1-Bromoethene-1-sulfonyl fluoride (1-Br-ESF), a new SuFEx clickable reagent, and its application for regioselective construction of 5-sulfonylfluoro isoxazoles

Discovery of a Small Molecule Probe That Post-Translationally Stabilizes the Survival Motor Neuron Protein for the Treatment of Spinal Muscular Atrophy

(2017) Anne Rietz et al.   JOURNAL OF MEDICINAL CHEMISTRY

Pd-Catalyzed Conversion of Aryl Iodides to Sulfonyl Fluorides Using SO2 Surrogate DABSO and Selectfluor

(2017) Ariana L. Tribby et al.   JOURNAL OF ORGANIC CHEMISTRY

Broad-Spectrum Kinase Profiling in Live Cells with Lysine-Targeted Sulfonyl Fluoride Probes

(2017) Qian Zhao et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Bifluoride-catalysed sulfur(VI) fluoride exchange reaction for the synthesis of polysulfates and polysulfonates

(2017) Bing Gao et al.   Nature Chemistry

A Synthesis of “Dual Warhead” β-Aryl Ethenesulfonyl Fluorides and One-Pot Reaction to β-Sultams

(2017) Praveen K. Chinthakindi et al.   ORGANIC LETTERS

One-pot palladium-catalyzed synthesis of sulfonyl fluorides from aryl bromides

(2017) Alyn T. Davies et al.   Chemical Science

Ethenesulfonyl Fluoride: The Most Perfect Michael Acceptor Ever Found?

(2016) Quan Chen et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A Heck-Matsuda Process for the Synthesis of β-Arylethenesulfonyl Fluorides: Selectively Addressable Bis-electrophiles for SuFEx Click Chemistry

(2016) Hua-Li Qin et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Proteasome inhibition by new dual warhead containing peptido vinyl sulfonyl fluorides

(2016) Arwin J. Brouwer et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Ethenesulfonyl Fluoride (ESF): An On-Water Procedure for the Kilogram-Scale Preparation

(2016) Qinheng Zheng et al.   JOURNAL OF ORGANIC CHEMISTRY

Selective and Orthogonal Post-Polymerization Modification using Sulfur(VI) Fluoride Exchange (SuFEx) and Copper-Catalyzed Azide–Alkyne Cycloaddition (CuAAC) Reactions

(2016) James S. Oakdale et al.   MACROMOLECULES

Recent Developments in the Synthesis and Reactivity of Isoxazoles: Metal Catalysis and Beyond

(2015) Feng Hu et al.   ADVANCED SYNTHESIS & CATALYSIS

Palladium(II)-Catalyzed Synthesis of Sulfinates from Boronic Acids and DABSO: A Redox-Neutral, Phosphine-Free Transformation

(2015) Alex S. Deeming et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Stable gold(III) catalysts by oxidative addition of a carbon–carbon bond

(2015) Chung-Yeh Wu et al.   NATURE

Sulfur(VI) Fluoride Exchange (SuFEx): Another Good Reaction for Click Chemistry

(2014) Jiajia Dong et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Preparation of 3,5-Disubstituted Pyrazoles and Isoxazoles from Terminal Alkynes, Aldehydes, Hydrazines, and Hydroxylamine

(2014) Ryo Harigae et al.   JOURNAL OF ORGANIC CHEMISTRY

Pd(II)-Catalyzed C–H Iodination Using Molecular I2 as the Sole Oxidant

(2013) Xiao-Chen Wang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Aromatic Sulfonyl Fluorides Covalently Kinetically Stabilize Transthyretin to Prevent Amyloidogenesis while Affording a Fluorescent Conjugate

(2013) Neil P. Grimster et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Exceptionally fast carbon–carbon bond reductive elimination from gold(III)

(2013) William J. Wolf et al.   Nature Chemistry

Synthesis of Isoxazole Triflones

(2012) Hiroyuki Kawai et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Weak Coordination as a Powerful Means for Developing Broadly Useful C–H Functionalization Reactions

(2011) Keary M. Engle et al.   ACCOUNTS OF CHEMICAL RESEARCH

Cascade Formation of Isoxazoles: Facile Base-Mediated Rearrangement of Substituted Oxetanes

(2011) Johannes A. Burkhard et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Iodocyclization of Hydroxylamine Derivatives Based on the Control of Oxidative Aromatization Leading to 2,5-Dihydroisoxazoles and Isoxazoles

(2011) Takashi Okitsu et al.   JOURNAL OF ORGANIC CHEMISTRY

New Synthesis of 1-Substituted-1H-indazoles via 1,3-Dipolar Cycloaddition ofin situGenerated Nitrile Imines and Benzyne

(2010) Christian Spiteri et al.   ORGANIC LETTERS