Enantioselective Synthesis of Tetrahydrocarbazoles through a Michael Addition/Ciamician-Plancher Rearrangement Sequence: Asymmetric Synthesis of a Potent Constrained Analogue of MS-245

Gold-Catalysis: Highly Efficient and Regio-Selective Carbonyl Migration in Alkynyl-Substituted Indole-3-Carboxamides Leading to Azepino[3,4-b]indol-1-ones

(2012) A. Stephen K. Hashmi et al.   ADVANCED SYNTHESIS & CATALYSIS

Recent Developments in Asymmetric Organocatalytic Domino Reactions

(2012) Hélène Pellissier   ADVANCED SYNTHESIS & CATALYSIS

Enantioselective Synthesis of Spiro Cyclopentane-1,3′-indoles and 2,3,4,9-Tetrahydro-1H-carbazoles by Iridium-Catalyzed Allylic Dearomatization and Stereospecific Migration

(2012) Qing-Feng Wu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A concise route to indoloazocines via a sequential Ugi–gold-catalyzed intramolecular hydroarylation

(2012) Sachin G. Modha et al.   CHEMICAL COMMUNICATIONS

Indoles in Multicomponent Processes (MCPs)

(2012) Morteza Shiri   CHEMICAL REVIEWS

Gold(I)-Catalyzed Rearrangement of 3-Silyloxy-1,5-enynes: An Efficient Synthesis of Benzo[b]thiophenes, Dibenzothiophenes, Dibenzofurans, and Indole Derivatives

(2012) A. Stephen K. Hashmi et al.   CHEMISTRY-A EUROPEAN JOURNAL

Merging Organocatalysis and Gold Catalysis-A Critical Evaluation of the Underlying Concepts

(2012) Charles C. J. Loh et al.   CHEMISTRY-A EUROPEAN JOURNAL

Evolution of asymmetric organocatalysis: multi- and retrocatalysis

(2012) Raffael C. Wende et al.   GREEN CHEMISTRY

Organocatalyzed Enantioselective Formal [4 + 2] Cycloaddition of 2,3-Disubstituted Indole and Methyl Vinyl Ketone

(2012) Quan Cai et al.   ORGANIC LETTERS

Enantioselective Gold-Catalyzed Synthesis of Polycyclic Indolines

(2012) Gianpiero Cera et al.   ORGANIC LETTERS

Multicatalytic Asymmetric Synthesis of Complex Tetrahydrocarbazoles via a Diels–Alder/Benzoin Reaction Sequence

(2012) Yankai Liu et al.   ORGANIC LETTERS

The Serotonin-6 Receptor as a Novel Therapeutic Target

(2012) Hyung-Mun Yun et al.   Experimental Neurobiology

Organocatalytic Multiple Cascade Reactions: A New Strategy for the Construction of Enantioenriched Tetrahydrocarbazoles

(2011) Yi-Ju Cao et al.   ADVANCED SYNTHESIS & CATALYSIS

Organocatalyzed Dynamic Kinetic Resolution

(2011) Hélène Pellissier   ADVANCED SYNTHESIS & CATALYSIS

One-Pot Reactions Accelerate the Synthesis of Active Pharmaceutical Ingredients

(2011) Carine Vaxelaire et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Enantioselective Michael/Mannich Polycyclization Cascade of Indolyl Enones Catalyzed by Quinine-Derived Primary Amines

(2011) Quan Cai et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Exploiting the Electrophilic Properties of Indole Intermediates: New Options in Designing Asymmetric Reactions

(2011) Charles C. J. Loh et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Direct Asymmetric Hydrosilylation of Indoles: Combined Lewis Base and Brønsted Acid Activation

(2011) You-Cai Xiao et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A Simple Recipe for Sophisticated Cocktails: Organocatalytic One-Pot Reactions-Concept, Nomenclature, and Future Perspectives

