Potent mechanism-based sirtuin-2-selective inhibition by an in situ-generated occupant of the substrate-binding site, “selectivity pocket” and NAD+-binding site
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Title
Potent mechanism-based sirtuin-2-selective inhibition by an in situ-generated occupant of the substrate-binding site, “selectivity pocket” and NAD+-binding site
Authors
Keywords
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Journal
Chemical Science
Volume 8, Issue 9, Pages 6400-6408
Publisher
Royal Society of Chemistry (RSC)
Online
2017-07-21
DOI
10.1039/c7sc02738a
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