Synthesis of naked amino-pyrroloindoline via direct aminocyclization of tryptamine

Copper-Mediated Dimerization to Access 3a,3a′-Bispyrrolidinoindoline: Diastereoselective Synthesis of (+)-WIN 64821 and (−)-Ditryptophenaline

(2015) Kangjiang Liang et al.   ORGANIC LETTERS

Chiral Anion Phase Transfer of Aryldiazonium Cations: An Enantioselective Synthesis of C3-Diazenated Pyrroloindolines

(2014) Hosea M. Nelson et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Highly Asymmetric Bromocyclization of Tryptophol: Unexpected Accelerating Effect of DABCO-Derived Bromine Complex

(2014) Huan Liu et al.   ORGANIC LETTERS

Thionium-Based One-Pot Construction of Homo-/Heterodimeric Pyrroloindoline from Tryptamine

(2014) Masanori Tayu et al.   ORGANIC LETTERS

Direct Stereospecific Synthesis of Unprotected N-H and N-Me Aziridines from Olefins

(2014) Jawahar L. Jat et al.   SCIENCE

Highly Enantioselective Bromocyclization of Tryptamines and Its Application in the Synthesis of (−)-Chimonanthine

(2013) Weiqing Xie et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Stereoselective copper-catalyzed Chan–Lam–Evans N-arylation of glucosamines with arylboronic acids at room temperature

(2013) Alexandre Bruneau et al.   CHEMICAL COMMUNICATIONS

Nickel-catalyzed dimerization of pyrrolidinoindoline scaffolds: systematic access to chimonanthines, folicanthines and (+)-WIN 64821

(2013) Mitsuhiro Wada et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Organocatalytic Michael Addition of Indoles to Isatylidene-3-acetaldehydes: Application to the Formal Total Synthesis of (−)-Chimonanthine

(2013) Renrong Liu et al.   ORGANIC LETTERS

Application of diazene-directed fragment assembly to the total synthesis and stereochemical assignment of (+)-desmethyl-meso-chimonanthine and related heterodimeric alkaloids

(2013) Stephen P. Lathrop et al.   Chemical Science

Enantioselective Construction of Pyrroloindolines Catalyzed by Chiral Phosphoric Acids: Total Synthesis of (−)-Debromoflustramine B

(2012) Zuhui Zhang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic Asymmetric Total Synthesis of Chimonanthine, Folicanthine, and Calycanthine through Double Michael Reaction of Bisoxindole

(2012) Harunobu Mitsunuma et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Elusive Metal-Free Primary Amination of Arylboronic Acids: Synthetic Studies and Mechanism by Density Functional Theory

(2012) Chen Zhu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Diastereoselective Intramolecular Carbamoylketene/Alkene [2 + 2] Cycloaddition: Enantioselective Access to Pyrrolidinoindoline Alkaloids

(2012) Takaaki Araki et al.   ORGANIC LETTERS

Core-Structure-Oriented Asymmetric Organocatalytic Substitution of 3-Hydroxyoxindoles: Application in the Enantioselective Total Synthesis of (+)-Folicanthine

(2011) Chang Guo et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Structure, Bioactivity and Synthesis of Natural Products with Hexahydropyrrolo[2,3-b]indole

(2011) Pau Ruiz-Sanchis et al.   CHEMISTRY-A EUROPEAN JOURNAL

Directed Heterodimerization: Stereocontrolled Assembly via Solvent-Caged Unsymmetrical Diazene Fragmentation

(2011) Mohammad Movassaghi et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Oxaziridine-Mediated Oxyamination of Indoles: An Approach to 3-Aminoindoles and Enantiomerically Enriched 3-Aminopyrroloindolines

(2010) Tamas Benkovics et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic Oxyamidation of Indoles

(2010) Stéphane Beaumont et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Scalable Total Syntheses ofN-Linked Tryptamine Dimers by Direct Indole−Aniline Coupling: Psychotrimine and Kapakahines B and F

(2010) Timothy Newhouse et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

An Expeditious Synthesis of C(3)−N(1′) Heterodimeric Indolines

(2008) Vinson R. Espejo et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Total Synthesis of (±)-Psychotrimine

(2008) Timothy Newhouse et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

First Total Synthesis of Trimeric Indole Alkaloid, Psychotrimine

(2007) Yohei Matsuda et al.   ORGANIC LETTERS