Direct enantioselective access to 4-substituted tetrahydroquinolines by catalytic asymmetric transfer hydrogenation of quinolines

Phosphoric Acid-Catalyzed Enantioselective Transfer Hydrogenation of N-Aryl-ortho-Hydroxybenzophenone Ketimines

(2011) Thanh Binh Nguyen et al.   ADVANCED SYNTHESIS & CATALYSIS

Asymmetric Brønsted Acid-Catalyzed Friedel-Crafts Reactions of Indoles with Cyclic Imines - Efficient Generation of Nitrogen-Substituted Quaternary Carbon Centers

(2011) Magnus Rueping et al.   ADVANCED SYNTHESIS & CATALYSIS

Asymmetric Binary Acid Catalysis: A Regioselectivity Switch between Enantioselective 1,2- and 1,4-Addition through Different Counteranions of InIII

(2011) Jian Lv et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Modulating the Acidity: Highly Acidic Brønsted Acids in Asymmetric Catalysis

(2011) Magnus Rueping et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Brønsted Acid Catalysis: Hydrogen Bonding versus Ion Pairing in Imine Activation

(2011) Matthias Fleischmann et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Enantioselective N-H Functionalization of Indoles with α,β-Unsaturated γ-Lactams Catalyzed by Chiral Brønsted Acids

(2011) Yinjun Xie et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Chiral Brønsted acids in enantioselective carbonyl activations – activation modes and applications

(2011) Magnus Rueping et al.   CHEMICAL SOCIETY REVIEWS

Chiral Brønsted Acid-Promoted Enantioselective Desymmetrization in an Intramolecular Schmidt Reaction of Symmetric Azido 1,3-Hexanediones: Asymmetric Synthesis of Azaquaternary Pyrroloazepine Skeletons

(2011) Ming Yang et al.   Chemistry-An Asian Journal

Organocatalyzed Enantioselective Synthesis of Quaternary Carbon-Containing Isoindolin-1-ones

(2011) Xiaolei Yu et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Advances in catalytic metal-free reductions: from bio-inspired concepts to applications in the organocatalytic synthesis of pharmaceuticals and natural products

(2011) Magnus Rueping et al.   GREEN CHEMISTRY

Chiral Organic Contact Ion Pairs in Metal-Free Catalytic Asymmetric Allylic Substitutions

(2011) Magnus Rueping et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Selective Activation of Enantiotopic C(sp3)−Hydrogen by Means of Chiral Phosphoric Acid: Asymmetric Synthesis of Tetrahydroquinoline Derivatives

(2011) Keiji Mori et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Convergent Asymmetric Disproportionation Reactions: Metal/Brønsted Acid Relay Catalysis for Enantioselective Reduction of Quinoxalines

(2011) Qing-An Chen et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Chiral Phosphoric Acid Catalyzed Enantioselective Synthesis of β-Amino-α,α-difluoro Carbonyl Compounds

(2011) Wataru Kashikura et al.   ORGANIC LETTERS

Enantioselective Organocatalytic Synthesis of Quaternary α-Amino Acids Bearing a CF3Moiety

(2011) Ralph Husmann et al.   ORGANIC LETTERS

Chiral Brønsted Acids and Their Calcium Salts in Catalytic Asymmetric Mannich Reactions of Cyclic 1,3-Diketones

(2011) Magnus Rueping et al.   SYNLETT

Enantioselective Synthesis of Quinolizidines and Indolizidines via a Catalytic Asymmetric Hydrogenation Cascade

(2011) Magnus Rueping et al.   SYNLETT

Chiral phosphoric acid-catalysed Friedel–Crafts alkylation reaction of indoles with racemic spiro indolin-3-ones

(2011) Qin Yin et al.   Chemical Science

Diastereoselective Hydrogenation of Substituted Quinolines to Enantiomerically Pure Decahydroquinolines

(2010) Maja Heitbaum et al.   ADVANCED SYNTHESIS & CATALYSIS

Chiral Brønsted Acid-Catalyzed Enantioselective Friedel-Crafts Reaction of 4,7-Dihydroindoles with Trifluoromethyl Ketones

(2010) Teng Wang et al.   ADVANCED SYNTHESIS & CATALYSIS

First Highly Enantioselective Synthesis of Benzodiazepinones by Catalytic Hydrogenation

(2010) Magnus Rueping et al.   ADVANCED SYNTHESIS & CATALYSIS

Enantioselective Organocatalytic Transfer Hydrogenation of α-Imino Esters by Utilization of Benzothiazoline as Highly Efficient Reducing Agent

