Calcium-mediated one-pot preparation of isoxazoles with deuterium incorporation

A solid acetylene reagent with enhanced reactivity: fluoride-mediated functionalization of alcohols and phenols

(2017) Georg Werner et al.   GREEN CHEMISTRY

Calcium Carbide: A Unique Reagent for Organic Synthesis and Nanotechnology

(2016) Konstantin S. Rodygin et al.   Chemistry-An Asian Journal

Antipsychotic Drug-Induced Somnolence: Incidence, Mechanisms, and Management

(2016) Fang Fang et al.   CNS DRUGS

Anti-methicillin resistant Staphylococcus aureus activity, synergism with oxacillin and molecular docking studies of metronidazole-triazole hybrids

(2016) Beena Negi et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

An Atom-Economic Approach for Vinylation of Indoles and Phenols Using Calcium Carbide as Acetylene Surrogate

(2016) Eakkaphon Rattanangkool et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Synthesis of vinyl ethers of alcohols using calcium carbide under superbasic catalytic conditions (KOH/DMSO)

(2016) Ryosuke Matake et al.   GREEN CHEMISTRY

An efficient metal-free pathway to vinyl thioesters with calcium carbide as the acetylene source

(2016) Konstantin S. Rodygin et al.   GREEN CHEMISTRY

Clinical outcomes of long-acting injectable risperidone in patients with bipolar I disorder: A 1-year retrospective cohort study

(2016) Hsue-Wei Chan et al.   JOURNAL OF AFFECTIVE DISORDERS

Different spectrophotometric methods applied for the analysis of binary mixture of flucloxacillin and amoxicillin: A comparative study

(2016) Khalid A.M. Attia et al.   SPECTROCHIMICA ACTA PART A-MOLECULAR AND BIOMOLECULAR SPECTROSCOPY

Highly regioselective dipolar cycloadditions of nitrile oxides with α,β-acetylenic aldehydes

(2016) Longqiang Jiang et al.   TETRAHEDRON LETTERS

A base promoted multigram synthesis of aminoisoxazoles: valuable building blocks for drug discovery and peptidomimetics

(2016) Bohdan A. Chalyk et al.   RSC Advances

Palladium-Catalyzed Direct CH Arylation of Isoxazoles at the 5-Position

(2015) Masashi Shigenobu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Direct synthesis of aryl substituted pyrroles from calcium carbide: an underestimated chemical feedstock

(2015) Narongpol Kaewchangwat et al.   GREEN CHEMISTRY

Calcium carbide as a convenient acetylene source in the synthesis of unsaturated sulfides, promising functionalized monomers

(2015) Konstantin S. Rodygin et al.   MENDELEEV COMMUNICATIONS

Fluoride-Assisted Activation of Calcium Carbide: A Simple Method for the Ethynylation of Aldehydes and Ketones

(2015) Abolfazl Hosseini et al.   ORGANIC LETTERS

Phase-Vanishing Method with Acetylene Evolution and Its Utilization in Several Organic Syntheses

(2015) Ryosuke Matake et al.   ORGANIC LETTERS

Kinetics and mechanism of the thermal decomposition of the isoxazoline compounds

(2015) T. K. Goncharov et al.   Russian Journal of Physical Chemistry B

Synthesis of functionalized 2-isoxazolines as three-dimensional fragments for fragment-based drug discovery

(2015) Ngoc Chau Tran et al.   TETRAHEDRON LETTERS

5-Substituted pyridylisoxazoles as effective inhibitors of platelet aggregation

(2015) O. V. Demina et al.   RUSSIAN CHEMICAL BULLETIN

Short-course oral co-trimoxazole versus intramuscular benzathine benzylpenicillin for impetigo in a highly endemic region: an open-label, randomised, controlled, non-inferiority trial

(2014) Asha C Bowen et al.   LANCET

Heavy drugs draw heavy interest from pharma backers

(2013) Alla Katsnelson   NATURE MEDICINE

Nitrile Oxide/Alkyne Cycloadditions - A Credible Platform for Synthesis of Bioinspired Molecules by Metal-Free Molecular Clicking

(2012) Frances Heaney   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Highly regioselective nitrile oxide dipolar cycloadditions with ortho-nitrophenyl alkynes

(2012) Melissa L. McIntosh et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Platinum-catalyzed cyclizations viacarbene intermediates: syntheses of complementary positional isomers of isoxazoles

(2012) Paul A. Allegretti et al.   Chemical Science

Synopsis of Some Recent Tactical Application of Bioisosteres in Drug Design

(2011) Nicholas A. Meanwell   JOURNAL OF MEDICINAL CHEMISTRY

Regioselective Synthesis and Slow-Release Suzuki–Miyaura Cross-Coupling of MIDA Boronate-Functionalized Isoxazoles and Triazoles

(2011) Jonathan E. Grob et al.   JOURNAL OF ORGANIC CHEMISTRY

Direct Synthesis of Polysubstituted Aluminoisoxazoles and Pyrazoles by a Metalative Cyclization

(2011) Olivier Jackowski et al.   ORGANIC LETTERS

In Vitro and In Vivo Isotope Effects with Hepatitis C Protease Inhibitors: Enhanced Plasma Exposure of Deuterated Telaprevir versus Telaprevir in Rats

(2009) François Maltais et al.   JOURNAL OF MEDICINAL CHEMISTRY

A Regioselective Route to 5-Substituted Isoxazole- and Isoxazoline-3-phos­phonates

(2009) Paola Conti et al.   SYNTHESIS-STUTTGART

Ruthenium-Catalyzed Cycloaddition of Nitrile Oxides and Alkynes: Practical Synthesis of Isoxazoles

(2008) Scott Grecian et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Palladium-Catalyzed Arylation and Alkylation of 3,5-Diphenylisoxazole with Boronic Acids via C−H Activation

(2008) Jean-Ho Chu et al.   ORGANOMETALLICS