Rhodium(iii)-catalyzed regioselective C2-amidation of indoles with N-(2,4,6-trichlorobenzoyloxy)amides and its synthetic application to the development of a novel potential PPARγ modulator
Published 2014 View Full Article
- Home
- Publications
- Publication Search
- Publication Details
Title
Rhodium(iii)-catalyzed regioselective C2-amidation of indoles with N-(2,4,6-trichlorobenzoyloxy)amides and its synthetic application to the development of a novel potential PPARγ modulator
Authors
Keywords
-
Journal
ORGANIC & BIOMOLECULAR CHEMISTRY
Volume 12, Issue 35, Pages 6831-6836
Publisher
Royal Society of Chemistry (RSC)
Online
2014-05-09
DOI
10.1039/c4ob00637b
References
Ask authors/readers for more resources
Related references
Note: Only part of the references are listed.- Rhodium(III)-Catalyzed Regioselective Direct C-2 Alkenylation of Indoles Assisted by the Removable N-(2-Pyrimidyl) Group
- (2014) Binwei Gong et al. ADVANCED SYNTHESIS & CATALYSIS
- Rhodium(iii)-catalyzed C2-selective carbenoid functionalization and subsequent C7-alkenylation of indoles
- (2014) Jingjing Shi et al. CHEMICAL COMMUNICATIONS
- Mechanistic Studies of the Rhodium-Catalyzed Direct C–H Amination Reaction Using Azides as the Nitrogen Source
- (2014) Sae Hume Park et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Carboxylate-Assisted Ruthenium-Catalyzed Alkyne Annulations by C–H/Het–H Bond Functionalizations
- (2013) Lutz Ackermann ACCOUNTS OF CHEMICAL RESEARCH
- Carboxylate-Assisted Ruthenium(II)-Catalyzed Hydroarylations of Unactivated Alkenes through C-H Cleavage
- (2013) Marvin Schinkel et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Mild Rhodium(III)-Catalyzed Direct CH Allylation of Arenes with Allyl Carbonates
- (2013) Honggen Wang et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Palladium-catalyzed decarboxylative C2-acylation of indoles with α-oxocarboxylic acids
- (2013) Changduo Pan et al. CHEMICAL COMMUNICATIONS
- Rh(iii)-catalyzed dehydrogenative alkylation of (hetero)arenes with allylic alcohols, allowing aldol condensation to indenes
- (2013) Zhuangzhi Shi et al. CHEMICAL COMMUNICATIONS
- Aerobic Ru-catalyzed direct C2-olefination of N-heteroarenes with alkenes directed by a removable N-dimethylcarbamoyl group
- (2013) Luo-Qiang Zhang et al. CHEMICAL COMMUNICATIONS
- C–H nitrogenation and oxygenation by ruthenium catalysis
- (2013) Vedhagiri S. Thirunavukkarasu et al. CHEMICAL COMMUNICATIONS
- Rhodium-Catalyzed Directed Sulfenylation of Arene CH Bonds
- (2013) Yaxi Yang et al. CHEMISTRY-A EUROPEAN JOURNAL
- Optimization of Novel Indole-2-carboxamide Inhibitors of Neurotropic Alphavirus Replication
- (2013) Janice A. Sindac et al. JOURNAL OF MEDICINAL CHEMISTRY
- Design of Potent Poxvirus Inhibitors of the Heterodimeric Processivity Factor Required for Viral Replication
- (2013) Manunya Nuth et al. JOURNAL OF MEDICINAL CHEMISTRY
- Copper-Mediated Direct C2-Cyanation of Indoles Using Acetonitrile as the Cyanide Source
- (2013) Changduo Pan et al. JOURNAL OF ORGANIC CHEMISTRY
- Synthesis of C-2 Arylated Tryptophan Amino Acids and Related Compounds through Palladium-Catalyzed C–H Activation
- (2013) Sara Preciado et al. JOURNAL OF ORGANIC CHEMISTRY
- Ruthenium-Catalyzed Regioselective C2 Alkenylation of Indoles and Pyrroles via C–H Bond Functionalization
- (2013) Bin Li et al. JOURNAL OF ORGANIC CHEMISTRY
- RhIII/CuII-Cocatalyzed Synthesis of 1H-Indazoles through C–H Amidation and N–N Bond Formation
