Efficient Synthesis of Substituted 3-Azabicyclo[3.1.0]hexan-2-ones from 2-Iodocyclopropanecarboxamides Using a Copper-Free Sonogashira Coupling

Suzuki Coupling of Potassium Cyclopropyl- and Alkoxymethyltrifluoroborates with Benzyl Chlorides

(2012) Virginie Colombel et al.   JOURNAL OF ORGANIC CHEMISTRY

The Pictet-Spengler Reaction in Nature and in Organic Chemistry

(2011) Joachim Stöckigt et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Discovery and synthesis of a new class of opioid ligand having a 3-azabicyclo[3.1.0]hexane core. An example of a ‘magic methyl’ giving a 35-fold improvement in binding

(2011) Graham Lunn et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

A gold(i)-catalyzed intramolecular oxidation–cyclopropanation sequence of 1,6-enynes: a convenient access to [n.1.0]bicycloalkanes

(2011) Deyun Qian et al.   CHEMICAL COMMUNICATIONS

Recent advances in Sonogashira reactions

(2011) Rafael Chinchilla et al.   CHEMICAL SOCIETY REVIEWS

Alkynylcyclopropanes from Terminal Alkynes through Consecutive Coupling to Fischer Carbene Complexes and Selective Propargylene Transfer

(2011) José Barluenga et al.   CHEMISTRY-A EUROPEAN JOURNAL

Ruthenium-Catalysed Synthesis of Fluorinated Bicyclic Amino Esters through Tandem Carbene Addition/Cyclopropanation of Enynes

(2011) Matthieu Eckert et al.   CHEMISTRY-A EUROPEAN JOURNAL

Titanium(IV) Chloride-Mediated Carbocyclization of 1,6-Enynes: Selective Synthesis of 3-Azabicyclo[3.1.0]hexanes and Functionalized Allenes by Controlling the Reaction Temperature

(2011) Zhen Zhang et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Diastereoselectivity Control in Formal Nucleophilic Substitution of Bromocyclopropanes with Oxygen- and Sulfur-Based Nucleophiles

(2011) Joseph E. Banning et al.   JOURNAL OF ORGANIC CHEMISTRY

Cross-Coupling of Mesylated Phenol Derivatives with Potassium Cyclopropyltrifluoroborate

(2011) Gary A. Molander et al.   JOURNAL OF ORGANIC CHEMISTRY

An Atom-Economic Synthesis of Bicyclo[3.1.0]hexanes by Rhodium N-Heterocyclic Carbene-Catalyzed Diastereoselective Tandem Hetero-[5 + 2] Cycloaddition/Claisen Rearrangement Reaction of Vinylic Oxiranes with Alkynes

(2011) Jian-Jun Feng et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Total Synthesis of (±)-Cycloclavine and (±)-5-epi-Cycloclavine

(2011) Filip R. Petronijevic et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Copper-Mediated Aerobic Synthesis of 3-Azabicyclo[3.1.0]hex-2-enes and 4-Carbonylpyrroles fromN-Allyl/Propargyl Enamine Carboxylates

(2011) Kah Kah Toh et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Palladium-Catalyzed Addition of Alkynes to Cyclopropenes: An Entry to Stereodefined Alkynylcyclopropanes

(2011) Alphonse Tenaglia et al.   ORGANIC LETTERS

Copper-Free Sonogashira Coupling of Cyclopropyl Iodides with Terminal Alkynes

(2011) Benoît de Carné-Carnavalet et al.   ORGANIC LETTERS

Influence of reaction conditions on products of the Pictet–Spengler condensation

(2011) Karolina Pulka et al.   TETRAHEDRON

Theoretical Investigation of Solvent Effects on Glycosylation Reactions: Stereoselectivity Controlled by Preferential Conformations of the Intermediate Oxacarbenium-Counterion Complex

(2010) Hiroko Satoh et al.   Journal of Chemical Theory and Computation

1-(Aryl)-6-[alkoxyalkyl]-3-azabicyclo[3.1.0]hexanes and 6-(Aryl)-6-[alkoxyalkyl]-3-azabicyclo[3.1.0]hexanes: A New Series of Potent and Selective Triple Reuptake Inhibitors

(2010) Fabrizio Micheli et al.   JOURNAL OF MEDICINAL CHEMISTRY

Enantiomerically Pure Polyheterocyclic Spiro-β-lactams from trans-4-Hydroxy-l-proline

(2010) Giuseppe Cremonesi et al.   JOURNAL OF ORGANIC CHEMISTRY

Mechanistic Studies on theCistoTransEpimerization of Trisubstituted 1,2,3,4-Tetrahydro-β-carbolines

(2010) Michael L. Van Linn et al.   JOURNAL OF ORGANIC CHEMISTRY

Pd(II)-Catalyzed Olefination ofsp3C−H Bonds

(2010) Masayuki Wasa et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Dual Role of Silanol Groups in Cyclopropanation and Hiyama−Denmark Cross-Coupling Reactions

(2010) Louis-Philippe B. Beaulieu et al.   ORGANIC LETTERS

Arylcyclopropanes: Properties, Synthesis and Use in Medicinal Chemistry

(2010) Alexandre Gagnon et al.   ORGANIC PREPARATIONS AND PROCEDURES INTERNATIONAL

Stereoselective Synthesis of Bicyclic Nitrocyclopropanes by a Radical-Anion Domino Reaction

(2009) Akio Kamimura et al.   CHEMISTRY-A EUROPEAN JOURNAL

A General Solution for Unstable Boronic Acids: Slow-Release Cross-Coupling from Air-Stable MIDA Boronates

(2009) David M. Knapp et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Highly Diastereoselective Formal Nucleophilic Substitution of Bromocyclopropanes

(2009) Bassam K. Alnasleh et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

New approaches for the synthesis of erythrinan alkaloids

(2009) Fengzhi Zhang et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

General and user-friendly protocol for the synthesis of functionalized aryl- and heteroaryl-cyclopropanes by Negishi cross-coupling reactions

(2009) Brian M. Coleridge et al.   TETRAHEDRON LETTERS

Cycloisomerization of 1,n-Enynes: Challenging Metal-Catalyzed Rearrangements and Mechanistic Insights

(2008) Véronique Michelet et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Studies on the structure–activity relationship of bicifadine analogs as monoamine transporter inhibitors

(2008) Mingzhu Zhang et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Gold-Catalyzed Cycloisomerizations of Enynes: A Mechanistic Perspective

(2008) Eloísa Jiménez-Núñez et al.   CHEMICAL REVIEWS

Cross-Coupling of Cyclopropyl- and Cyclobutyltrifluoroborates with Aryl and Heteroaryl Chlorides

(2008) Gary A. Molander et al.   JOURNAL OF ORGANIC CHEMISTRY

Recent developments in asymmetric cyclopropanation

(2008) Hélène Pellissier   TETRAHEDRON

Strictosidine Synthase:  Mechanism of a Pictet−Spengler Catalyzing Enzyme†

(2007) Justin J. Maresh et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

An efficient stereoselective synthesis of 1-iodo- or 1-phenyl selenenyl-2-aryl-3-azabicyclo[3.1.0]hexane via electrophilic cyclization of benzyl-2-arylmethylidenecyclopropylmethyl-amines

(2007) Weijun Fu et al.   TETRAHEDRON LETTERS