Identified from Reaction Screening: Nucleophilic Addition to ArylN-Phosphinylimines Employing La(III)-TFAA Activation

(2010) Hidenori Kinoshita et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

A combinatorial approach to the identification of self-assembled ligands for rhodium-catalysed asymmetric hydrogenation

(2010) Joerg Wieland et al.   Nature Chemistry

Organocatalyzed Friedel–Crafts arylation of benzylic alcohols

(2010) J. Adam McCubbin et al.   TETRAHEDRON LETTERS

A pentafluorophenylboron oxalate additive in non-aqueous electrolytes for lithium batteries

(2009) L.F. Li et al.   ELECTROCHEMISTRY COMMUNICATIONS

Mass Spectrometric Screening of Chiral Catalysts by Monitoring the Back Reaction of Quasienantiomeric Products: Palladium-Catalyzed Allylic Substitution

(2008) Constanze A. Müller et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Mass Spectrometric Screening of Enantioselective Diels–Alder Reactions

(2008) Antje Teichert et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Combinatorial Ligand Development Based on Mass Spectrometric Screening and a Double Mass-Labeling Strategy

(2008) Christian Markert et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY