Arylcyclopropanes: Properties, Synthesis and Use in Medicinal Chemistry

Novel N-substituted 2-phenyl-1-sulfonylamino-cyclopropane carboxylates as selective ADAMTS-5 (Aggrecanase-2) inhibitors

(2009) Makoto Shiozaki et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

PdII-Catalyzed Enantioselective Activation of C(sp2)H and C(sp3)H Bonds Using Monoprotected Amino Acids as Chiral Ligands

(2008) Bing-Feng Shi et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis of Optically Active Boron-Silicon Bifunctional Cyclopropane Derivatives through Enantioselective Copper(I)-Catalyzed Reaction of Allylic Carbonates with a Diboron Derivative

(2008) Hajime Ito et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Achieving multi-isoform PI3K inhibition in a series of substituted 3,4-dihydro-2H-benzo[1,4]oxazines

(2008) Benjamin Perry et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Suzuki–Miyaura Cross-Coupling Reactions of Alkylboronic Acid Derivatives or Alkyltrifluoroborates with Aryl, Alkenyl or Alkyl Halides and Triflates

(2008) Henri Doucet   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Identification of (R)-1-(5-tert-Butyl-2,3-dihydro-1H-inden-1-yl)-3-(1H-indazol-4-yl)urea (ABT-102) as a Potent TRPV1 Antagonist for Pain Management

(2008) Arthur Gomtsyan et al.   JOURNAL OF MEDICINAL CHEMISTRY

Cross-Coupling of Cyclopropyl- and Cyclobutyltrifluoroborates with Aryl and Heteroaryl Chlorides

(2008) Gary A. Molander et al.   JOURNAL OF ORGANIC CHEMISTRY

Palladium-Catalyzed Cross-Coupling Reaction of Tricyclopropylbismuth with Aryl Halides and Triflates

(2008) Alexandre Gagnon et al.   JOURNAL OF ORGANIC CHEMISTRY

Melatonin agonist tasimelteon (VEC-162) for transient insomnia after sleep-time shift: two randomised controlled multicentre trials

(2008) Shantha MW Rajaratnam et al.   LANCET

Recent developments in asymmetric cyclopropanation

(2008) Hélène Pellissier   TETRAHEDRON

Characterization of thyroid hormone receptor α (TRα)-specific analogs with varying inner- and outer-ring substituents

(2007) Cory A. Ocasio et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Facially Selective and Regioselective Carbometalation of Cyclopropenes by Aryl Grignard Reagents

(2007) Ni Yan et al.   JOURNAL OF ORGANIC CHEMISTRY

The first example of direct cyclopropylation of arylamines at the 2-position with magnesium cyclopropylidenes

(2007) Yukie Yamada et al.   TETRAHEDRON LETTERS