(2011) Łukasz Albrecht et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

The Pictet-Spengler Reaction in Nature and in Organic Chemistry

(2011) Joachim Stöckigt et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Stereoselective synthesis of tetracyclic indolines via gold-catalyzed cascade cyclization reactions

(2011) Gianpiero Cera et al.   CHEMICAL COMMUNICATIONS

Low-loading asymmetric organocatalysis

(2011) Francesco Giacalone et al.   CHEMICAL SOCIETY REVIEWS

Merging Organocatalysis and Gold Catalysis: Enantioselective Synthesis of Tetracyclic Indole Derivatives through a Sequential Double Friedel-Crafts Type Reaction

(2011) Charles C. J. Loh et al.   CHEMISTRY-A EUROPEAN JOURNAL

An Enantioselective Approach to 2,3-Disubstituted Indolines through Consecutive Brønsted Acid/Pd-Complex-Promoted Tandem Reactions

(2011) Ying Duan et al.   CHEMISTRY-A EUROPEAN JOURNAL

Enhanced Efficiency of Thiourea Catalysts by External Brønsted Acids in the Friedel-Crafts Alkylation of Indoles

(2011) Eugenia Marqués-López et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

One-Pot Synthesis of Indole-Fused Scaffolds via Gold-Catalyzed Tandem Annulation Reactions of 1,2-Bis(alkynyl)-2-en-1-ones with Indoles

(2011) Xin Xie et al.   JOURNAL OF ORGANIC CHEMISTRY

Asymmetric Catalysis of Diels–Alder Reactions with in Situ Generated Heterocyclicortho-Quinodimethanes

(2011) Yankai Liu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Redox-Neutral Indole Annulation Cascades

(2011) Michael C. Haibach et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

The Catalytic Asymmetric Fischer Indolization

(2011) Steffen Müller et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

A one-pot catalysis: the strategic classification with some recent examples

(2011) Nitin T. Patil et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Dehydration triggered asymmetric hydrogenation of 3-(α-hydroxyalkyl)indoles

(2011) Duo-Sheng Wang et al.   Chemical Science

A Practical and Enantioselective Approach to Tetrahydrocarbazoles by Asymmetric Organocatalysis

(2010) Xiao-Yu Zhu et al.   ChemCatChem

Creating Chemical Diversity in Indole Compounds by Merging Au and Ru Catalysis

(2010) Marco Bandini et al.   ChemCatChem

Mechanisms in aminocatalysis

(2010) Martin Nielsen et al.   CHEMICAL COMMUNICATIONS

Organocatalytic strategies for the asymmetric functionalization of indoles

(2010) Giuseppe Bartoli et al.   CHEMICAL SOCIETY REVIEWS

The Enantioselective, Organocatalyzed Diels-Alder Reaction of 2-Vinylindoles with α,β-Unsaturated Aldehydes: An Efficient Route to Functionalized Tetrahydrocarbazoles

(2010) Changwu Zheng et al.   CHEMISTRY-A EUROPEAN JOURNAL

Highly Efficient Route to Functionalized Tetrahydrocarbazoles Using a Tandem Cross-Metathesis/Intramolecular-Hydroarylation Sequence

(2010) Xiao-Lei An et al.   Chemistry-An Asian Journal

Recent Advances in Multicatalyst Promoted Asymmetric Tandem Reactions

(2010) Jian Zhou   Chemistry-An Asian Journal

Rapid and General Protocol towards Catalyst-Free Friedel-Crafts C-Alkylation of Indoles in Water Assisted by Microwave Irradiation

(2010) Margherita De Rosa et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Organocatalyzed Asymmetric Friedel-Crafts Reactions

(2010) Vincent Terrasson et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Pd-Catalyzed Asymmetric Hydrogenation of Unprotected Indoles Activated by Brønsted Acids

(2010) Duo-Sheng Wang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Organocatalytic cascade reactions as a new tool in total synthesis

(2010) Christoph Grondal et al.   Nature Chemistry

An Enantioselective Approach to Highly Substituted Tetrahydrocarbazoles through Hydrogen Bonding-Catalyzed Cascade Reactions

(2010) Xu-Fan Wang et al.   ORGANIC LETTERS

Cinchona Alkaloids in Asymmetric Organocatalysis

(2010) Tommaso Marcelli et al.   SYNTHESIS-STUTTGART

Gold-Catalyzed Intermolecular Reactions of (Z)-Enynols with Indoles for the Construction of Dihydrocyclohepta[b]indole Skeletons through a Cascade Friedel-Crafts/Hydroarylation Sequence

(2009) Yuhua Lu et al.   ADVANCED SYNTHESIS & CATALYSIS

Enantioselective Gold-Catalyzed Allylic Alkylation of Indoles with Alcohols: An Efficient Route to Functionalized Tetrahydrocarbazoles

(2009) Marco Bandini et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Catalytic Functionalization of Indoles in a New Dimension

(2009) Marco Bandini et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Chiral Brønsted acid catalyzed Friedel–Crafts alkylation reactions

(2009) Shu-Li You et al.   CHEMICAL SOCIETY REVIEWS

Organocatalysis—after the gold rush

(2009) Søren Bertelsen et al.   CHEMICAL SOCIETY REVIEWS

Organocatalytic Formation of Quaternary Stereocenters

(2009) Marco Bella et al.   SYNTHESIS-STUTTGART

Enantioselective Organocatalytic Diels-Alder Reactions

(2009) Pedro Merino et al.   SYNTHESIS-STUTTGART

Synthesis of the tetracyclic core skeleton of the lundurines by a gold-catalyzed cyclization

(2009) Catalina Ferrer et al.   TETRAHEDRON

Chiral Phosphoric Acid Catalyzed Enantioselective Friedel–Crafts Alkylation of Indoles with Nitroalkenes: Cooperative Effect of 3 Å Molecular Sieves

(2008) Junji Itoh et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Organocatalytic Asymmetric Diels-Alder Reactions of 3-Vinylindoles

(2008) Claudio Gioia et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Asymmetric Aminocatalysis-Gold Rush in Organic Chemistry

(2008) Paolo Melchiorre et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Asymmetric Organocatalysis: From Infancy to Adolescence

(2008) Alessandro Dondoni et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A Highly Strained Planar-Chiral Platinacycle for Catalytic Activation of Internal Olefins in the Friedel-Crafts Alkylation of Indoles

(2008) Haoxi Huang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Serotonin Receptors

(2008) David E. Nichols et al.   CHEMICAL REVIEWS

Catalytic Asymmetric Friedel−Crafts Alkylation ReactionsCopper Showed the Way

(2008) Thomas B. Poulsen et al.   CHEMICAL REVIEWS

Binding of Serotonin and N1-Benzenesulfonyltryptamine-Related Analogs at Human 5-HT6Serotonin Receptors: Receptor Modeling Studies

(2008) Małgorzata Dukat et al.   JOURNAL OF MEDICINAL CHEMISTRY

Enantioselective BINOL-Phosphoric Acid Catalyzed Pictet−Spengler Reactions ofN-Benzyltryptamine

(2008) Nishant V. Sewgobind et al.   JOURNAL OF ORGANIC CHEMISTRY

Lessons from Nature: Biomimetic Organocatalytic Carbon−Carbon Bond Formations§

(2008) Dieter Enders et al.   JOURNAL OF ORGANIC CHEMISTRY

Catalytic Enantioselective Additions of Indoles to Nitroalkenes

(2008) Madhu Ganesh et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

The advent and development of organocatalysis

(2008) David W. C. MacMillan   NATURE

5-HT6 receptor antagonists as novel cognitive enhancing agents for Alzheimer’s disease

(2008) Neil Upton et al.   Neurotherapeutics

Organocatalysis Lost: Modern Chemistry, Ancient Chemistry, and an Unseen Biosynthetic Apparatus

(2007) Carlos F. Barbas   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION