Antinociceptive effect of two novel transient receptor potential melastatin 8 antagonists in acute and chronic pain models in rat

The IUPHAR/BPS Guide to PHARMACOLOGY in 2018: updates and expansion to encompass the new guide to IMMUNOPHARMACOLOGY

(2017) Simon D Harding et al.   NUCLEIC ACIDS RESEARCH

The preventive effect of resiniferatoxin on the development of cold hypersensitivity induced by spinal nerve ligation: involvement of TRPM8

(2016) Won Uk Koh et al.   BMC NEUROSCIENCE

Role of spinal 5-HT 2 receptors subtypes in formalin-induced long-lasting hypersensitivity

(2016) Claudia Cervantes-Durán et al.   Pharmacological Reports

TRP channels: potential drug target for neuropathic pain

(2016) Lovish Marwaha et al.   INFLAMMOPHARMACOLOGY

Functional role of the transient receptor potential melastatin 8 (TRPM8) ion channel in the urinary bladder assessed by conscious cystometry andex vivomeasurements of single-unit mechanosensitive bladder afferent activities in the rat

(2015) Hiroki Ito et al.   BJU INTERNATIONAL

Experimental design and analysis and their reporting: new guidance for publication in BJP

(2015) Michael J Curtis et al.   BRITISH JOURNAL OF PHARMACOLOGY

Implementing guidelines on reporting research using animals (ARRIVE etc.): new requirements for publication in BJP

(2015) John C McGrath et al.   BRITISH JOURNAL OF PHARMACOLOGY

Antinociceptive activity of transient receptor potential channel TRPV1, TRPA1, and TRPM8 antagonists in neurogenic and neuropathic pain models in mice

(2015) Kinga Sałat et al.   Journal of Zhejiang University-SCIENCE B

AMG2850, a potent and selective TRPM8 antagonist, is not effective in rat models of inflammatory mechanical hypersensitivity and neuropathic tactile allodynia

(2015) Sonya G. Lehto et al.   NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY

TRPs and pain

(2015) Yi Dai   Seminars in Immunopathology

Evidence for the participation of Ca2+-activated chloride channels in formalin-induced acute and chronic nociception

(2014) Guadalupe García et al.   BRAIN RESEARCH

TRPM8 has a key role in experimental colitis-induced visceral hyperalgesia in mice

(2014) T. Hosoya et al.   NEUROGASTROENTEROLOGY AND MOTILITY

Operant Behavioral Responses to Orofacial Cold Stimuli in Rats with Chronic Constrictive Trigeminal Nerve Injury: Effects of Menthol and Capsazepine

(2013) Xiaozhuo Zuo et al.   Molecular Pain

The p21-activated kinase PAK 5 is involved in formalin-induced nociception through regulation of MAP-kinase signaling and formalin-specific receptors

(2012) Ovidiu Coste et al.   BEHAVIOURAL BRAIN RESEARCH

Fused Piperidines as a Novel Class of Potent and Orally Available Transient Receptor Potential Melastatin Type 8 (TRPM8) Antagonists

(2012) Nuria A. Tamayo et al.   JOURNAL OF MEDICINAL CHEMISTRY

Sensory Discrimination between Innocuous and Noxious Cold by TRPM8-Expressing DRG Neurons of Rats

(2012) Ignacio Sarria et al.   Molecular Pain

Transient Receptor Potential Melastatin 8 (TRPM8) Channels are Involved in Body Temperature Regulation

(2012) Narender R Gavva et al.   Molecular Pain

Role of TRPM8 in dorsal root ganglion in nerve injury-induced chronic pain

(2011) Lin Su et al.   BMC NEUROSCIENCE

Oxaliplatin-induced cold hypersensitivity is due to remodelling of ion channel expression in nociceptors

(2011) Juliette Descoeur et al.   EMBO Molecular Medicine

Spinal transient receptor potential ankyrin 1 channel contributes to central pain hypersensitivity in various pathophysiological conditions in the rat

(2011) Hong Wei et al.   PAIN

A novel role for TRPM8 in visceral afferent function

(2011) Andrea M. Harrington et al.   PAIN

Implication of allopregnanolone in the antinociceptive effect of N-palmitoylethanolamide in acute or persistent pain

(2011) Oscar Sasso et al.   PAIN

Cooling-Sensitive TRPM8 Is Thermostat of Skin Temperature against Cooling

(2011) Koji Tajino et al.   PLoS One

Pharmacological Blockade of TRPM8 Ion Channels Alters Cold and Cold Pain Responses in Mice

(2011) Wendy M. Knowlton et al.   PLoS One

Animal research: Reporting in vivo experiments: The ARRIVE guidelines

(2010) Carol Kilkenny et al.   BRITISH JOURNAL OF PHARMACOLOGY

Design and Optimization of Benzimidazole-Containing Transient Receptor Potential Melastatin 8 (TRPM8) Antagonists

(2010) Daniel J. Parks et al.   JOURNAL OF MEDICINAL CHEMISTRY

TRPA1 Contributes to Cold Hypersensitivity

(2010) D. del Camino et al.   JOURNAL OF NEUROSCIENCE

Ocular surface wetness is regulated by TRPM8-dependent cold thermoreceptors of the cornea

(2010) Andrés Parra et al.   NATURE MEDICINE

TRPM8, but not TRPA1, is required for neural and behavioral responses to acute noxious cold temperatures and cold-mimetics in vivo

(2010) Wendy M. Knowlton et al.   PAIN

Dose-Dependent Effects of Icilin on Thermal Preference in the Hindpaw and Face of Rats

(2009) Heather L. Rossi et al.   JOURNAL OF PAIN

Human cutaneous C fibres activated by cooling, heating and menthol

(2009) M. Campero et al.   JOURNAL OF PHYSIOLOGY-LONDON

Injury-induced mechanical hypersensitivity requires C-low threshold mechanoreceptors

(2009) Rebecca P. Seal et al.   NATURE

Involvement of increased expression of transient receptor potential melastatin 8 in oxaliplatin-induced cold allodynia in mice

(2009) Punam Gauchan et al.   NEUROSCIENCE LETTERS

Visualizing Cold Spots: TRPM8-Expressing Sensory Neurons and Their Projections

(2008) A. Dhaka et al.   JOURNAL OF NEUROSCIENCE

Pharmacological blockade of the vanilloid receptor TRPV1 elicits marked hyperthermia in humans

(2008) Narender R. Gavva et al.   PAIN