Catalytic Michael/Ring-Closure Reaction of α,β-Unsaturated Pyrazoleamides with Amidomalonates: Asymmetric Synthesis of (−)-Paroxetine
出版年份 2016 全文链接
标题
Catalytic Michael/Ring-Closure Reaction of α,β-Unsaturated Pyrazoleamides with Amidomalonates: Asymmetric Synthesis of (−)-Paroxetine
作者
关键词
-
出版物
CHEMISTRY-A EUROPEAN JOURNAL
Volume 22, Issue 42, Pages 15119-15124
出版商
Wiley
发表日期
2016-08-31
DOI
10.1002/chem.201603056
参考文献
相关参考文献
注意:仅列出部分参考文献,下载原文获取全部文献信息。- A ChiralN,N′-Dioxide-ZnIIComplex Catalyzes the Enantioselective [2+2] Cycloaddition of Alkynones with Cyclic Enol Silyl Ethers
- (2016) Tengfei Kang et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Chiral Nanoparticles/Lewis Acids as Cooperative Catalysts for Asymmetric 1,4-Addition of Arylboronic Acids to α,β-Unsaturated Amides
- (2016) Tomohiro Yasukawa et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Enantioselective Synthesis of Chiral Piperidines via the Stepwise Dearomatization/Borylation of Pyridines
- (2016) Koji Kubota et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Highly enantioselective Michael addition of malononitrile to α,β-unsaturated pyrazolamides catalyzed by a bifunctional thiourea
- (2016) Yuanqin Zheng et al. TETRAHEDRON
- Asymmetric [3 + 2] cycloaddition of donor–acceptor aziridines with aldehydes via carbon–carbon bond cleavage
- (2016) Yuting Liao et al. Chemical Science
- Regio- and Enantioselective Aza-Diels-Alder Reactions of 3-Vinylindoles: A Concise Synthesis of the Antimalarial Spiroindolone NITD609
- (2015) Haifeng Zheng et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Efficient Synthesis of Chiral Trisubstituted 1,2-Allenyl Ketones by Catalytic Asymmetric Conjugate Addition of Malonic Esters to Enynes
- (2015) Qian Yao et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- The asymmetric synthesis of polycyclic 3-spirooxindole alkaloids via the cascade reaction of 2-isocyanoethylindoles
- (2015) Xiaohu Zhao et al. CHEMICAL COMMUNICATIONS
- N,N′-Dioxide/Gadolinium(III)-Catalyzed Asymmetric Conjugate Addition of Nitroalkanes to α,β-Unsaturated Pyrazolamides
- (2015) Qian Yao et al. JOURNAL OF ORGANIC CHEMISTRY
- Enantioselective Synthesis of Carbo- and Heterocycles through a CuH-Catalyzed Hydroalkylation Approach
- (2015) Yi-Ming Wang et al. JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
- Unprecedented Hydrophobic Amplification in Noncovalent Organocatalysis “on Water”: Hydrophobic Chiral Squaramide Catalyzed Michael Addition of Malonates to Nitroalkenes
- (2015) Han Yong Bae et al. ACS Catalysis
- Asymmetric Synthesis of 2,3-Dihydropyrroles by Ring-Opening/Cyclization of Cyclopropyl Ketones Using Primary Amines
- (2014) Yong Xia et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Magnesium Complexes as Highly Effective Catalysts for Conjugate Cyanation of α,β-Unsaturated Amides and Ketones
- (2014) Jinlong Zhang et al. CHEMISTRY-A EUROPEAN JOURNAL
- Total Synthesis of (±)-Paroxetine by Diastereoconvergent Cobalt-Catalysed Arylation
- (2014) Carole F. Despiau et al. EUROPEAN JOURNAL OF ORGANIC CHEMISTRY
- Chiral N,N′-dioxide ligands: synthesis, coordination chemistry and asymmetric catalysis
- (2014) Xiaohua Liu et al. Organic Chemistry Frontiers
