Remote C−H Activation of Quinolines through Copper-Catalyzed Radical Cross-Coupling

Oxidative “reverse-esterification” of ethanol with benzyl/alkyl alcohols or aldehydes catalyzed by supported rhodium nanoparticles

(2016) Nitul Ranjan Guha et al.   GREEN CHEMISTRY

Sodium Iodide-Catalyzed Direct α-Alkoxylation of Ketones with AlcoholsviaOxidation of α-Iodo Ketone Intermediates

(2015) Cuiju Zhu et al.   ADVANCED SYNTHESIS & CATALYSIS

Selective remote C–H sulfonylation of aminoquinolines with arylsulfonyl chlorides via copper catalysis

(2015) Hong-Wen Liang et al.   CHEMICAL COMMUNICATIONS

H-phosphonate-mediated sulfonylation of heteroaromatic N-oxides: a mild and metal-free one-pot synthesis of 2-sulfonyl quinolines/pyridines

(2015) Kai Sun et al.   CHEMICAL COMMUNICATIONS

Copper-mediated ortho C–H sulfonylation of benzoic acid derivatives with sodium sulfinates

(2015) Jidan Liu et al.   CHEMICAL COMMUNICATIONS

Recent advances in C–S bond formation via C–H bond functionalization and decarboxylation

(2015) Chao Shen et al.   CHEMICAL SOCIETY REVIEWS

RhIII-Catalyzed C−H Olefination of Benzoic Acids under Mild Conditions using Oxygen as the Sole Oxidant

(2015) Quandi Jiang et al.   Chemistry-An Asian Journal

Palladium-Catalyzed Thioetherification of Quinolone Derivatives via Decarboxylative C−S Cross-Couplings

(2015) Chengcai Xia et al.   Chemistry-An Asian Journal

Ligand-enabled meta-C–H activation using a transient mediator

(2015) Xiao-Chen Wang et al.   NATURE

Nickel-catalyzed synthesis of diarylsulfides and sulfones via C–H bond functionalization of arylamides

(2015) Vutukuri Prakash Reddy et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Regioselective, Molecular Iodine-Mediated C3 Iodination of Quinolines

(2015) Kai Sun et al.   ORGANIC LETTERS

Copper-Mediated Remote C–H Bond Chalcogenation of Quinolines on the C5 Position

(2015) Longzhi Zhu et al.   ORGANIC LETTERS

Copper(I)-Catalyzed Sulfonylation of 8-Aminoquinoline Amides with Sulfonyl Chlorides in Air

(2015) Huijie Qiao et al.   ORGANIC LETTERS

Copper(II)-Catalyzed Direct Sulfonylation of C(sp2)–H Bonds with Sodium Sulfinates

(2015) Wei-Hao Rao et al.   ORGANIC LETTERS

Pd(II)-Catalyzed Direct Sulfonylation of Unactivated C(sp3)–H Bonds with Sodium Sulfinates

(2015) Wei-Hao Rao et al.   ORGANIC LETTERS

Palladium-catalyzed direct ortho-sulfonylation of azobenzenes with arylsulfonyl chlorides via C–H activation

(2015) Chengcai Xia et al.   RSC Advances

Remotemeta-CH Olefination of Phenylacetic Acids Directed by a Versatile U-Shaped Template

(2014) Youqian Deng et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Gold-Catalyzed Intermolecular CS Bond Formation: Efficient Synthesis of α-Substituted Vinyl Sulfones

(2014) Yumeng Xi et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Application of Fundamental Organometallic Chemistry to the Development of a Gold-Catalyzed Synthesis of Sulfinate Derivatives

(2014) Miles W. Johnson et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Copper-Catalyzed Coupling of Oxime Acetates with Sodium Sulfinates: An Efficient Synthesis of Sulfone Derivatives

(2014) Xiaodong Tang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Rhodium(III)-Catalyzed CC and CO Coupling of QuinolineN-Oxides with Alkynes: Combination of CH Activation with O-Atom Transfer

(2014) Xueyun Zhang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Iron-catalyzed aerobic difunctionalization of alkenes: a highly efficient approach to construct oxindoles by C–S and C–C bond formation

(2014) Tao Shen et al.   CHEMICAL COMMUNICATIONS

Direct regioselective phosphonation of heteroaryl N-oxides with H-phosphonates under metal and external oxidant free conditions

(2014) Hui Wang et al.   CHEMICAL COMMUNICATIONS

A highly active and easily recoverable chitosan@copper catalyst for the C–S coupling and its application in the synthesis of zolimidine

(2014) Chao Shen et al.   GREEN CHEMISTRY

Syntheses, Radiolabelings, and in Vitro Evaluations of Fluorinated PET Radioligands of 5-HT6 Serotoninergic Receptors

(2014) Julie Colomb et al.   JOURNAL OF MEDICINAL CHEMISTRY

Cu(II)–Cu(I) Synergistic Cooperation to Lead the Alkyne C–H Activation

(2014) Ruopeng Bai et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Regioselective Introduction of Heteroatoms at the C-8 Position of Quinoline N-Oxides: Remote C–H Activation Using N-Oxide as a Stepping Stone

(2014) Heejun Hwang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Conformation-induced remote meta-C–H activation of amines

(2014) Ri-Yuan Tang et al.   NATURE

Rhodium(III)-Catalyzed C–C Bond Formation of Quinoline N-Oxides at the C-8 Position under Mild Conditions

(2014) Jisu Jeong et al.   ORGANIC LETTERS

Iron-Catalyzed, Chelation-Induced Remote C–H Allylation of Quinolines via 8-Amido Assistance