- (2013) Da-Gang Yu et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- C–H bond activation enables the rapid construction and late-stage diversification of functional molecules
- (2013) Joanna Wencel-Delord et al. Nature Chemistry
- Aryne Insertion Reactions Leading to Bioactive Fused Quinazolinones: Diastereoselective Total Synthesis of Cruciferane
- (2013) Sagar D. Vaidya et al. ORGANIC LETTERS
- Rh(III)-Catalyzed Intermolecular C–H Amination of 1-Aryl-1H-pyrazol-5(4H)-ones with Alkylamines
- (2013) Kui Wu et al. ORGANIC LETTERS
- Highly Regioselective C2-Alkenylation of Indoles Using the N-Benzoyl Directing Group: An Efficient Ru-Catalyzed Coupling Reaction
- (2013) Veeranjaneyulu Lanke et al. ORGANIC LETTERS
- Sulfoximine Directed Intermolecular o-C–H Amidation of Arenes with Sulfonyl Azides
- (2013) M. Ramu Yadav et al. ORGANIC LETTERS
- Rhodium-Catalyzed Intermolecular Oxidative Cross-Coupling of (Hetero)Arenes with Chalcogenophenes
- (2013) Vutukuri Prakash Reddy et al. ORGANIC LETTERS
- Double Annulative Cascade of Tryptophan-Containing Peptides Triggered by Selectfluor
- (2013) Bret Tréguier et al. ORGANIC LETTERS
- Rhodium(III)-Catalyzed C–H Activation and Amidation of Arenes Using N-Arenesulfonated Imides as Amidating Reagents
- (2013) Songjie Yu et al. ORGANIC LETTERS
- Rh[III]-Catalyzed C–H Amidation Using Aroyloxycarbamates To Give N-Boc Protected Arylamines
- (2013) Christoph Grohmann et al. ORGANIC LETTERS
- Rhodium(III)-Catalyzed Intermolecular N-Chelator-Directed Aromatic C–H Amidation with Amides
- (2013) Huaiqing Zhao et al. ORGANIC LETTERS
- Rh(III)-Catalyzed C–H Amidation with N-Hydroxycarbamates: A New Entry to N-Carbamate-Protected Arylamines
- (2013) Bing Zhou et al. ORGANIC LETTERS
- Intramolecular C(sp3)–H amination
- (2013) Jenna L. Jeffrey et al. Chemical Science
- Rh(iii)-catalyzed C–H activation/cycloaddition of benzamides and methylenecyclopropanes: divergence in ring formation
- (2013) Sunliang Cui et al. Chemical Science
- Rh(iii)-catalyzed C–H activation–desymmetrization of diazabicycles with arenes: facile synthesis of functionalized cyclopentenes
- (2013) Yan Zhang et al. Chemical Science
- Controlling Site Selectivity in Palladium-Catalyzed C–H Bond Functionalization
- (2012) Sharon R. Neufeldt et al. ACCOUNTS OF CHEMICAL RESEARCH
- Rhodium(III)-Catalyzed Oxidative CH Functionalization of Azomethine Ylides
- (2012) Wencui Zhen et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Copper-Mediated and Copper-Catalyzed Cross-Coupling of Indoles and 1,3-Azoles: Double CH Activation
- (2012) Mayuko Nishino et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Rhodium-Catalyzed Direct CH Amination of Benzamides with Aryl Azides: A Synthetic Route to Diarylamines
- (2012) Jaeyune Ryu et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Mild and Efficient C2-Alkenylation of Indoles with Alkynes Catalyzed by a Cobalt Complex
- (2012) Zhenhua Ding et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Beyond Directing Groups: Transition-Metal-Catalyzed CH Activation of Simple Arenes
- (2012) Nadine Kuhl et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- C2-Alkylation ofN-pyrimidylindole with vinylsilane via cobalt-catalyzed C–H bond activation
- (2012) Zhenhua Ding et al. Beilstein Journal of Organic Chemistry
- 2,5-Diketopiperazines: Synthesis, Reactions, Medicinal Chemistry, and Bioactive Natural Products
