Bis-isoquinolinium and bis-pyridinium acetylcholinesterase inhibitors: in vitro screening of probes for novel selective insecticides
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Title
Bis-isoquinolinium and bis-pyridinium acetylcholinesterase inhibitors: in vitro screening of probes for novel selective insecticides
Authors
Keywords
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Journal
RSC Advances
Volume 7, Issue 62, Pages 39279-39291
Publisher
Royal Society of Chemistry (RSC)
Online
2017-08-10
DOI
10.1039/c7ra05838a
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- Molecular Dynamics, Monte Carlo Simulations, and Langevin Dynamics: A Computational Review
- (2015) Eric Paquet et al. Biomed Research International
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- (2015) Sang Kwang Lee et al. BULLETIN OF THE KOREAN CHEMICAL SOCIETY
- Bispyridinium Compounds Inhibit Both Muscle and Neuronal Nicotinic Acetylcholine Receptors in Human Cell Lines
- (2015) Avi Ring et al. PLoS One
- 7-MEOTA–donepezil like compounds as cholinesterase inhibitors: Synthesis, pharmacological evaluation, molecular modeling and QSAR studies
- (2014) Jan Korabecny et al. EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
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- (2014) Daniel R Swale et al. PEST MANAGEMENT SCIENCE
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- Re-engineering aryl methylcarbamates to confer high selectivity for inhibition of Anopheles gambiae versus human acetylcholinesterase
- (2012) Joshua A. Hartsel et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Novel and Viable Acetylcholinesterase Target Site for Developing Effective and Environmentally Safe Insecticides
- (2012) Yuan-Ping Pang et al. CURRENT DRUG TARGETS
- Structures of Human Acetylcholinesterase in Complex with Pharmacologically Important Ligands
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- Cholinergic and non-cholinergic functions of two acetylcholinesterase genes revealed by gene-silencing in Tribolium castaneum
- (2012) Yanhui Lu et al. Scientific Reports
- Preparation, in vitro screening and molecular modelling of symmetrical bis-quinolinium cholinesterase inhibitors—implications for early Myasthenia gravis treatment
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- Molecular dynamics simulations and drug discovery
- (2011) Jacob D Durrant et al. BMC BIOLOGY
- The preparation,in vitroscreening and molecular docking of symmetrical bisquaternary cholinesterase inhibitors containing a but-(2E)-en-1,4-diyl connecting linkage
- (2011) Kamil Musilek et al. JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY
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- (2010) Y. H. Kim et al. INSECT MOLECULAR BIOLOGY
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- (2009) Yuan-Ping Pang et al. PLoS One
- Evidence of multiple pyrethroid resistance mechanisms in the malaria vector Anopheles gambiae sensu stricto from Nigeria
- (2008) T.S. Awolola et al. TRANSACTIONS OF THE ROYAL SOCIETY OF TROPICAL MEDICINE AND HYGIENE
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