(2010) Chen Zhu et al.   ADVANCED SYNTHESIS & CATALYSIS

Chiral Phosphoric Acid Catalyzed Peroxidation of Imines

(2010) Wenhua Zheng et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic Asymmetric Reductive Amination of α-Branched Ketones

(2010) Vijay N. Wakchaure et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Chiral Phosphoric Acids as Versatile Catalysts for Enantioselective Carbon–Carbon Bond Forming Reactions

(2010) Masahiro Terada   BULLETIN OF THE CHEMICAL SOCIETY OF JAPAN

Brønsted acid differentiated metal catalysis by kinetic discrimination

(2010) Magnus Rueping et al.   CHEMICAL COMMUNICATIONS

Catalytic Asymmetric Mannich-Ketalization Reaction: Highly Enantioselective Synthesis of Aminobenzopyrans

(2010) Magnus Rueping et al.   CHEMISTRY-A EUROPEAN JOURNAL

The Brønsted Acid Catalyzed, Enantioselective Vinylogous Mannich Reaction

(2010) Marcel Sickert et al.   CHEMISTRY-A EUROPEAN JOURNAL

The First General, Efficient and Highly Enantioselective Reduction of Quinoxalines and Quinoxalinones

(2010) Magnus Rueping et al.   CHEMISTRY-A EUROPEAN JOURNAL

DFT Study of Chiral-Phosphoric-Acid-Catalyzed Enantioselective Friedel-Crafts Reaction of Indole with Nitroalkene: Bifunctionality and Substituent Effect of Phosphoric Acid

(2010) Takashi Hirata et al.   Chemistry-An Asian Journal

Desymmetrization of Cyclohexadienones via Brønsted Acid-Catalyzed Enantioselective Oxo-Michael Reaction

(2010) Qing Gu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Asymmetric organocatalysis in total synthesis – a trial by fire

(2010) Eugenia Marqués-López et al.   NATURAL PRODUCT REPORTS

Asymmetric Synthesis of Indolines by Catalytic Enantioselective Reduction of 3H-Indoles

(2010) Magnus Rueping et al.   ORGANIC LETTERS

Chiral Phosphoric Acid-Catalyzed Enantioselective Transfer Hydrogenation ofortho-Hydroxyaryl Alkyl N−H Ketimines

(2010) Thanh Binh Nguyen et al.   ORGANIC LETTERS

Thieme Chemistry Journal Awardees - Where Are They Now? Asymmetric Brønsted Acid Catalyzed Transfer Hydrogenations

(2010) Magnus Rueping et al.   SYNLETT

Chiral Phosphoric Acids as Versatile Catalysts for Enantioselective Transformations

(2010) Masahiro Terada   SYNTHESIS-STUTTGART

Asymmetric metal-free synthesis of fluoroquinolones by organocatalytic hydrogenation

(2010) Magnus Rueping et al.   TETRAHEDRON

Asymmetric Brønsted acid catalysis in aqueous solution

(2010) Magnus Rueping et al.   Chemical Science

A Catalytic Asymmetric Electrocyclization-Protonation Reaction

(2009) Magnus Rueping et al.   ADVANCED SYNTHESIS & CATALYSIS

Highly Efficient and Versatile Phosphine-Phosphoramidite Ligands for Asymmetric Hydrogenation

(2009) Matthias Eggenstein et al.   ADVANCED SYNTHESIS & CATALYSIS

Brønsted Acid Catalyzed Enantioselective Semipinacol Rearrangement for the Synthesis of Chiral Spiroethers

(2009) Qing-Wei Zhang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Brønsted Acid Catalyzed Enantioselective Three-Component Reaction Involving the α Addition of Isocyanides to Imines

(2009) Tao Yue et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Dynamic kinetic asymmetric transfer hydrogenation of racemic 2,4-diaryl-2,3-dihydrobenzo[b][1,4]diazepines catalyzed by chiral phosphoric acids

(2009) Zhi-Yong Han et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Unprecedented Halide Dependence on Catalytic Asymmetric Hydrogenation of 2-Aryl- and 2-Alkyl-Substituted Quinolinium Salts by Using Ir Complexes with Difluorphos and Halide Ligands

(2009) Hiroshi Tadaoka et al.   CHEMISTRY-A EUROPEAN JOURNAL

Highly enantioselective hydrogenation of quinolines under solvent-free or highly concentrated conditions

(2009) Zhi-Jian Wang et al.   GREEN CHEMISTRY

Chiral Brønsted Acid-Catalyzed Enantioselective α-Hydroxylation of β-Dicarbonyl Compounds

(2009) Min Lu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Enantioselective Brønsted Acid-CatalyzedN-Acyliminium Cyclization Cascades