(2014) Xuefeng Cong et al.   ORGANIC LETTERS

Copper-Catalyzed Direct Amination of Quinoline N-Oxides via C–H Bond Activation under Mild Conditions

(2014) Chongwei Zhu et al.   ORGANIC LETTERS

Development of an Enantioselective Hydrogenation Route to (S)-1-(2-(Methylsulfonyl)pyridin-4-yl)propan-1-amine

(2014) Jonathan T. Reeves et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

d-Glucosamine as a green ligand for copper catalyzed synthesis of aryl sulfones from aryl halides and sodium sulfinates

(2014) Ming Yang et al.   RSC Advances

Recent advances in directed C–H functionalizations using monodentate nitrogen-based directing groups

(2014) Min Zhang et al.   Organic Chemistry Frontiers

Palladium-Catalyzed Three-Component Diaryl Sulfone Synthesis Exploiting the Sulfur Dioxide Surrogate DABSO

(2013) Edward J. Emmett et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Aerobic Oxysulfonylation of Alkenes Leading to Secondary and Tertiary β-Hydroxysulfones

(2013) Qingquan Lu et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Direct 2-acetoxylation of quinoline N-oxides via copper catalyzed C–H bond activation

(2013) Xuan Chen et al.   CHEMICAL COMMUNICATIONS

Aerobic Copper-Catalyzed Organic Reactions

(2013) Scott E. Allen et al.   CHEMICAL REVIEWS

Meta-Selective C–H Functionalization Using a Nitrile-Based Directing Group and Cleavable Si-Tether

(2013) Sunggi Lee et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Cross-Coupling of Remote meta-C–H Bonds Directed by a U-Shaped Template

(2013) Li Wan et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Divergence between Organometallic and Single-Electron-Transfer Mechanisms in Copper(II)-Mediated Aerobic C–H Oxidation

(2013) Alison M. Suess et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Dioxygen-Triggered Oxidative Radical Reaction: Direct Aerobic Difunctionalization of Terminal Alkynes toward β-Keto Sulfones

(2013) Qingquan Lu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Copper-Catalyzed Intermolecular Dehydrogenative Amidation/Amination of Quinoline N-Oxides with Lactams/Cyclamines

(2013) Gang Li et al.   ORGANIC LETTERS

Synthesis of Sulfones from Organozinc Reagents, DABSO, and Alkyl Halides

(2013) Benjamin N. Rocke et al.   ORGANIC LETTERS

2,5-Bis-(sulfonyl)pyrazines as unprecedented building blocks and their SNAr reactions

(2013) Jie Jack Li et al.   TETRAHEDRON LETTERS

On the Interpretation of Deuterium Kinetic Isotope Effects in CH Bond Functionalizations by Transition-Metal Complexes

(2012) Eric M. Simmons et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Labile Cu(I) Catalyst/Spectator Cu(II) Species in Copper-Catalyzed C–C Coupling Reaction: Operando IR, in Situ XANES/EXAFS Evidence and Kinetic Investigations

(2012) Chuan He et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Activation of remote meta-C–H bonds assisted by an end-on template

(2012) Dasheng Leow et al.   NATURE

A concise, efficient synthesis of sugar-based benzothiazoles through chemoselective intramolecular C–S coupling

(2012) Chao Shen et al.   Chemical Science

Kinetic Isotope Effects in the Study of Organometallic Reaction Mechanisms

(2011) Mar Gómez-Gallego et al.   CHEMICAL REVIEWS

5-HT6 receptor and cognition

(2011) Xabier Codony et al.   CURRENT OPINION IN PHARMACOLOGY

Indolylarylsulfones as HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors: New Cyclic Substituents at Indole-2-carboxamide

(2011) Giuseppe La Regina et al.   JOURNAL OF MEDICINAL CHEMISTRY

Synthesis and Structure–Activity Relationship (SAR) of (5,7-Disubstituted 3-phenylsulfonyl-pyrazolo[1,5-a]pyrimidin-2-yl)-methylamines as Potent Serotonin 5-HT6Receptor (5-HT6R) Antagonists

(2011) Alexandre V. Ivachtchenko et al.   JOURNAL OF MEDICINAL CHEMISTRY

Copper-Mediated C–H Activation/C–S Cross-Coupling of Heterocycles with Thiols

(2011) Sadananda Ranjit et al.   JOURNAL OF ORGANIC CHEMISTRY

Ruthenium-Catalyzed Meta Sulfonation of 2-Phenylpyridines

(2011) Ourida Saidi et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthesis of Vinyl Sulfides by Copper-Catalyzed Decarboxylative C−S Cross-Coupling

(2010) Sadananda Ranjit et al.   ORGANIC LETTERS

Synthesis of Aryl Sulfides by Decarboxylative CS Cross-Couplings

(2009) Zhongyu Duan et al.   CHEMISTRY-A EUROPEAN JOURNAL

Palladium-Catalyzed Direct Arylation of Azine and AzoleN-Oxides: Reaction Development, Scope and Applications in Synthesis

(2009) Louis-Charles Campeau et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Palladium-Catalyzed C−H Bond Functionalization with Arylsulfonyl Chlorides

(2009) Xiaodan Zhao et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

A Meta-Selective Copper-Catalyzed C-H Bond Arylation

(2009) R. J. Phipps et al.   SCIENCE

5-HT6 receptor antagonists as novel cognitive enhancing agents for Alzheimer’s disease

(2008) Neil Upton et al.   Neurotherapeutics

Highly selective catalytic Friedel–Crafts sulfonylation of aromatic compounds using a FeCl3-based ionic liquid

(2008) Kiumars Bahrami et al.   TETRAHEDRON LETTERS