The role of G-protein-coupled membrane estrogen receptor in mouse Leydig cell function—in vivo and in vitro evaluation

Xenoestrogen regulation of ERα/ERβ balance in hormone-associated cancers

(2017) Filippo Acconcia et al.   MOLECULAR AND CELLULAR ENDOCRINOLOGY

Opposite Function of ERα and ERβ in Controlling 17β-Estradiol-mediated Osteogenesis in Osteoblasts

(2016) Yu-xiang Wang et al.   ARCHIVES OF MEDICAL RESEARCH

The role of estradiol in male reproductive function

(2016) Ranjith Ramasamy et al.   ASIAN JOURNAL OF ANDROLOGY

Extra-gonadal sites of estrogen biosynthesis and function

(2016) Radwa Barakat et al.   BMB Reports

Everolimus downregulates estrogen receptor and induces autophagy in aromatase inhibitor-resistant breast cancer cells

(2016) Asona Lui et al.   BMC CANCER

GPR30 Promotes Prostate Stromal Cell Activation via Suppression of ERα Expression and Its Downstream Signaling Pathway

(2016) Bona Jia et al.   ENDOCRINOLOGY

Lipid droplets and steroidogenic cells

(2016) Wen-Jun Shen et al.   EXPERIMENTAL CELL RESEARCH

Divergent Regulation of ER and Kiss Genes by 17β-Estradiol in Hypothalamic ARC Versus AVPV Models

(2016) Alice K. Treen et al.   MOLECULAR ENDOCRINOLOGY

Are aryl hydrocarbon receptor and G-protein–coupled receptor 30 involved in the regulation of seasonal testis activity in photosensitive rodent—the bank vole (Myodes glareolus)?

(2016) Marta Zarzycka et al.   THERIOGENOLOGY

Primary and tumor mouse Leydig cells exposed to polychlorinated naphthalenes mixture: Effect on estrogen related-receptors expression, intracellular calcium level and sex hormones secretion

(2016) L. Pardyak et al.   TISSUE & CELL

Estrogen receptor-β in mitochondria: implications for mitochondrial bioenergetics and tumorigenesis

(2015) Tien-Ling Liao et al.   Annals of the New York Academy of Sciences

Osteoprotective effect of combination therapy of low-dose oestradiol with G15, a specific antagonist of GPR30/GPER in ovariectomy-induced osteoporotic rats

(2015) W.-B. Kang et al.   BIOSCIENCE REPORTS

Oestrogen action and male fertility: experimental and clinical findings

(2015) Xiangdong Li et al.   CELLULAR AND MOLECULAR LIFE SCIENCES

The G-protein coupled estrogen receptor, GPER: The inside and inside-out story

(2015) H.M. Gaudet et al.   MOLECULAR AND CELLULAR ENDOCRINOLOGY

Sex Hormones and Their Receptors Regulate Liver Energy Homeostasis

(2015) Minqian Shen et al.   International Journal of Endocrinology

Estrogens Induce Rapid Cytoskeleton Re-Organization in Human Dermal Fibroblasts via the Non-Classical Receptor GPR30

(2015) Julie Carnesecchi et al.   PLoS One

Low levels of 3,3′-diindolylmethane activate estrogen receptor α and induce proliferation of breast cancer cells in the absence of estradiol

(2014) Maud Marques et al.   BMC CANCER

Tamoxifen through GPER upregulates aromatase expression: a novel mechanism sustaining tamoxifen-resistant breast cancer cell growth

(2014) Stefania Catalano et al.   BREAST CANCER RESEARCH AND TREATMENT

GPCR signaling along the endocytic pathway

(2014) Roshanak Irannejad et al.   CURRENT OPINION IN CELL BIOLOGY

Early expression of aromatase and the membrane estrogen receptor GPER in neuromasts reveals a role for estrogens in the development of the frog lateral line system

(2014) Christine K. Hamilton et al.   GENERAL AND COMPARATIVE ENDOCRINOLOGY

Expression pattern of estrogen receptors α and β and G-protein-coupled estrogen receptor 1 in the human testis

(2014) Daniela Fietz et al.   HISTOCHEMISTRY AND CELL BIOLOGY

Estrogen Rapidly Enhances Incisional Pain of Ovariectomized Rats Primarily through the G Protein-Coupled Estrogen Receptor

(2014) Guanghui An et al.   INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES

Activation of GPER-1 Estradiol Receptor Downregulates Production of Testosterone in Isolated Rat Leydig Cells and Adult Human Testis

(2014) Laurent Vaucher et al.   PLoS One

Direct estradiol and diethylstilbestrol actions on early- versus late-stage prostate cancer cells

(2014) Luke Y. Koong et al.   PROSTATE

Expression of the oestrogen receptor GPER by testicular peritubular cells is linked to sexual maturation and male fertility

(2014) F. Sandner et al.   Andrology

The G Protein-Coupled Estrogen Receptor-1, GPER-1, Promotes Fibrillogenesis via a Shc-Dependent Pathway Resulting in Anchorage-Independent Growth

(2014) Hilary T. Magruder et al.   Hormones & Cancer

Golgi tubules: their structure, formation and role in intra-Golgi transport

(2013) Emma Martínez-Alonso et al.   HISTOCHEMISTRY AND CELL BIOLOGY

Classical Estrogen Receptors and ERα Splice Variants in the Mouse

(2013) Debra L. Irsik et al.   PLoS One

Does 4-tert-octylphenol affect estrogen signaling pathways in bank vole Leydig cells and tumor mouse Leydig cells in vitro?

(2013) Malgorzata Kotula-Balak et al.   REPRODUCTIVE TOXICOLOGY

Minireview: G Protein-Coupled Estrogen Receptor-1, GPER-1: Its Mechanism of Action and Role in Female Reproductive Cancer, Renal and Vascular Physiology

(2012) Edward J. Filardo et al.   ENDOCRINOLOGY

G Protein-coupled Estrogen Receptor Mediates the Up-regulation of Fatty Acid Synthase Induced by 17β-Estradiol in Cancer Cells and Cancer-associated Fibroblasts

(2012) Maria Francesca Santolla et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

G Protein-Coupled Estrogen Receptor (GPER) Expression in Normal and Abnormal Endometrium

(2012) Beth J. Plante et al.   Reproductive Sciences

The G-Protein-Coupled Estrogen Receptor (GPER) is Expressed in Normal Human Ovaries and is Upregulated in Ovarian Endometriosis and Pelvic Inflammatory Disease Involving the Ovary

(2012) Sabine Heublein et al.   Reproductive Sciences

Estrogen Signaling and Cardiovascular Disease

(2011) Elizabeth Murphy   CIRCULATION RESEARCH

Prenatal and neonatal exposure to flutamide affects function of Leydig cells in adult boar

(2011) M. Kotula-Balak et al.   DOMESTIC ANIMAL ENDOCRINOLOGY

Mechanisms of Estradiol-Induced Insulin Secretion by the G Protein-Coupled Estrogen Receptor GPR30/GPER in Pancreatic β-Cells

(2011) Geetanjali Sharma et al.   ENDOCRINOLOGY

Down-modulation of the G-protein-coupled Estrogen Receptor, GPER, from the Cell Surface Occurs via atrans-Golgi-Proteasome Pathway

(2011) Shi-Bin Cheng et al.   JOURNAL OF BIOLOGICAL CHEMISTRY

Identification of a GPER/GPR30 antagonist with improved estrogen receptor counterselectivity

(2011) Megan K. Dennis et al.   JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY

Development of subtype-selective oestrogen receptor-based therapeutics

(2011) Stefan Nilsson et al.   NATURE REVIEWS DRUG DISCOVERY

The G-protein-coupled estrogen receptor GPER in health and disease

(2011) Eric R. Prossnitz et al.   Nature Reviews Endocrinology

β-arrestin-mediated receptor trafficking and signal transduction

(2011) Sudha K. Shenoy et al.   TRENDS IN PHARMACOLOGICAL SCIENCES

Estrogen receptors and function in the male reproductive system

(2010) Maria Fatima Magalhães Lazari et al.   Arquivos Brasileiros de Endocrinologia e Metabologia

Expression and Signaling of G Protein-Coupled Estrogen Receptor 1 (GPER) in Rat Sertoli Cells1

