A Multicomponent Coupling Reaction Induced by Insertion of Arynes into the CO Bond of Formamide

Preparation and Regioselective Diels-Alder Reactions of Borylbenzynes: Synthesis of Functionalized Arylboronates

(2010) Takashi Ikawa et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Intermolecular N-Heterocyclic Carbene Catalyzed Hydroacylation of Arynes

(2010) Akkattu T. Biju et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Total Synthesis of Dictyodendrin A and B

(2010) Kentaro Okano et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Aryne,ortho-Quinone Methide, andortho-Quinodimethane: Synthesis of Multisubstituted Arenes Using the Aromatic Reactive Intermediates

(2010) Hiroto Yoshida et al.   BULLETIN OF THE CHEMICAL SOCIETY OF JAPAN

Palladium-catalyzed annulations of arynes with 2-(2-iodophenoxy)-1-substituted ethanones

(2010) Rong-Jiang Li et al.   CHEMICAL COMMUNICATIONS

Crystal structure of thioflavin-T and its binding to amyloid fibrils: insights at the molecular level

(2010) Cristina Rodríguez-Rodríguez et al.   CHEMICAL COMMUNICATIONS

Platinum-catalysed diborylation of arynes: synthesis and reaction of 1,2-diborylarenes

(2010) Hiroto Yoshida et al.   CHEMICAL COMMUNICATIONS

Indolyne and Aryne Distortions and Nucleophilic Regioselectivites

(2010) Paul H.-Y. Cheong et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Indolyne Experimental and Computational Studies: Synthetic Applications and Origins of Selectivities of Nucleophilic Additions

(2010) G-Yoon J. Im et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Regioselective Reactions of Highly Substituted Arynes

(2010) Pamela M. Tadross et al.   ORGANIC LETTERS

Aryne Acyl-Alkylation in the General and Convergent Synthesis of Benzannulated Macrolactone Natural Products: An Enantioselective Synthesis of (−)-Curvularin

(2010) Pamela M. Tadross et al.   ORGANIC LETTERS

Sequential Reaction of Arynes via Insertion into the π-Bond of Amides and Trapping Reaction with Dialkylzincs

(2010) Eito Yoshioka et al.   ORGANIC LETTERS

New Synthesis of 1-Substituted-1H-indazoles via 1,3-Dipolar Cycloaddition ofin situGenerated Nitrile Imines and Benzyne

(2010) Christian Spiteri et al.   ORGANIC LETTERS

Synthesis of Substituted Indoles from 2-Azidoacrylates andortho-Silyl Aryltriflates†

(2010) Deng Hong et al.   ORGANIC LETTERS

Intermolecular C−O Addition of Carboxylic Acids to Arynes

(2010) Anton V. Dubrovskiy et al.   ORGANIC LETTERS

The Benzyne Aza-Claisen Reaction

(2009) Alastair A. Cant et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Nickel-Catalyzed Three-Component [2+2+2] Cycloaddition Reaction of Arynes, Alkenes, and Alkynes

(2009) Zaozao Qiu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A Multicomponent Reaction of Arynes, Isocyanides, and Terminal Alkynes: Highly Chemo- and Regioselective Synthesis of Polysubstituted Pyridines and Isoquinolines

(2009) Feng Sha et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

α-Glucosidase inhibitory antihyperglycemic activity of substituted chromenone derivatives

(2009) B. China Raju et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis, Molecular Modeling, and Selective Inhibitory Activity against Human Monoamine Oxidases of 3-Carboxamido-7-Substituted Coumarins†

(2009) Franco Chimenti et al.   JOURNAL OF MEDICINAL CHEMISTRY

Selective Synthesis ofo-Acylbenzylphosphonates by Insertion Reactions of Arynes into β-Ketophosphonates

(2009) Yi-Lin Liu et al.   JOURNAL OF ORGANIC CHEMISTRY

Insertion of Benzene Rings into the Amide Bond: One-Step Synthesis of Acridines and Acridones from Aryl Amides

(2009) Didier G. Pintori et al.   ORGANIC LETTERS

Ring expansion reaction of α-sulfonyl cyclic ketones via insertion of arynes into C–C: a facile and mild access to medium- and large-sized benzannulated carbocycles

(2009) Tiexin Zhang et al.   TETRAHEDRON LETTERS

Decoupling Deprotonation from Metalation: Thia-Fries Rearrangement

(2008) Alan M. Dyke et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Palladium-Catalyzed Annulation of Acyloximes with Arynes (or Alkynes): Synthesis of Phenanthridines and Isoquinolines

(2008) Thibaud Gerfaud et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Gold-catalyzed efficient tandem assembly of terminal alkynes and arynes: synthesis of alkynylated biphenyl derivatives

(2008) Chunsong Xie et al.   CHEMICAL COMMUNICATIONS

Fluorenes as new molecular scaffolds for carbon–carbon σ-bond cleavage reaction: acylfluorenylation of arynes

(2008) Hiroto Yoshida et al.   CHEMICAL COMMUNICATIONS

(9S)-9-(2-Hydroxy-4,4-dimethyl-6-oxo-1-cyclohexen-1-yl)-3,3-dimethyl-2,3,4,9-tetrahydro-1H-xanthen-1-one, a Selective and Orally Active Neuropeptide Y Y5 Receptor Antagonist

(2008) Nagaaki Sato et al.   JOURNAL OF MEDICINAL CHEMISTRY

Novel 3-Carboxamide-coumarins as Potent and Selective FXIIa Inhibitors

(2008) Séverine Robert et al.   JOURNAL OF MEDICINAL CHEMISTRY

A Concise Total Synthesis of (−)-Quinocarcin via Aryne Annulation

(2008) Kevin M. Allan et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Orthogonal Synthesis of Indolines and Isoquinolines via Aryne Annulation

(2008) Christopher D. Gilmore et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Carbocupration−Functionalization of Arynes: Rapid Access to Variably Ortho-Substituted ((E)-3-Phenylprop-1-enyl)silanes

(2008) Ashok Ganta et al.   ORGANIC LETTERS

Four-Component Benzyne Coupling Reactions: A Concise Total Synthesis of Dehydroaltenuene B

(2008) Darunee Soorukram et al.   ORGANIC LETTERS

Cycloaddition of Arynes with Iodonium Ylides:  a Mild and General Route for the Synthesis of Benzofuran Derivatives

(2008) Xiao-Cheng Huang et al.   ORGANIC LETTERS

Reaction of Benzyne with Salicylaldehydes: General Synthesis of Xanthenes, Xanthones, and Xanthols

(2008) Kentaro Okuma et al.   ORGANIC LETTERS

A novel α,β-unsaturated nitrone-aryne [3+2] cycloaddition and its application in the synthesis of the cortistatin core

(2008) Mingji Dai et al.   TETRAHEDRON LETTERS