- (2012) Alan D. Borthwick CHEMICAL REVIEWS
- C–C, C–O and C–N bond formation via rhodium(iii)-catalyzed oxidative C–H activation
- (2012) Guoyong Song et al. CHEMICAL SOCIETY REVIEWS
- Elements of Regiocontrol in the Direct Heteroarylation of Indoles/Pyrroles: Synthesis of Bi- and Fused Polycyclic Heteroarenes by Twofold or Tandem Fourfold CH Activation
- (2012) Zhen Wang et al. CHEMISTRY-A EUROPEAN JOURNAL
- Amide-Directed Tandem CC/CN Bond Formation through CH Activation
- (2012) Chen Zhu et al. Chemistry-An Asian Journal
- Rh(III)-Catalyzed Regioselective Synthesis of Pyridines from Alkenes and α,β-Unsaturated Oxime Esters
- (2012) Jamie M. Neely et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Ir(I)-Catalyzed C–H Bond Alkylation of C2-Position of Indole with Alkenes: Selective Synthesis of Linear or Branched 2-Alkylindoles
- (2012) Shiguang Pan et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Rh-Catalyzed Intermolecular Carbenoid Functionalization of Aromatic C–H Bonds by α-Diazomalonates
- (2012) Wai-Wing Chan et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Rhodium(III)-Catalyzed N-Nitroso-Directed C–H Olefination of Arenes. High-Yield, Versatile Coupling under Mild Conditions
- (2012) Baoqing Liu et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Synthesis of pyrido[2,3-b]indoles and pyrimidoindoles via Pd-catalyzed amidation and cyclization
- (2012) Arepalli Sateesh Kumar et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- Rhodium-catalyzed regioselective amidation of indoles with sulfonyl azides via C–H bond activation
- (2012) Jingjing Shi et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- Rhodium-Catalyzed Oxidative Annulation of Sulfonylhydrazones with Alkenes
- (2012) Guifei Li et al. ORGANIC LETTERS
- Palladium-Assisted Regioselective C–H Cyanation of Heteroarenes Using Isonitrile as Cyanide Source
- (2012) Shuguang Xu et al. ORGANIC LETTERS
- Copper-Mediated Multiple C–H Functionalization of Aromatic N-Heterocycles: Bromoamination of Indoles and Pyrroles
- (2012) Alex John et al. ORGANOMETALLICS
- Couple Dynamics: PPARγ and Its Ligand Partners
- (2012) Shanghai Yu et al. STRUCTURE
- Rhodium(iii)-catalyzed synthesis of phthalides by cascade addition and cyclization of benzimidates with aldehydes
- (2012) Yajing Lian et al. Chemical Science
- Ruthenium-catalyzed direct oxidative alkenylation of arenes through twofold C–H bond functionalization
- (2012) Sergei I. Kozhushkov et al. Chemical Science
- Rhodium Catalyzed Chelation-Assisted C–H Bond Functionalization Reactions
- (2011) Denise A. Colby et al. ACCOUNTS OF CHEMICAL RESEARCH
- Weak Coordination as a Powerful Means for Developing Broadly Useful C–H Functionalization Reactions
- (2011) Keary M. Engle et al. ACCOUNTS OF CHEMICAL RESEARCH
- Catalytic Dehydrogenative Cross-Coupling: Forming Carbon−Carbon Bonds by Oxidizing Two Carbon−Hydrogen Bonds
- (2011) Charles S. Yeung et al. CHEMICAL REVIEWS
- Carboxylate-Assisted Transition-Metal-Catalyzed C−H Bond Functionalizations: Mechanism and Scope
- (2011) Lutz Ackermann CHEMICAL REVIEWS
- Towards mild metal-catalyzed C–H bond activation
- (2011) Joanna Wencel-Delord et al. CHEMICAL SOCIETY REVIEWS
- Recent advances in the transition metal-catalyzed twofold oxidative C–H bond activation strategy for C–C and C–N bond formation
- (2011) Seung Hwan Cho et al. CHEMICAL SOCIETY REVIEWS
