The orexin OX1receptor exists predominantly as a homodimer in the basal state: potential regulation of receptor organization by both agonist and antagonist ligands

Applications of fluorescence and bioluminescence resonance energy transfer to drug discovery at G protein coupled receptors

(2010) Elisa Alvarez-Curto et al.   ANALYTICAL AND BIOANALYTICAL CHEMISTRY

Influence of MT7 toxin on the oligomerization state of the M1 muscarinic receptor1

(2010) Catherine Marquer et al.   BIOLOGY OF THE CELL

Ligand-induced internalization of the orexin OX1 and cannabinoid CB1 receptors assessed via N-terminal SNAP and CLIP-tagging

(2010) Richard J Ward et al.   BRITISH JOURNAL OF PHARMACOLOGY

A new approach to analyze cell surface protein complexes reveals specific heterodimeric metabotropic glutamate receptors

(2010) Etienne Doumazane et al.   FASEB JOURNAL

Oligomeric Size of the M2Muscarinic Receptor in Live Cells as Determined by Quantitative Fluorescence Resonance Energy Transfer

(2010) Luca F. Pisterzi et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Ligand Regulation of the Quaternary Organization of Cell Surface M3Muscarinic Acetylcholine Receptors Analyzed by Fluorescence Resonance Energy Transfer (FRET) Imaging and Homogeneous Time-resolved FRET

(2010) Elisa Alvarez-Curto et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Spatial control of EGF receptor activation by reversible dimerization on living cells

(2010) Inhee Chung et al.   NATURE

The properties of thermostabilised G protein-coupled receptors (StaRs) and their use in drug discovery

(2010) Nathan Robertson et al.   NEUROPHARMACOLOGY

Formation and dissociation of M1 muscarinic receptor dimers seen by total internal reflection fluorescence imaging of single molecules

(2010) J. A. Hern et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

Structures of the CXCR4 Chemokine GPCR with Small-Molecule and Cyclic Peptide Antagonists

(2010) B. Wu et al.   SCIENCE

Lighting up multiprotein complexes: lessons from GPCR oligomerization

(2010) Francisco Ciruela et al.   TRENDS IN BIOTECHNOLOGY

Reversible Dimerization of EGFR Revealed by Single-Molecule Fluorescence Imaging Using Quantum Dots

(2009) Nagako Kawashima et al.   CHEMISTRY-A EUROPEAN JOURNAL

The Hypocretins and their Role in Narcolepsy

(2009) Daniel Kroeger et al.   CNS & Neurological Disorders-Drug Targets

Ligand-regulated oligomerization of β2-adrenoceptors in a model lipid bilayer

(2009) Juan José Fung et al.   EMBO JOURNAL

BRET3: a red-shifted bioluminescence resonance energy transfer (BRET)-based integrated platform for imaging protein-protein interactions from single live cells and living animals

(2009) Abhijit De et al.   FASEB JOURNAL

The Action and Mode of Binding of Thiazolidinedione Ligands at Free Fatty Acid Receptor 1

(2009) Nicola J. Smith et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Pirenzepine Promotes the Dimerization of Muscarinic M1 Receptors through a Three-step Binding Process

(2009) Brigitte Ilien et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Semisynthetic Fluorescent Sensor Proteins Based on Self-Labeling Protein Tags

(2009) Matthias A. Brun et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Instability of a Class A G Protein-Coupled Receptor Oligomer Interface

(2009) J. M. Fonseca et al.   MOLECULAR PHARMACOLOGY

The structure and function of G-protein-coupled receptors

(2009) Daniel M. Rosenbaum et al.   NATURE

Allosteric communication between protomers of dopamine class A GPCR dimers modulates activation

(2009) Yang Han et al.   Nature Chemical Biology

Analysis of receptor oligomerization by FRAP microscopy

(2009) Sandra Dorsch et al.   NATURE METHODS

Cell-surface protein-protein interaction analysis with time-resolved FRET and snap-tag technologies: application to GPCR oligomerization

(2008) Damien Maurel et al.   NATURE METHODS

Co-evolving stability and conformational homogeneity of the human adenosine A2a receptor

(2008) F. Magnani et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

Light resonance energy transfer-based methods in the study of G protein-coupled receptor oligomerization

(2007) Jorge Gandía et al.   BIOESSAYS

CB2cannabinoid receptors as an emerging target for demyelinating diseases: from neuroimmune interactions to cell replacement strategies

(2007) Arévalo-Martín et al.   BRITISH JOURNAL OF PHARMACOLOGY