Enantioselective Synthesis of 3a-Amino-Pyrroloindolines by Copper-Catalyzed Direct Asymmetric Dearomative Amination of Tryptamines

Asymmetric Dearomatization of Indoles through a Michael/Friedel-Crafts-Type Cascade To Construct Polycyclic Spiroindolines

(2015) Xiaohu Zhao et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Enantioselective Arylative Dearomatization of Indoles via Pd-Catalyzed Intramolecular Reductive Heck Reactions

(2015) Chong Shen et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthesis of naked amino-pyrroloindoline via direct aminocyclization of tryptamine

(2015) Zhigao Shen et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Enantioselective and diastereoselective azo-coupling/iminium-cyclizations: a unified strategy for the total syntheses of (−)-psychotriasine and (+)-pestalazine B

(2015) Qi Li et al.   Chemical Science

Ligand-enabled Ir-catalyzed intermolecular diastereoselective and enantioselective allylic alkylation of 3-substituted indoles

(2015) Xiao Zhang et al.   Chemical Science

Transition-Metal-Catalyzed Asymmetric Allylic Dearomatization Reactions

(2014) Chun-Xiang Zhuo et al.   ACCOUNTS OF CHEMICAL RESEARCH

Highly Enantioselective [3+2] Coupling of Indoles with Quinone Monoimines Promoted by a Chiral Phosphoric Acid

(2014) Lihua Liao et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Chiral Anion Phase Transfer of Aryldiazonium Cations: An Enantioselective Synthesis of C3-Diazenated Pyrroloindolines

(2014) Hosea M. Nelson et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic Asymmetric Synthesis of [2,3]-Fused Indoline Heterocycles through Inverse-Electron-Demand Aza-Diels-Alder Reaction of Indoles with Azoalkenes

(2014) Min-Chao Tong et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Organocatalytic Asymmetric Arylative Dearomatization of 2,3-Disubstituted Indoles Enabled by Tandem Reactions

(2014) Yu-Chen Zhang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Metal-Free Enantioselective Electrophilic Activation of Allenamides: Stereoselective Dearomatization of Indoles

(2014) Ciro Romano et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Recent advances in dearomatization of heteroaromatic compounds

(2014) Qiuping Ding et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Construction of the N1–C3 Linkage Stereogenic Centers by Catalytic Asymmetric Amination Reaction of 3-Bromooxindoles with Indolines

(2014) Hailong Zhang et al.   ORGANIC LETTERS

Copper-Catalyzed Oxoazidation and Alkoxyazidation of Indoles

(2014) Hang Yin et al.   ORGANIC LETTERS

Direct Stereospecific Synthesis of Unprotected N-H and N-Me Aziridines from Olefins

(2014) Jawahar L. Jat et al.   SCIENCE

Recent Developments in the Catalytic, Asymmetric Construction of Pyrroloindolines Bearing All-Carbon Quaternary Stereocenters

(2013) Lindsay M. Repka et al.   JOURNAL OF ORGANIC CHEMISTRY

Catalytic Asymmetric Synthesis of Pyrroloindolines via a Rhodium(II)-Catalyzed Annulation of Indoles

(2013) Jillian E. Spangler et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Copper-Catalyzed Highly Enantioselective Cyclopentannulation of Indoles with Donor–Acceptor Cyclopropanes

(2013) Hu Xiong et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Application of diazene-directed fragment assembly to the total synthesis and stereochemical assignment of (+)-desmethyl-meso-chimonanthine and related heterodimeric alkaloids

(2013) Stephen P. Lathrop et al.   Chemical Science

Ir-catalyzed intermolecular asymmetric allylic dearomatization reaction of indoles

(2013) Xiao Zhang et al.   Chemical Science

Enantioselective Construction of Pyrroloindolines Catalyzed by Chiral Phosphoric Acids: Total Synthesis of (−)-Debromoflustramine B

(2012) Zuhui Zhang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic Asymmetric Dearomatization Reactions

(2012) Chun-Xiang Zhuo et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Makomotindoline from Makomotake, Zizania latifolia infected with Ustilago esculenta

(2012) Tomohiro Suzuki et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Elusive Metal-Free Primary Amination of Arylboronic Acids: Synthetic Studies and Mechanism by Density Functional Theory

(2012) Chen Zhu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Enantioselective Copper-Catalyzed Construction of Aryl Pyrroloindolines via an Arylation–Cyclization Cascade

(2012) Shaolin Zhu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Diastereoselective Intramolecular Carbamoylketene/Alkene [2 + 2] Cycloaddition: Enantioselective Access to Pyrrolidinoindoline Alkaloids

(2012) Takaaki Araki et al.   ORGANIC LETTERS

Total Synthesis Guided Structure Elucidation of (+)-Psychotetramine

(2011) Klement Foo et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Iridium-Catalyzed Intramolecular Asymmetric Allylic Dearomatization of Phenols

(2011) Qing-Feng Wu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Organocatalyzed Enantioselective Fluorocyclizations

(2011) Oscar Lozano et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Directed Heterodimerization: Stereocontrolled Assembly via Solvent-Caged Unsymmetrical Diazene Fragmentation

(2011) Mohammad Movassaghi et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Flustramine inspired synthesis and biological evaluation of pyrroloindoline triazole amides as novel inhibitors of bacterial biofilms

(2011) Cynthia Bunders et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Oxaziridine-Mediated Oxyamination of Indoles: An Approach to 3-Aminoindoles and Enantiomerically Enriched 3-Aminopyrroloindolines

(2010) Tamas Benkovics et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic Oxyamidation of Indoles

(2010) Stéphane Beaumont et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Determination of absolute configuration of trimeric indole alkaloid, psychotrimine, by first asymmetric total synthesis

(2010) Nobuaki Takahashi et al.   CHEMICAL COMMUNICATIONS

A New Dimeric Alkaloid from the Leaf of Psychotria calocarpa

(2010) Hua Zhou et al.   HELVETICA CHIMICA ACTA

The psychotrimine natural products have antibacterial activity against Gram-positive bacteria and act via membrane disruption

(2010) Mark A Schallenberger et al.   JOURNAL OF ANTIBIOTICS

Enantioselective Construction of Spiroindolenines by Ir-Catalyzed Allylic Alkylation Reactions

(2010) Qing-Feng Wu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Enantioselective Synthesis of Pyrroloindolines by a Formal [3 + 2] Cycloaddition Reaction

(2010) Lindsay M. Repka et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Scalable Total Syntheses ofN-Linked Tryptamine Dimers by Direct Indole−Aniline Coupling: Psychotrimine and Kapakahines B and F

(2010) Timothy Newhouse et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Concise total synthesis and structural revision of (+)-pestalazine B

(2010) Carlos Pérez-Balado et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Epidithiodiketopiperazines Block the Interaction between Hypoxia-inducible Factor-1α (HIF-1α) and p300 by a Zinc Ejection Mechanism

(2009) Kristina M. Cook et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Nine-Step Enantioselective Total Synthesis of (+)-Minfiensine

(2009) Spencer B. Jones et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Enantiospecific Total Syntheses of Kapakahines B and F

(2009) Timothy Newhouse et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Pestalazines and Pestalamides, Bioactive Metabolites from the Plant Pathogenic FungusPestalotiopsis theae

(2008) Gang Ding et al.   JOURNAL OF NATURAL PRODUCTS

Total Synthesis of (±)-Psychotrimine

(2008) Timothy Newhouse et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

First Total Synthesis of Trimeric Indole Alkaloid, Psychotrimine

(2007) Yohei Matsuda et al.   ORGANIC LETTERS