(2009) Michael E. Muratore et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Organocatalytic Synthesis of Spiro[pyrrolidin-3,3′-oxindoles] with High Enantiopurity and Structural Diversity

(2009) Xiao-Hua Chen et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Consecutive Intramolecular Hydroamination/Asymmetric Transfer Hydrogenation under Relay Catalysis of an Achiral Gold Complex/Chiral Brønsted Acid Binary System

(2009) Zhi-Yong Han et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Benzothiazoline: Highly Efficient Reducing Agent for the Enantioselective Organocatalytic Transfer Hydrogenation of Ketimines

(2009) Chen Zhu et al.   ORGANIC LETTERS

Highly Enantioselective Hydrogenation of Enamides Catalyzed by Chiral Phosphoric Acids

(2009) Guilong Li et al.   ORGANIC LETTERS

Asymmetric Counterion Pair Catalysis: An Enantioselective Brønsted Acid-Catalyzed Protonation

(2008) Magnus Rueping et al.   ADVANCED SYNTHESIS & CATALYSIS

Synthesis of Sulfoximine-Derived P,N Ligands and their Applications in Asymmetric Quinoline Hydrogenations

(2008) Sheng-Mei Lu et al.   ADVANCED SYNTHESIS & CATALYSIS

Asymmetric Hydrogenation of Quinolines Catalyzed by Iridium Complexes of Monodentate BINOL-Derived Phosphoramidites

(2008) Nataša Mršić et al.   ADVANCED SYNTHESIS & CATALYSIS

Catalytic Asymmetric Aminoallylation of Aldehydes: A Catalytic Enantioselective Aza-Cope Rearrangement

(2008) Magnus Rueping et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Chiral Brønsted Acid Catalyzed Asymmetric Baeyer–Villiger Reaction of 3-Substituted Cyclobutanones by Using Aqueous H2O2

(2008) Senmiao Xu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Highly Enantioselective Organocatalytic Carbonyl-Ene Reaction with Strongly Acidic, Chiral Brønsted Acids as Efficient Catalysts

(2008) Magnus Rueping et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Asymmetric Brønsted Acid Catalyzed Isoindoline Synthesis: Enhancement of Enantiomeric Ratio by Stereoablative Kinetic Resolution

(2008) Dieter Enders et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

The Development of Double Axially Chiral Phosphoric Acids and Their Catalytic Transfer Hydrogenation of Quinolines

(2008) Qun-Sheng Guo et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Hydrogenation of Quinolines Using a Recyclable Phosphine-Free Chiral Cationic Ruthenium Catalyst: Enhancement of Catalyst Stability and Selectivity in an Ionic Liquid

(2008) Haifeng Zhou et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Asymmetric Brønsted Acid Catalysis: Catalytic Enantioselective Synthesis of Highly Biologically Active Dihydroquinazolinones

(2008) Magnus Rueping et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Highly enantioselective organocatalytic formation of a quaternary carbon center via chiral Brønsted acid catalyzed self-coupling of enamides

(2008) Christine Baudequin et al.   CHEMICAL COMMUNICATIONS

Binaphthol-derived phosphoric acid as a versatile catalyst for enantioselective carbon–carbon bond forming reactions

(2008) Masahiro Terada   CHEMICAL COMMUNICATIONS

Phosphoric Acid Catalyzed Enantioselective Transfer Hydrogenation of Imines: A Density Functional Theory Study of Reaction Mechanism and the Origins of Enantioselectivity

(2008) Tommaso Marcelli et al.   CHEMISTRY-A EUROPEAN JOURNAL

Broader, Greener, and More Efficient: Recent Advances in Asymmetric Transfer Hydrogenation

(2008) Chao Wang et al.   Chemistry-An Asian Journal

Theoretical Study of the Mechanism of Hantzsch Ester Hydrogenation of Imines Catalyzed by Chiral BINOL-Phosphoric Acids

(2008) Luis Simón et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Air-Stable and Phosphine-Free Iridium Catalysts for Highly Enantioselective Hydrogenation of Quinoline Derivatives†

(2008) Zhi-Wei Li et al.   ORGANIC LETTERS

Brønsted-Acid-Catalyzed Activation of Nitroalkanes: A Direct Enantioselective Aza-Henry Reaction

(2008) Magnus Rueping et al.   ORGANIC LETTERS

Asymmetric Transfer Hydrogenation of β,γ-Alkynyl α-Imino Esters by a Brønsted Acid

(2008) Qiang Kang et al.   ORGANIC LETTERS

Brønsted Acid Catalyzed Asymmetric Reduction of 2- and 2,9-Substituted 1,10-Phenanthrolines

(2008) Costa Metallinos et al.   SYNLETT