- Identification and Mechanism of 10-Carbon Fatty Acid as Modulating Ligand of Peroxisome Proliferator-activated Receptors
- (2011) Raghu R. V. Malapaka et al. JOURNAL OF BIOLOGICAL CHEMISTRY
- Palladium-Catalyzed Direct 2-Alkylation of Indoles by Norbornene-Mediated Regioselective Cascade C–H Activation
- (2011) Lei Jiao et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Antidiabetic actions of a non-agonist PPARγ ligand blocking Cdk5-mediated phosphorylation
- (2011) Jang Hyun Choi et al. NATURE
- Synthesis of α-Carbolines via Pd-Catalyzed Amidation and Vilsmeier−Haack Reaction of 3-Acetyl-2-chloroindoles
- (2011) Arepalli Sateesh Kumar et al. ORGANIC LETTERS
- Palladium-/Copper-Catalyzed Regioselective Amination and Chloroamination of Indoles
- (2011) Xue-Yuan Liu et al. ORGANIC LETTERS
- Rhodium(III)-Catalyzed Intermolecular Direct Amination of Aromatic C–H Bonds with N-Chloroamines
- (2011) Ka-Ho Ng et al. ORGANIC LETTERS
- Ruthenium-Catalyzed Direct C–H Bond Arylations of Heteroarenes
- (2011) Lutz Ackermann et al. ORGANIC LETTERS
- Rh[III]-Catalyzed Direct C–H Amination Using N-Chloroamines at Room Temperature
- (2011) Christoph Grohmann et al. ORGANIC LETTERS
- “On Water” Direct and Site-Selective Pd-Catalysed CH Arylation of (NH)-Indoles
- (2010) Lionel Joucla et al. ADVANCED SYNTHESIS & CATALYSIS
- Copper-Catalyzed Highly Regioselective Oxidative CH Bond Amidation of 2-Arylpyridine Derivatives and 1-Methylindoles
- (2010) Qi Shuai et al. ADVANCED SYNTHESIS & CATALYSIS
- Marine Indole Alkaloids: Potential New Drug Leads for the Control of Depression and Anxiety
- (2010) Anna J. Kochanowska-Karamyan et al. CHEMICAL REVIEWS
- PdII-Catalysed CH Functionalisation of Indoles and Pyrroles Assisted by the Removable N-(2-Pyridyl)sulfonyl Group: C2-Alkenylation and Dehydrogenative Homocoupling
- (2010) Alfonso García-Rubia et al. CHEMISTRY-A EUROPEAN JOURNAL
- Palladium(II)-Catalyzed Regioselective Direct C2 Alkenylation of Indoles and Pyrroles Assisted by theN-(2-Pyridyl)sulfonyl Protecting Group
- (2009) Alfonso García-Rubia et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Facile Synthesis of Fluorinated Benzofuro- and Benzothieno[2,3-b]pyridines, α-Carbolines and Nucleosides Containing the α-Carboline Framework
- (2009) Viktor Iaroshenko et al. SYNTHESIS-STUTTGART
- Palladium-Catalyzed Direct Arylation of (Hetero)Arenes with Aryl Boronic Acids
- (2008) Shang-Dong Yang et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Rosiglitazone-Associated Fractures in Type 2 Diabetes: An analysis from A Diabetes Outcome Progression Trial (ADOPT)
- (2008) S. E. Kahn et al. DIABETES CARE
- Palladium-Catalyzed Direct C-2 Arylation of Indoles with Potassium Aryltrifluoroborate Salts
- (2008) Jinlong Zhao et al. JOURNAL OF ORGANIC CHEMISTRY
- Regioselective C−H Functionalization Directed by a Removable Carboxyl Group: Palladium-Catalyzed Vinylation at the Unusual Position of Indole and Related Heteroaromatic Rings
- (2008) Atsushi Maehara et al. ORGANIC LETTERS
- Copper-Catalyzed Cyclization of Iodo-tryptophans: A Straightforward Synthesis of Pyrroloindoles
- (2008) Alexis Coste et al. ORGANIC LETTERS
Find Funding. Review Successful Grants.
Explore over 25,000 new funding opportunities and over 6,000,000 successful grants.
ExploreBecome a Peeref-certified reviewer
The Peeref Institute provides free reviewer training that teaches the core competencies of the academic peer review process.
Get Started