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Title
Efforts to Develop KRAS Inhibitors
Authors
Keywords
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Journal
Cold Spring Harbor Perspectives in Medicine
Volume 8, Issue 7, Pages a031864
Publisher
Cold Spring Harbor Laboratory
Online
2017-11-04
DOI
10.1101/cshperspect.a031864
References
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Related references
Note: Only part of the references are listed.- Inhibition of RAS function through targeting an allosteric regulatory site
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- Identification of pyrazolopyridazinones as PDEδ inhibitors
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- Selective Inhibition of Oncogenic KRAS Output with Small Molecules Targeting the Inactive State
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- (2014) Malte Schmick et al. CELL
- A Phase Ib Dose-Escalation Study of the Oral Pan-PI3K Inhibitor Buparlisib (BKM120) in Combination with the Oral MEK1/2 Inhibitor Trametinib (GSK1120212) in Patients with Selected Advanced Solid Tumors
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