Synthesis of Isoxazole Triflones

A regioselective synthesis of poly-substituted aryl triflones through self-promoting three component reaction

(2011) Hikaru Yanai et al.   CHEMICAL COMMUNICATIONS

Direct Synthesis of Polysubstituted Aluminoisoxazoles and Pyrazoles by a Metalative Cyclization

(2011) Olivier Jackowski et al.   ORGANIC LETTERS

Synthesis of Indole and Biindolyl Triflones: Trifluoromethanesulfonylation of Indoles with Tf2O/TTBP (2,4,6-tri-tert-butylpyridine) System

(2011) Xiu-Hua Xu et al.   ORGANIC LETTERS

Stereoselective synthesis of ambiphilic alkenes via regioselective methylation of α-trifluoromethanesulfonyl carbonyl compounds with trimethylsilyldiazomethane

(2011) Han Il Kong et al.   TETRAHEDRON LETTERS

Cinchona Alkaloid/TiIV-Catalyzed Enantioselective Enamine-Trifluoropyruvate Condensation-Cyclization Reaction and Its Application to Drug-like Heterocycles

(2010) Shinichi Ogawa et al.   CHEMISTRY-A EUROPEAN JOURNAL

An Alkynyliodide Cycloaddition Strategy for the Construction of Iodoisoxazoles

(2010) James A. Crossley et al.   JOURNAL OF ORGANIC CHEMISTRY

Enantioselective Friedel−Crafts Reaction of β-Trifluoromethylated Acrylates with Pyrroles and Its Application to the Synthesis of Trifluorinated Heliotridane

(2010) Yiyong Huang et al.   ORGANIC LETTERS

Sequential Reaction of Arynes via Insertion into the π-Bond of Amides and Trapping Reaction with Dialkylzincs

(2010) Eito Yoshioka et al.   ORGANIC LETTERS

Direct Synthesis of Trisubstituted Isoxazoles through Gold-Catalyzed Domino Reaction of Alkynyl Oxime Ethers

(2010) Masafumi Ueda et al.   ORGANIC LETTERS

Benchmark and Solvent-Free Preparation of Sulfonium Salt Based Electrophilic Trifluoromethylating Reagents

(2009) Yohan Macé et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Efficient and Regioselective One-Pot Synthesis of 3-Substituted and 3,5-Disubstituted Isoxazoles

(2009) Shibing Tang et al.   ORGANIC LETTERS

A New Class of 3′-Sulfonyl BINAPHOS Ligands: Modulation of Activity and Selectivity in Asymmetric Palladium-Catalysed Hydrophosphorylation of Styrene

(2008) Katalin Barta et al.   ADVANCED SYNTHESIS & CATALYSIS

Tetrahydropyridine-4-carboxamides as novel, potent transient receptor potential vanilloid 1 (TRPV1) antagonists

(2008) Brian S. Brown et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Discovery of an Orally Bioavailable Small Molecule Inhibitor of Prosurvival B-Cell Lymphoma 2 Proteins

(2008) Cheol-Min Park et al.   JOURNAL OF MEDICINAL CHEMISTRY

Ultrasound promoted synthesis of substituted pyrazoles and isoxazoles containing sulphone moiety

(2008) Tamer S. Saleh et al.   ULTRASONICS SONOCHEMISTRY