An Enolate-Mediated Organocatalytic Azide-Ketone [3+2]-Cycloaddition Reaction: Regioselective High-Yielding Synthesis of Fully Decorated 1,2,3-Triazoles

Iridium-Catalyzed Intermolecular Azide-Alkyne Cycloaddition of Internal Thioalkynes under Mild Conditions

(2014) Shengtao Ding et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

An Organocatalytic Azide-Aldehyde [3+2] Cycloaddition: High-Yielding Regioselective Synthesis of 1,4-Disubstituted 1,2,3-Triazoles

(2014) Dhevalapally B. Ramachary et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A Metal-Free Three-Component Reaction for the Regioselective Synthesis of 1,4,5-Trisubstituted 1,2,3-Triazoles

(2014) Joice Thomas et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

An efficient one-pot strategy for the highly regioselective metal-free synthesis of 1,4-disubstituted-1,2,3-triazoles

(2014) Akbar Ali et al.   CHEMICAL COMMUNICATIONS

1,2,3-Triazole in Heterocyclic Compounds, Endowed with Biological Activity, through 1,3-Dipolar Cycloadditions

(2014) Antonino Lauria et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Direct access to 1,2,3-triazoles through organocatalytic 1,3-dipolar cycloaddition reaction of allyl ketones with azides

(2014) Wenjun Li et al.   GREEN CHEMISTRY

Synthesis and Evaluation of New Hsp90 Inhibitors Based on a 1,4,5-Trisubstituted 1,2,3-Triazole Scaffold

(2014) Maurizio Taddei et al.   JOURNAL OF MEDICINAL CHEMISTRY

Copper-Mediated Synthesis of 1,2,3-Triazoles fromN-Tosylhydrazones and Anilines

(2013) Zhengkai Chen et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A Metal-Free Multicomponent Cascade Reaction for the Regiospecific Synthesis of 1,5-Disubstituted 1,2,3-Triazoles

(2013) Guolin Cheng et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis and antiproliferative activity of conformationally restricted 1,2,3-triazole analogues of combretastatins in the sea urchin embryo model and against human cancer cell lines

(2013) Dmitry V. Demchuk et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Direct access to triazole-olefins through catalytic cycloaddition of azides to unsaturated aldehydes

(2013) Wenjun Li et al.   CHEMICAL COMMUNICATIONS

Organocatalytic Triazole Formation, Followed by Oxidative Aromatization: Regioselective Metal-Free Synthesis of Benzotriazoles

(2013) Dhevalapally B. Ramachary et al.   CHEMISTRY-A EUROPEAN JOURNAL

In Vivo Imaging of the Metabotropic Glutamate Receptor 1 (mGluR1) with Positron Emission Tomography: Recent Advance and Perspective

(2013) Songye Li et al.   CURRENT MEDICINAL CHEMISTRY

Organocatalytic Synthesis of (Arylselanyl)phenyl-1H-1,2,3-triazole-4-carboxamides by Cycloaddition between Azidophenyl Arylselenides and β-Oxo-amides

(2013) Natália Seus et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Organocatalytic 1,3-dipolar cycloaddition reactions of ketones and azides with water as a solvent

(2013) Dwun Kit Jonathan Yeung et al.   GREEN CHEMISTRY

Iridium-Catalyzed Cycloaddition of Azides and 1-Bromoalkynes at Room Temperature

(2013) Evelia Rasolofonjatovo et al.   ORGANIC LETTERS

Regioselective Rapid Synthesis of Fully Substituted 1,2,3-Triazoles Mediated by Propargyl Cations

(2013) Huan Zhang et al.   ORGANIC LETTERS

Zinc Mediated Azide–Alkyne Ligation to 1,5- and 1,4,5-Substituted 1,2,3-Triazoles

(2013) Christopher D. Smith et al.   ORGANIC LETTERS

Functionalization of 5-telluro-1,2,3-triazoles: Te/Li exchange and Suzuki–Miyaura cross-coupling reaction

(2013) Hélio A. Stefani et al.   TETRAHEDRON LETTERS

Amine-Catalyzed [3+2] Huisgen Cycloaddition Strategy for the Efficient Assembly of Highly Substituted 1,2,3-Triazoles

(2012) Lei Wang et al.   CHEMISTRY-A EUROPEAN JOURNAL

Synthesis and Computational Analysis of Densely Functionalized Triazoles Using o-Nitrophenylalkynes

(2012) Melissa L. McIntosh et al.   JOURNAL OF ORGANIC CHEMISTRY

Moderating Strain without Sacrificing Reactivity: Design of Fast and Tunable Noncatalyzed Alkyne–Azide Cycloadditions via Stereoelectronically Controlled Transition State Stabilization

(2012) Brian Gold et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

[3 + 2]-Dipolar Cycloaddition Reactions of an N-Heterocyclic Carbene Boryl Azide

(2012) Everett Merling et al.   ORGANIC LETTERS

Copper-Catalysed Multicomponent Click Synthesis of 5-Alkynyl 1,2,3-Triazoles under Ambient Conditions

(2012) Francisco Alonso et al.   SYNLETT

Synthesis of arylselanyl-1H-1,2,3-triazole-4-carboxylates by organocatalytic cycloaddition of azidophenyl arylselenides with β-keto-esters

(2012) Natália Seus et al.   TETRAHEDRON

Organocatalytic Synthesis of 1,2,3-Triazoles from Unactivated Ketones and Arylazides

(2011) Mokhtaria Belkheira et al.   CHEMISTRY-A EUROPEAN JOURNAL

Organocatalytic Enamide-Azide Cycloaddition Reactions: Regiospecific Synthesis of 1,4,5-Trisubstituted-1,2,3-Triazoles

(2011) Lee Jin Tu Danence et al.   CHEMISTRY-A EUROPEAN JOURNAL

Click Chemistry: 1,2,3-Triazoles as Pharmacophores

(2011) Sandip G. Agalave et al.   Chemistry-An Asian Journal

Synthesis and Antimalarial Activities of a Diverse Set of Triazole-Containing Furamidine Analogues

(2011) Olivier Berger et al.   ChemMedChem

Scope and regioselectivity of the 1,3-dipolar cycloaddition of azides with methyl 2-perfluoroalkynoates for an easy, metal-free route to perfluoroalkylated 1,2,3-triazoles

(2011) Jiamei Wei et al.   JOURNAL OF FLUORINE CHEMISTRY

Synthesis and evaluation of 6-[1-(2-[18F]fluoro-3-pyridyl)-5-methyl-1H-1,2,3-triazol-4-yl]quinoline for positron emission tomography imaging of the metabotropic glutamate receptor type 1 in brain

(2010) Masayuki Fujinaga et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Cu-free click cycloaddition reactions in chemical biology

(2010) John C. Jewett et al.   CHEMICAL SOCIETY REVIEWS

Zn/C-Catalyzed Cycloaddition of Azides and Aryl Alkynes

(2010) Xu Meng et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Transition-Metal-Free Catalytic Synthesis of 1,5-Diaryl-1,2,3-triazoles

(2010) Sen W. Kwok et al.   ORGANIC LETTERS

Intramolecular Azide-Alkyne [3+2] Cycloaddition: A Versatile Route for the Synthesis of 1,2,3-Triazole Fused Dibenzo[1,5]diazocine Derivatives

(2010) K. Majumdar et al.   SYNTHESIS-STUTTGART

Copper-Catalyzed Azide-Alkyne Cycloaddition: Regioselective Synthesis of 1,4,5-Trisubstituted 1,2,3-Triazoles

(2009) Christian Spiteri et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Copper(I)-Catalyzed Cycloaddition of Organic Azides and 1-Iodoalkynes

(2009) Jason E. Hein et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Discovery and biological profile of isoindolinone derivatives as novel metabotropic glutamate receptor 1 antagonists: A potential treatment for psychotic disorders

(2009) Satoru Ito et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Copper(I)-Catalyzed Direct Arylation of 1,4-Disubstituted 1,2,3-Triazoles with Aryl Iodides

(2009) Shin-ichi Fukuzawa et al.   HETEROCYCLES

Efficient Synthesis of 1,4-Diaryl-5-methyl-1,2,3-triazole, A Potential mGluR1 Antagonist, and the Risk Assessment Study of Arylazides

(2009) Takayuki Tsuritani et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Efficient construction of therapeutics, bioconjugates, biomaterials and bioactive surfaces using azide–alkyne “click” chemistry☆

(2008) J LUTZ et al.   ADVANCED DRUG DELIVERY REVIEWS

Palladium-Catalyzed Direct Arylations of Heteroarenes with Tosylates and Mesylates

(2008) Lutz Ackermann et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Discovery and biological profile of 4-(1-aryltriazol-4-yl)-tetrahydropyridines as an orally active new class of metabotropic glutamate receptor 1 antagonist

(2008) Satoru Ito et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Amino Acid-Catalyzed Cascade [3+2]-Cycloaddition/Hydrolysis Reactions Based on the Push-Pull Dienamine Platform: Synthesis of Highly FunctionalizedNH-1,2,3-Triazoles

(2008) Dhevalapally B. Ramachary et al.   CHEMISTRY-A EUROPEAN JOURNAL

Ruthenium-Catalyzed Azide−Alkyne Cycloaddition: Scope and Mechanism

(2008) Brant C. Boren et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Copper-Catalyzed “Click” Reaction/Direct Arylation Sequence: Modular Syntheses of 1,2,3-Triazoles

(2008) Lutz Ackermann et al.   ORGANIC LETTERS