- Optically pure γ-butyrolactones and epoxy esters via two stereocentered HKR of 3-substituted epoxy esters: a formal synthesis of (−)-paroxetine, Ro 67-8867 and (+)-eldanolide
- (2013) Dattatray A. Devalankar et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- Organocatalytic asymmetric domino sulfa-Michael–aldol reactions of 2-mercaptobenzaldehyde with α,β-unsaturated N-acylpyrazoles for the construction of thiochromane
- (2012) Xiu-Qin Dong et al. CHEMICAL COMMUNICATIONS
- Asymmetric Synthesis of γ-Nitroesters by an Organocatalytic One-Pot Strategy
- (2012) Kim L. Jensen et al. ORGANIC LETTERS
- Rhodium/diene-catalyzed asymmetric arylation of N-Boc-protected α,β-unsaturated δ-lactam with arylboronic acids: enantioselective synthesis of 4-aryl-2-piperidinones
- (2012) Zhi-Tao He et al. TETRAHEDRON
- An enantiodivergent and formal synthesis of paroxetine enantiomers by asymmetric desymmetrization of 3-(4-fluorophenyl)glutaric anhydride with a chiral SuperQuat oxazolidin-2-one
- (2012) Narendra R. Chaubey et al. TETRAHEDRON-ASYMMETRY
- ChiralN,N′-Dioxides: New Ligands and Organocatalysts for Catalytic Asymmetric Reactions
- (2011) XiaoHua Liu et al. ACCOUNTS OF CHEMICAL RESEARCH
- Highly enantioselective organocatalytic cascade reaction for the synthesis of piperidines and oxazolidines
- (2011) Sylva Číhalová et al. TETRAHEDRON
- An efficient and stereoselective synthesis of (3S,4R)-(−)-trans-4-(4′-fluorophenyl)-3-hydroxymethyl-N-methylpiperidine
- (2011) Sripathi Somaiah et al. TETRAHEDRON-ASYMMETRY
- Synthesis of (−)-Paroxetine via Enantioselective Phase-Transfer Catalytic Monoalkylation of Malonamide Ester
- (2010) Mi-hyun Kim et al. ORGANIC LETTERS
- Highly enantioselective synthesis of 1,3-bis(hydroxymethyl)-2-oxindoles from unprotected oxindoles and formalin using a chiral NdIII complex
- (2010) Ke Shen et al. Chemical Science
- Nonlinear Effects in Asymmetric Catalysis
- (2009) Tummanapalli Satyanarayana et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Highly enantioselective organocatalytic synthesis of piperidines. Formal synthesis of (−)-Paroxetine
- (2009) Guillem Valero et al. TETRAHEDRON LETTERS
- Enantioseparation of Paroxetine Precursors by HPLC on Amylose and Tartardiamide‐Based Chiral Stationary Phases
- (2008) Zongbi Bao et al. JOURNAL OF LIQUID CHROMATOGRAPHY & RELATED TECHNOLOGIES
- Organocatalytic Asymmetric Total Synthesis of (R)-Rolipram and Formal Synthesis of (3S,4R)-Paroxetine
- (2008) Peter S. Hynes et al. ORGANIC LETTERS
- Enantioselective organocatalytic Michael addition of malonates to α,β-unsaturated aldehydes in water
- (2008) Anqi Ma et al. TETRAHEDRON LETTERS
- Recent advances in the stereoselective synthesis of trans-3,4-disubstituted-piperidines: applications to (−)-paroxetine
- (2008) Carmela De Risi et al. TETRAHEDRON-ASYMMETRY
Become a Peeref-certified reviewer
The Peeref Institute provides free reviewer training that teaches the core competencies of the academic peer review process.
Get StartedAsk a Question. Answer a Question.
Quickly pose questions to the entire community. Debate answers and get clarity on the most important issues facing researchers.
Get Started