(2010) Thaís F. G. Lucas et al.   BIOLOGY OF REPRODUCTION

Role of G protein-coupled estrogen receptor 1, GPER, in inhibition of oocyte maturation by endogenous estrogens in zebrafish

(2010) Yefei Pang et al.   DEVELOPMENTAL BIOLOGY

Gper and ESRs are expressed in rat round spermatids and mediate oestrogen-dependent rapid pathways modulating expression of cyclin B1 and Bax

(2010) A. Chimento et al.   INTERNATIONAL JOURNAL OF ANDROLOGY

17β-Estradiol activates rapid signaling pathways involved in rat pachytene spermatocytes apoptosis through GPR30 and ERα

(2010) Adele Chimento et al.   MOLECULAR AND CELLULAR ENDOCRINOLOGY

Regulation of GPCR signal networks via membrane trafficking

(2010) F. Jean-Alphonse et al.   MOLECULAR AND CELLULAR ENDOCRINOLOGY

Oestrogens and spermatogenesis

(2010) S. Carreau et al.   PHILOSOPHICAL TRANSACTIONS OF THE ROYAL SOCIETY B-BIOLOGICAL SCIENCES

Effects of 4-tert-octylphenol on the testes and seminal vesicles in adult male bank voles

(2010) Anna Hejmej et al.   REPRODUCTIVE TOXICOLOGY

A novel estrogen receptor GPER inhibits mitochondria permeability transition pore opening and protects the heart against ischemia-reperfusion injury

(2009) Jean Chrisostome Bopassa et al.   AMERICAN JOURNAL OF PHYSIOLOGY-HEART AND CIRCULATORY PHYSIOLOGY

Testicular Steroid Hormone Secretion in the Boar and Expression of Testicular and Epididymal Steroid Sulphatase and Estrogen Sulphotransferase Activity

(2009) B. Hoffmann et al.   EXPERIMENTAL AND CLINICAL ENDOCRINOLOGY & DIABETES

Morphological comparison of the testis and efferent ductules between wild-type and estrogen receptor α knockout mice during postnatal development

(2009) Ki-Ho Lee et al.   JOURNAL OF ANATOMY

In vivo effects of a GPR30 antagonist

(2009) Megan K Dennis et al.   Nature Chemical Biology

GPR30 Does Not Mediate Estrogenic Responses in Reproductive Organs in Mice

(2008) Christiane Otto et al.   BIOLOGY OF REPRODUCTION

Opposite Roles of Estrogen Receptor (ER)-α and ERβ in the Modulation of Luteinizing Hormone Responses to Kisspeptin in the Female Rat: Implications for the Generation of the Preovulatory Surge

(2008) J. Roa et al.   ENDOCRINOLOGY

The Novel Estrogen Receptor, G Protein-Coupled Receptor 30, Mediates the Proliferative Effects Induced by 17β-Estradiol on Mouse Spermatogonial GC-1 Cell Line

(2008) Rosa Sirianni et al.   ENDOCRINOLOGY

Expression Pattern of G Protein-Coupled Receptor 30 in LacZ Reporter Mice

(2008) Jörg Isensee et al.   ENDOCRINOLOGY

Deletion of the G Protein-Coupled Receptor 30 Impairs Glucose Tolerance, Reduces Bone Growth, Increases Blood Pressure, and Eliminates Estradiol-Stimulated Insulin Release in Female Mice

(2008) Ulrika E. A. Mårtensson et al.   ENDOCRINOLOGY

Estrogenic control of mitochondrial function and biogenesis

(2008) Carolyn M. Klinge   JOURNAL OF CELLULAR BIOCHEMISTRY

Regulation of Steroid Hormone Biosynthesis by the Cytoskeleton

(2008) Marion B. Sewer et al.   LIPIDS

Estrogen Receptors α and β as Determinants of Gene Expression: Influence of Ligand, Dose, and Chromatin Binding

(2008) Edmund C. Chang et al.   MOLECULAR ENDOCRINOLOGY

Sterility and absence of histopathological defects in nonreproductive organs of a mouse ER -null mutant

(2008) M. C. Antal et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA