An efficient one-pot strategy for the highly regioselective metal-free synthesis of 1,4-disubstituted-1,2,3-triazoles

Iridium-Catalyzed Intermolecular Azide-Alkyne Cycloaddition of Internal Thioalkynes under Mild Conditions

(2014) Shengtao Ding et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Beyond click chemistry – supramolecular interactions of 1,2,3-triazoles

(2014) Benjamin Schulze et al.   CHEMICAL SOCIETY REVIEWS

Direct access to 1,2,3-triazoles through organocatalytic 1,3-dipolar cycloaddition reaction of allyl ketones with azides

(2014) Wenjun Li et al.   GREEN CHEMISTRY

Ce(OTf)3-Catalyzed [3 + 2] Cycloaddition of Azides with Nitroolefins: Regioselective Synthesis of 1,5-Disubstituted 1,2,3-Triazoles

(2014) Ying-Chun Wang et al.   JOURNAL OF ORGANIC CHEMISTRY

Regioselectivity of Vinyl Sulfone Based 1,3-Dipolar Cycloaddition Reactions with Sugar Azides by Computational and Experimental Studies

(2014) Debashis Sahu et al.   ORGANIC LETTERS

A general route to 1,5-disubstituted 1,2,3-triazoles with alkyl/alkyl, alkyl/aryl, aryl/aryl combinations: a metal-free, regioselective, one-pot three component approach

(2014) Santu Dey et al.   RSC Advances

A Metal-Free Multicomponent Cascade Reaction for the Regiospecific Synthesis of 1,5-Disubstituted 1,2,3-Triazoles

(2013) Guolin Cheng et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Direct access to triazole-olefins through catalytic cycloaddition of azides to unsaturated aldehydes

(2013) Wenjun Li et al.   CHEMICAL COMMUNICATIONS

Ln[N(SiMe3)2]3-catalyzed cycloaddition of terminal alkynes to azides leading to 1,5-disubstituted 1,2,3-triazoles: new mechanistic features

(2013) Longcheng Hong et al.   CHEMICAL COMMUNICATIONS

Click Chemistry for Drug Development and Diverse Chemical–Biology Applications

(2013) Prakasam Thirumurugan et al.   CHEMICAL REVIEWS

Organocatalytic Triazole Formation, Followed by Oxidative Aromatization: Regioselective Metal-Free Synthesis of Benzotriazoles

(2013) Dhevalapally B. Ramachary et al.   CHEMISTRY-A EUROPEAN JOURNAL

Efficient TMG catalyzed synthesis of 1,2,3-triazoles

(2013) Fereshteh Ahmadi et al.   COMPTES RENDUS CHIMIE

Organocatalytic Synthesis of (Arylselanyl)phenyl-1H-1,2,3-triazole-4-carboxamides by Cycloaddition between Azidophenyl Arylselenides and β-Oxo-amides

(2013) Natália Seus et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

A Convenient Route to 1-Alkyl-5-trifluoromethyl-1,2,3-triazole-4-carboxylic Acids Employing a Diazo Transfer Reaction

(2013) Rustam T. Iminov et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Organocatalytic 1,3-dipolar cycloaddition reactions of ketones and azides with water as a solvent

(2013) Dwun Kit Jonathan Yeung et al.   GREEN CHEMISTRY

1,5-Disubstituted 1,2,3-Triazolylation at C1, C2, C3, C4, and C6 of Pyranosides: A Metal-Free Route to Triazolylated Monosaccharides and Triazole-Linked Disaccharides

(2013) Anirban Kayet et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of Densely Functionalized 3a,4-Dihydro-1H-Pyrrolo[1,2-b]Pyrazoles via Base Mediated Domino Reaction of Vinyl Malononitriles with 1,2-Diaza-1,3-dienes

(2013) Orazio A. Attanasi et al.   ORGANIC LETTERS

Zinc Mediated Azide–Alkyne Ligation to 1,5- and 1,4,5-Substituted 1,2,3-Triazoles

(2013) Christopher D. Smith et al.   ORGANIC LETTERS

The CuI-catalyzed alkyne–azide cycloaddition as direct conjugation/cyclization method of peptides to steroids

(2013) Radell Echemendía et al.   TETRAHEDRON

Synthesis of biologically as well as industrially important 1,4,5-trisubstituted-1,2,3-triazoles using a highly efficient, green and recyclable DBU–H2O catalytic system

(2013) Harjinder Singh et al.   RSC Advances

Traceless Tosylhydrazone-Based Triazole Formation: A Metal-Free Alternative to Strain-Promoted Azide-Alkyne Cycloaddition

(2012) Sander S. van Berkel et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Amine-Catalyzed [3+2] Huisgen Cycloaddition Strategy for the Efficient Assembly of Highly Substituted 1,2,3-Triazoles

(2012) Lei Wang et al.   CHEMISTRY-A EUROPEAN JOURNAL

Synthesis of arylselanyl-1H-1,2,3-triazole-4-carboxylates by organocatalytic cycloaddition of azidophenyl arylselenides with β-keto-esters

(2012) Natália Seus et al.   TETRAHEDRON

Bioconjugation with Strained Alkenes and Alkynes

(2011) Marjoke F. Debets et al.   ACCOUNTS OF CHEMICAL RESEARCH

Organocatalytic Synthesis of 1,2,3-Triazoles from Unactivated Ketones and Arylazides

(2011) Mokhtaria Belkheira et al.   CHEMISTRY-A EUROPEAN JOURNAL

Organocatalytic Enamide-Azide Cycloaddition Reactions: Regiospecific Synthesis of 1,4,5-Trisubstituted-1,2,3-Triazoles

(2011) Lee Jin Tu Danence et al.   CHEMISTRY-A EUROPEAN JOURNAL

Click Chemistry: 1,2,3-Triazoles as Pharmacophores

(2011) Sandip G. Agalave et al.   Chemistry-An Asian Journal

Tandem Catalysis: From Alkynoic Acids and Aryl Iodides to 1,2,3-Triazoles in One Pot

(2011) Andrej Kolarovič et al.   JOURNAL OF ORGANIC CHEMISTRY

Selective Formation of 1,5-Substituted Sulfonyl Triazoles Using Acetylides and Sulfonyl Azides

(2011) Maria Elena Meza-Aviña et al.   ORGANIC LETTERS

Regioselective synthesis of 5-trifluoromethyl-1,2,3-triazoles via CF3-directed cyclization of 1-trifluoromethyl-1,3-dicarbonyl compounds with azides

(2011) Yury A. Rozin et al.   TETRAHEDRON

Advances in metal-induced oxidative stress and human disease

(2011) Klaudia Jomova et al.   TOXICOLOGY

Cyclative Cleavage through Dipolar Cycloaddition: Polymer-Bound Azidopeptidylphosphoranes Deliver Locked cis-Triazolylcyclopeptides as Privileged Protein Binders

(2010) Ahsanullah et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

In situ click chemistry: probing the binding landscapes of biological molecules

(2010) Sreeman K. Mamidyala et al.   CHEMICAL SOCIETY REVIEWS

Tricks with clicks: modification of peptidomimetic oligomers via copper-catalyzed azide-alkyne [3 + 2] cycloaddition

(2010) Justin M. Holub et al.   CHEMICAL SOCIETY REVIEWS

Copper-catalyzed azide–alkyne cycloaddition (CuAAC) and beyond: new reactivity of copper(i) acetylides

(2010) Jason E. Hein et al.   CHEMICAL SOCIETY REVIEWS

Click polymerization

(2010) Anjun Qin et al.   CHEMICAL SOCIETY REVIEWS

Cu-free click cycloaddition reactions in chemical biology

(2010) John C. Jewett et al.   CHEMICAL SOCIETY REVIEWS

Experimental Evidence for the Involvement of Dinuclear Alkynylcopper(I) Complexes in Alkyne-Azide Chemistry

(2010) Benjamin R. Buckley et al.   CHEMISTRY-A EUROPEAN JOURNAL

Transition-Metal-Free Catalytic Synthesis of 1,5-Diaryl-1,2,3-triazoles

(2010) Sen W. Kwok et al.   ORGANIC LETTERS

Highly efficient and safe procedure for the synthesis of aryl 1,2,3-triazoles from aromatic amine in a continuous flow reactor

(2010) Federica Stazi et al.   TETRAHEDRON LETTERS

Metal-Free, Regioselective Triazole Ligations that Deliver LockedcisPeptide Mimetics

(2009) Ahsanullah et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

α,α-Dicyanoalkenes: versatile vinylogous nucleophiles for organic synthesis

(2009) Hai-Lei Cui et al.   CHEMICAL COMMUNICATIONS

Aza-dibenzocyclooctynes for fast and efficient enzyme PEGylation via copper-free (3+2) cycloaddition

(2009) Marjoke F. Debets et al.   CHEMICAL COMMUNICATIONS

Marrying click chemistry with polymerization: expanding the scope of polymeric materials

(2009) Patricia L. Golas et al.   CHEMICAL SOCIETY REVIEWS

Surpassing the Use of Copper in the Click Functionalization of Polymeric Nanostructures: A Strain-Promoted Approach

(2009) Enrique Lallana et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Copper-Free Azide–Alkyne Cycloadditions: New Insights and Perspectives

(2008) Jean-François Lutz   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Visualizing Metabolically Labeled Glycoconjugates of Living Cells by Copper-Free and Fast Huisgen Cycloadditions

(2008) Xinghai Ning et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Cu-Catalyzed Azide−Alkyne Cycloaddition

(2008) Morten Meldal et al.   CHEMICAL REVIEWS

Amino Acid-Catalyzed Cascade [3+2]-Cycloaddition/Hydrolysis Reactions Based on the Push-Pull Dienamine Platform: Synthesis of Highly FunctionalizedNH-1,2,3-Triazoles

(2008) Dhevalapally B. Ramachary et al.   CHEMISTRY-A EUROPEAN JOURNAL

Click Chemistry and Medicinal Chemistry: A Case of “Cyclo-Addiction”

(2008) A. D. Moorhouse et al.   ChemMedChem

Theory of 1,3-Dipolar Cycloadditions: Distortion/Interaction and Frontier Molecular Orbital Models

(2008) Daniel H. Ess et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

A Hydrophilic Azacyclooctyne for Cu-Free Click Chemistry

(2008) Ellen M. Sletten et al.   ORGANIC LETTERS

Click chemistry reactions in medicinal chemistry: Applications of the 1,3-dipolar cycloaddition between azides and alkynes

(2007) Gian Cesare Tron et al.   MEDICINAL RESEARCH REVIEWS