Catalytic Michael/Ring-Closure Reaction of α,β-Unsaturated Pyrazoleamides with Amidomalonates: Asymmetric Synthesis of (−)-Paroxetine

A ChiralN,N′-Dioxide-ZnIIComplex Catalyzes the Enantioselective [2+2] Cycloaddition of Alkynones with Cyclic Enol Silyl Ethers

(2016) Tengfei Kang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Chiral Nanoparticles/Lewis Acids as Cooperative Catalysts for Asymmetric 1,4-Addition of Arylboronic Acids to α,β-Unsaturated Amides

(2016) Tomohiro Yasukawa et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Enantioselective Synthesis of Chiral Piperidines via the Stepwise Dearomatization/Borylation of Pyridines

(2016) Koji Kubota et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Highly enantioselective Michael addition of malononitrile to α,β-unsaturated pyrazolamides catalyzed by a bifunctional thiourea

(2016) Yuanqin Zheng et al.   TETRAHEDRON

Asymmetric [3 + 2] cycloaddition of donor–acceptor aziridines with aldehydes via carbon–carbon bond cleavage

(2016) Yuting Liao et al.   Chemical Science

Regio- and Enantioselective Aza-Diels-Alder Reactions of 3-Vinylindoles: A Concise Synthesis of the Antimalarial Spiroindolone NITD609

(2015) Haifeng Zheng et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Efficient Synthesis of Chiral Trisubstituted 1,2-Allenyl Ketones by Catalytic Asymmetric Conjugate Addition of Malonic Esters to Enynes

(2015) Qian Yao et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

The asymmetric synthesis of polycyclic 3-spirooxindole alkaloids via the cascade reaction of 2-isocyanoethylindoles

(2015) Xiaohu Zhao et al.   CHEMICAL COMMUNICATIONS

N,N′-Dioxide/Gadolinium(III)-Catalyzed Asymmetric Conjugate Addition of Nitroalkanes to α,β-Unsaturated Pyrazolamides

(2015) Qian Yao et al.   JOURNAL OF ORGANIC CHEMISTRY

Enantioselective Synthesis of Carbo- and Heterocycles through a CuH-Catalyzed Hydroalkylation Approach

(2015) Yi-Ming Wang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Unprecedented Hydrophobic Amplification in Noncovalent Organocatalysis “on Water”: Hydrophobic Chiral Squaramide Catalyzed Michael Addition of Malonates to Nitroalkenes

(2015) Han Yong Bae et al.   ACS Catalysis

Asymmetric Synthesis of 2,3-Dihydropyrroles by Ring-Opening/Cyclization of Cyclopropyl Ketones Using Primary Amines

(2014) Yong Xia et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Magnesium Complexes as Highly Effective Catalysts for Conjugate Cyanation of α,β-Unsaturated Amides and Ketones

(2014) Jinlong Zhang et al.   CHEMISTRY-A EUROPEAN JOURNAL

Total Synthesis of (±)-Paroxetine by Diastereoconvergent Cobalt-Catalysed Arylation

(2014) Carole F. Despiau et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Chiral N,N′-dioxide ligands: synthesis, coordination chemistry and asymmetric catalysis

(2014) Xiaohua Liu et al.   Organic Chemistry Frontiers

Optically pure γ-butyrolactones and epoxy esters via two stereocentered HKR of 3-substituted epoxy esters: a formal synthesis of (−)-paroxetine, Ro 67-8867 and (+)-eldanolide

(2013) Dattatray A. Devalankar et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Organocatalytic asymmetric domino sulfa-Michael–aldol reactions of 2-mercaptobenzaldehyde with α,β-unsaturated N-acylpyrazoles for the construction of thiochromane

(2012) Xiu-Qin Dong et al.   CHEMICAL COMMUNICATIONS

Asymmetric Synthesis of γ-Nitroesters by an Organocatalytic One-Pot Strategy

(2012) Kim L. Jensen et al.   ORGANIC LETTERS

Rhodium/diene-catalyzed asymmetric arylation of N-Boc-protected α,β-unsaturated δ-lactam with arylboronic acids: enantioselective synthesis of 4-aryl-2-piperidinones

(2012) Zhi-Tao He et al.   TETRAHEDRON

An enantiodivergent and formal synthesis of paroxetine enantiomers by asymmetric desymmetrization of 3-(4-fluorophenyl)glutaric anhydride with a chiral SuperQuat oxazolidin-2-one

(2012) Narendra R. Chaubey et al.   TETRAHEDRON-ASYMMETRY

ChiralN,N′-Dioxides: New Ligands and Organocatalysts for Catalytic Asymmetric Reactions

(2011) XiaoHua Liu et al.   ACCOUNTS OF CHEMICAL RESEARCH

Highly enantioselective organocatalytic cascade reaction for the synthesis of piperidines and oxazolidines

(2011) Sylva Číhalová et al.   TETRAHEDRON

An efficient and stereoselective synthesis of (3S,4R)-(−)-trans-4-(4′-fluorophenyl)-3-hydroxymethyl-N-methylpiperidine

(2011) Sripathi Somaiah et al.   TETRAHEDRON-ASYMMETRY

Synthesis of (−)-Paroxetine via Enantioselective Phase-Transfer Catalytic Monoalkylation of Malonamide Ester

(2010) Mi-hyun Kim et al.   ORGANIC LETTERS

Highly enantioselective synthesis of 1,3-bis(hydroxymethyl)-2-oxindoles from unprotected oxindoles and formalin using a chiral NdIII complex

(2010) Ke Shen et al.   Chemical Science

Nonlinear Effects in Asymmetric Catalysis

(2009) Tummanapalli Satyanarayana et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Highly enantioselective organocatalytic synthesis of piperidines. Formal synthesis of (−)-Paroxetine

(2009) Guillem Valero et al.   TETRAHEDRON LETTERS

Enantioseparation of Paroxetine Precursors by HPLC on Amylose and Tartardiamide‐Based Chiral Stationary Phases

(2008) Zongbi Bao et al.   JOURNAL OF LIQUID CHROMATOGRAPHY & RELATED TECHNOLOGIES

Organocatalytic Asymmetric Total Synthesis of (R)-Rolipram and Formal Synthesis of (3S,4R)-Paroxetine

(2008) Peter S. Hynes et al.   ORGANIC LETTERS

Enantioselective organocatalytic Michael addition of malonates to α,β-unsaturated aldehydes in water

(2008) Anqi Ma et al.   TETRAHEDRON LETTERS

Recent advances in the stereoselective synthesis of trans-3,4-disubstituted-piperidines: applications to (−)-paroxetine

(2008) Carmela De Risi et al.   TETRAHEDRON-ASYMMETRY