Ligand-induced internalization of the orexin OX1 and cannabinoid CB1 receptors assessed via N-terminal SNAP and CLIP-tagging

Rimonabant for the treatment of overweight and obese people

(2014) J Burch et al.   HEALTH TECHNOLOGY ASSESSMENT

Signal Transduction via Cannabinoid Receptors

(2012) George Dalton et al.   CNS & Neurological Disorders-Drug Targets

Orexins and Gastrointestinal Functions

(2010) M. Baccari   CURRENT PROTEIN & PEPTIDE SCIENCE

Orexin receptor antagonists: a review of promising compounds patented since 2006

(2010) Paul J Coleman et al.   EXPERT OPINION ON THERAPEUTIC PATENTS

Ligand Regulation of the Quaternary Organization of Cell Surface M3Muscarinic Acetylcholine Receptors Analyzed by Fluorescence Resonance Energy Transfer (FRET) Imaging and Homogeneous Time-resolved FRET

(2010) Elisa Alvarez-Curto et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

High content screening: seeing is believing

(2010) Fabian Zanella et al.   TRENDS IN BIOTECHNOLOGY

Biochemical and behavioural characterization of EMPA, a novel high-affinity, selective antagonist for the OX2 receptor

(2009) P Malherbe et al.   BRITISH JOURNAL OF PHARMACOLOGY

The Hypocretins and their Role in Narcolepsy

(2009) Daniel Kroeger et al.   CNS & Neurological Disorders-Drug Targets

The Current Status and Future Perspectives of Studies of Cannabinoid Receptor 1 Antagonists as Anti-Obesity Agents

(2009) Hyeon-Kyu Lee et al.   CURRENT TOPICS IN MEDICINAL CHEMISTRY

Emerging drugs for insomnia: new frontiers for old and novel targets

(2009) Shannon S Sullivan et al.   EXPERT OPINION ON EMERGING DRUGS

The Action and Mode of Binding of Thiazolidinedione Ligands at Free Fatty Acid Receptor 1

(2009) Nicola J. Smith et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Biochemical and Electrophysiological Characterization of Almorexant, a Dual Orexin 1 Receptor (OX1)/Orexin 2 Receptor (OX2) Antagonist: Comparison with Selective OX1 and OX2 Antagonists

(2009) P. Malherbe et al.   MOLECULAR PHARMACOLOGY

An Engineered Protein Tag for Multiprotein Labeling in Living Cells

(2008) Arnaud Gautier et al.   CHEMISTRY & BIOLOGY

Constitutive Activity of the Cannabinoid CB1 Receptor Regulates the Function of Co-expressed Mu Opioid Receptors

(2008) Meritxell Canals et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Morphine Desensitization, Internalization, and Down-Regulation of the   Opioid Receptor Is Facilitated by Serotonin 5-Hydroxytryptamine2A Receptor Coactivation

(2008) J. F. Lopez-Gimenez et al.   MOLECULAR PHARMACOLOGY

Cell-surface protein-protein interaction analysis with time-resolved FRET and snap-tag technologies: application to GPCR oligomerization

(2008) Damien Maurel et al.   NATURE METHODS

A day in the life of a G protein-coupled receptor: the contribution to function of G protein-coupled receptor dimerization

(2007) G Milligan   BRITISH JOURNAL OF PHARMACOLOGY

Role of receptor internalization in the agonist-induced desensitization of cannabinoid type 1 receptors

(2007) Dai-Fei Wu et al.   JOURNAL OF NEUROCHEMISTRY

Regulation of OX1 orexin/hypocretin receptor-coupling to phospholipase C by Ca2+ influx

(2006) L Johansson et al.   BRITISH JOURNAL OF PHARMACOLOGY