Synthesis of C2 Substituted Benzothiophenes via an Interrupted Pummerer/[3,3]-Sigmatropic/1,2-Migration Cascade of Benzothiophene S -Oxides

Dual vicinal functionalisation of heterocycles via an interrupted Pummerer coupling/[3,3]-sigmatropic rearrangement cascade

(2018) Mindaugas Šiaučiulis et al.   Chemical Science

An overview of benzo [b] thiophene-based medicinal chemistry

(2017) Rangappa S. Keri et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Ullmann-Type Intramolecular C–O Reaction Toward Thieno[3,2-b]furan Derivatives with up to Six Fused Rings

(2017) Daoliang Chen et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-catalyzed direct alkylation of heteroarenes

(2017) Cédric Theunissen et al.   Chemical Science

Metal-free O–H/C–H difunctionalization of phenols by o-hydroxyarylsulfonium salts in water

(2017) Dengfeng Chen et al.   Chemical Science

Regioselective synthesis of C3 alkylated and arylated benzothiophenes

(2017) Harry J. Shrives et al.   Nature Communications

Redox-Neutral Arylations of Vinyl Cation Intermediates

(2016) Daniel Kaiser et al.   ADVANCED SYNTHESIS & CATALYSIS

C−H Coupling Reactions Directed by Sulfoxides: Teaching an Old Functional Group New Tricks

(2016) Alexander P. Pulis et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Metal-free C–H thioarylation of arenes using sulfoxides: a direct, general diaryl sulfide synthesis

(2016) José A. Fernández-Salas et al.   CHEMICAL COMMUNICATIONS

Mild metal-catalyzed C–H activation: examples and concepts

(2016) T. Gensch et al.   CHEMICAL SOCIETY REVIEWS

Brønsted Acid-Mediated Hydrative Arylation of Unactivated Alkynes

(2016) Daniel Kaiser et al.   CHEMISTRY-A EUROPEAN JOURNAL

HOTf-Catalyzed, Solvent-Free Oxyarylation of Ynol Ethers and Thioethers

(2016) Liang Hu et al.   JOURNAL OF ORGANIC CHEMISTRY

Metal-Free Approach to Biaryls from Phenols and Aryl Sulfoxides by Temporarily Sulfur-Tethered Regioselective C–H/C–H Coupling

(2016) Tomoyuki Yanagi et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Metal-Free CH–CH-Type Cross-Coupling of Arenes and Alkynes Directed by a Multifunctional Sulfoxide Group

(2016) José A. Fernández-Salas et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Recent developments in synthetic methods for benzo[b]heteroles

(2016) Bin Wu et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

General synthesis, structure, and optical properties of benzothiophene-fused benzoheteroles containing Group 15 and 16 elements

(2016) Mio Matsumura et al.   TETRAHEDRON

Sulfoxide-directed metal-free cross-couplings in the expedient synthesis of benzothiophene-based components of materials

(2016) Andrew J. Eberhart et al.   Chemical Science

Cobalt-Catalyzed Negishi Cross-Coupling Reactions of (Hetero)Arylzinc Reagents with Primary and Secondary Alkyl Bromides and Iodides

(2015) Jeffrey M. Hammann et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis of Thieno[3,2-b]benzofurans by Palladium-catalyzed Intramolecular C–H/C–H Coupling

(2015) Hiroyuki Kaida et al.   CHEMISTRY LETTERS

Palladium-Catalyzed Construction of Heteroatom-Containing π-Conjugated Systems by Intramolecular Oxidative CH/CH Coupling Reaction

(2015) Kenta Saito et al.   CHEMISTRY-A EUROPEAN JOURNAL

Sulfoxide-Directed Metal-Freeortho-Propargylation of Aromatics and Heteroaromatics

(2015) Andrew J. Eberhart et al.   CHEMISTRY-A EUROPEAN JOURNAL

Evolution of C–H Bond Functionalization from Methane to Methodology

(2015) John F. Hartwig   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Liquid crystals for organic thin-film transistors

(2015) Hiroaki Iino et al.   Nature Communications

Organic Semiconductors Based on [1]Benzothieno[3,2-b][1]benzothiophene Substructure

(2014) Kazuo Takimiya et al.   ACCOUNTS OF CHEMICAL RESEARCH

Discovery of Desketoraloxifene Analogues as Inhibitors of Mammalian, Pseudomonas aeruginosa, and NAPE Phospholipase D Enzymes

(2014) Sarah A. Scott et al.   ACS Chemical Biology

A Brønsted Acid Catalyzed Redox Arylation

(2014) Bo Peng et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Chemoselective Intermolecular α-Arylation of Amides

(2014) Bo Peng et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Practical, Modular, and General Synthesis of Benzofurans through Extended Pummerer Annulation/Cross-Coupling Strategy

(2014) Kei Murakami et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Sulfur Mediated Allylic C–H Alkylation of Tri- and Disubstituted Olefins

(2014) Gang Hu et al.   ORGANIC LETTERS

Thionium-Based One-Pot Construction of Homo-/Heterodimeric Pyrroloindoline from Tryptamine

(2014) Masanori Tayu et al.   ORGANIC LETTERS

Metal Residues in Semiconducting Polymers: Impact on the Performance of Organic Electronic Devices

(2014) Özlem Usluer et al.   ACS Macro Letters

Nucleophilicortho-Propargylation of Aryl Sulfoxides: An Interrupted Pummerer/Allenyl Thio-Claisen Rearrangement Sequence

(2013) Andrew J. Eberhart et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Insights into the Mechanism of the Benzoannelated Thieno[3,2-b]furan Halogenation. Importance of HOMO–HOMO Interaction

(2013) Ausra Vektariene   JOURNAL OF PHYSICAL CHEMISTRY A

Iridium-Catalyzed Intermolecular Asymmetric Hydroheteroarylation of Bicycloalkenes

(2013) Christo S. Sevov et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Sulfur(IV)-Mediated Transformations: From Ylide Transfer to Metal-Free Arylation of Carbonyl Compounds

(2013) Xueliang Huang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Nucleophilic ortho-Allylation of Pyrroles and Pyrazoles: An Accelerated Pummerer/Thio-Claisen Rearrangement Sequence

(2013) Andrew J. Eberhart et al.   ORGANIC LETTERS

Iron(II) Bromide-Catalyzed Intramolecular C–H Bond Amination [1,2]-Shift Tandem Reactions of Aryl Azides

(2012) Quyen Nguyen et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Thienoacene-Based Organic Semiconductors

(2011) Kazuo Takimiya et al.   ADVANCED MATERIALS

Palladium-Catalyzed Decarboxylative CH Bond Arylation of Thiophenes

(2011) Peng Hu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Benzothiophene carboxamide derivatives as inhibitors of Plasmodium falciparum enoyl-ACP reductase

(2011) Tanushree Banerjee et al.   IUBMB LIFE

Fluorescence Properties and Dipole Moments of Novel Fused Thienobenzofurans. Solvent and Structural Effects

(2011) Jean-Jacques Aaron et al.   JOURNAL OF FLUORESCENCE

Synthesis and biological activity of some more heterocyclic compounds containing benzothiophene moiety

(2011) Gadada Naganagowda et al.   Journal of Sulfur Chemistry

Sulfoxide-Mediated α-Arylation of Carbonyl Compounds

(2011) Xueliang Huang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

NucleophilicOrthoAllylation of Aryl and Heteroaryl Sulfoxides

(2011) Andrew J. Eberhart et al.   ORGANIC LETTERS

How dual bridging atoms tune structural and optoelectronic properties of ladder-type heterotetracenes?—a theoretical study

(2011) Xian-Kai Chen et al.   PHYSICAL CHEMISTRY CHEMICAL PHYSICS

Beyond the Pummerer Reaction: Recent Developments in Thionium Ion Chemistry

(2010) Laura H. S. Smith et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

The Nickel/Copper-Catalyzed Direct Alkylation of Heterocyclic CH Bonds

(2010) Oleg Vechorkin et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Reaction of 2-(2,2,2-Trifluoroethylidene)-1,3-dithiane 1-Oxide with Ketones under Pummerer Conditions and Its Application to the Synthesis of 3-Trifluoromethyl-Substituted Five-Membered Heteroarenes

(2010) Takayuki Kobatake et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Synthesis of 3-Trifluoromethylbenzo[b]furans from Phenols via DirectOrthoFunctionalization by Extended Pummerer Reaction

(2010) Takayuki Kobatake et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Establishment of Broadly Applicable Reaction Conditions for the Palladium-Catalyzed Direct Arylation of Heteroatom-Containing Aromatic Compounds

(2009) Benoît Liégault et al.   JOURNAL OF ORGANIC CHEMISTRY

2-(2,2,2-Trifluoroethylidene)-1,3-dithiane Monoxide as a Trifluoromethylketene Equivalent

(2009) Suguru Yoshida et al.   ORGANIC LETTERS