Copper(ii)-catalyzed Chan–Lam cross-coupling: chemoselective N-arylation of aminophenols

Copper-Catalyzed CNH2Arylation of 2-Aminobenzimidazoles and Related C-Amino-NH-azoles

(2016) Desaboini Nageswar Rao et al.   ADVANCED SYNTHESIS & CATALYSIS

A quick Chan–Lam C–N and C–S cross coupling at room temperature in the presence of square pyramidal [Cu(DMAP)4I]I as a catalyst

(2016) Subhasish Roy et al.   CHEMICAL COMMUNICATIONS

Amine Directed Pd(II)-Catalyzed C–H Activation-Intramolecular Amination of N-Het(aryl)/Acyl Enaminonitriles and Enaminones: An Approach towards Multisubstituted Indoles and Heterofused Pyrroles

(2016) Somaraju Yugandar et al.   JOURNAL OF ORGANIC CHEMISTRY

Chan–Evans–Lam Amination of Boronic Acid Pinacol (BPin) Esters: Overcoming the Aryl Amine Problem

(2016) Julien C. Vantourout et al.   JOURNAL OF ORGANIC CHEMISTRY

Nickel-catalyzed Chan–Lam cross-coupling: chemoselective N-arylation of 2-aminobenzimidazoles

(2016) K. Anil Kumar et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Copper-catalyzed C–N cross-coupling of arylboronic acids with N-acylpyrazoles

(2016) Jin Zhang et al.   TETRAHEDRON LETTERS

Transition-Metal-Mediated Direct C–H Amination of Hydrocarbons with Amine Reactants: The Most Desirable but Challenging C–N Bond-Formation Approach

(2016) Hyunwoo Kim et al.   ACS Catalysis

Copper-CatalyzedN-Arylation of Tautomerizable Heterocycles with Boronic Acids and Its Application to Synthesis of Oxygenated Carbazoles

(2016) Karampoori Anil Kumar  et al.   ChemistrySelect

Visible-Light-Mediated Chan-Lam Coupling Reactions of Aryl Boronic Acids and Aniline Derivatives

(2015) Woo-Jin Yoo et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Construction of N-containing heterocycles via oxidative intramolecular N–H/X–H coupling

(2015) Jiwen Yuan et al.   CHEMICAL COMMUNICATIONS

A Synthetic Approach to N-Aryl Carbamates via Copper-Catalyzed Chan–Lam Coupling at Room Temperature

(2015) Soo-Yeon Moon et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-Catalyzed Inter- and Intramolecular C–N Bond Formation: Synthesis of Benzimidazole-Fused Heterocycles

(2015) Sk. Rasheed et al.   JOURNAL OF ORGANIC CHEMISTRY

Cu-catalyzed arylation of the amino group in the indazole ring: regioselective synthesis of pyrazolo-carbazoles

(2015) K. Anil Kumar et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Copper-catalyzed sequential N-arylation of C-amino-NH-azoles

(2014) D. Nageswar Rao et al.   CHEMICAL COMMUNICATIONS

Copper catalysed Ullmann type chemistry: from mechanistic aspects to modern development

(2014) Carlo Sambiagio et al.   CHEMICAL SOCIETY REVIEWS

The Development of Copper-Catalyzed Aerobic Oxidative Coupling of H-Tetrazoles with Boronic Acids and an Insight into the Reaction Mechanism

(2014) Chao-You Liu et al.   CHEMISTRY-A EUROPEAN JOURNAL

[Cu(OH)(TMEDA)]2Cl2-Catalyzed Regioselective 2-Arylation of 5-Substituted Tetrazoles with Boronic Acids under Mild Conditions

(2014) Takuya Onaka et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper(II)-Mediated O-Arylation of Protected Serines and Threonines

(2014) Mirna El Khatib et al.   ORGANIC LETTERS

Copper-Catalyzed Aerobic Oxidative Amination of sp3C–H Bonds: Efficient Synthesis of 2-Hetarylquinazolin-4(3H)-ones

(2014) Qiang Li et al.   ORGANIC LETTERS

Cu(i)-catalyzed intramolecular oxidative C–H amination of 2-aminoacetophenones: a convenient route toward isatins

(2013) Pang-Chi Huang et al.   CHEMICAL COMMUNICATIONS

Direct N-cyclopropylation of secondary acyclic amides promoted by copper

(2013) Emilie Racine et al.   CHEMICAL COMMUNICATIONS

C–N bond forming cross-coupling reactions: an overview

(2013) Jitender Bariwal et al.   CHEMICAL SOCIETY REVIEWS

Copper-Catalyzed Aerobic C(sp2)–H Functionalization for C–N Bond Formation: Synthesis of Pyrazoles and Indazoles

(2013) Xianwei Li et al.   JOURNAL OF ORGANIC CHEMISTRY

Selective Formation of Secondary Amides via the Copper-Catalyzed Cross-Coupling of Alkylboronic Acids with Primary Amides

(2013) Steven A. Rossi et al.   ORGANIC LETTERS

Copper-Catalyzed Oxidative Three-Component Synthesis of N, N′,N″-Trisubstituted Guanidines

(2013) Jihui Li et al.   ORGANIC LETTERS

Copper-Catalyzed Nondecarboxylative Cross Coupling of Alkenyltrifluoroborate Salts with Carboxylic Acids or Carboxylates: Synthesis of Enol Esters

(2013) Fang Huang et al.   ORGANIC LETTERS

Base and ligand free copper-catalyzed N-arylation of 2-amino-N-heterocycles with boronic acids in air

(2013) D. Nageswar Rao et al.   RSC Advances

C–N bond formation via Cu-catalyzed cross-coupling with boronic acids leading to methyl carbazole-3-carboxylate: synthesis of carbazole alkaloids

(2013) Sk. Rasheed et al.   RSC Advances

Transition metal-catalyzed N-arylations of amidines and guanidines

(2012) Tom R. M. Rauws et al.   CHEMICAL SOCIETY REVIEWS

Synthesis, biological evaluation and molecular modeling of 4,6-diarylpyrimidines and diarylbenzenes as novel non-nucleosides HIV-1 reverse transcriptase inhibitors

(2012) Sergio R. Ribone et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Microwave-Assisted One-Pot Synthesis of Isoquinolines, Furopyridines, and Thienopyridines by Palladium-Catalyzed Sequential Coupling–Imination–Annulation of 2-Bromoarylaldehydes with Terminal Acetylenes and Ammonium Acetate

(2012) Dingqiao Yang et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-Catalyzed Sequential Ullmann N-Arylation and Aerobic Oxidative C–H Amination: A Convenient Route to Indolo[1,2-c]quinazoline Derivatives

(2012) Peng Sang et al.   ORGANIC LETTERS

Copper Catalyzed N-Arylation of Amidines with Aryl Boronic Acids and One-Pot Synthesis of Benzimidazoles by a Chan–Lam–Evans N-Arylation and C–H Activation/C–N Bond Forming Process

(2012) Jihui Li et al.   ORGANIC LETTERS

The Complementary Competitors: Palladium and Copper in C–N Cross-Coupling Reactions

(2012) Irina P. Beletskaya et al.   ORGANOMETALLICS

Chan–Lam coupling reactions: synthesis of heterocycles

(2012) Kodepelly Sanjeeva Rao et al.   TETRAHEDRON

Palladium-catalyzed aerobic oxidative C–H amination: synthesis of 2-unsubstituted and 2-substituted N-aryl benzimidazoles

(2012) Rapolu Kiran Kumar et al.   RSC Advances

Palladium- and copper-mediatedN-aryl bond formation reactions for the synthesis of biological active compounds

(2011) Carolin Fischer et al.   Beilstein Journal of Organic Chemistry

On the Importance of an Acid Additive in the Synthesis of Pyrido[1,2-a]benzimidazoles by Direct Copper-Catalyzed Amination

(2011) Kye-Simeon Masters et al.   CHEMISTRY-A EUROPEAN JOURNAL

Pd-Catalyzed Intramolecular Oxidative C–H Amination: Synthesis of Carbazoles

(2011) So Won Youn et al.   ORGANIC LETTERS

Copper-Catalyzed Aerobic Oxidative Intramolecular C–H Amination Leading to Imidazobenzimidazole Derivatives

(2011) Xiaoqiang Wang et al.   ORGANIC LETTERS

Copper-Catalyzed Direct Synthesis of Di- and Triphenylamines: A Dramatic Accelerating Effect of 2-Aminophenols

(2010) Yaming Li et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Targeted cancer therapies

(2010) Saurabh Aggarwal   NATURE REVIEWS DRUG DISCOVERY

Copper-Promoted Carbon-Heteroatom Bond Cross-Coupling with Boronic Acids and Derivatives

(2010) Jennifer Qiao et al.   SYNTHESIS-STUTTGART

Amine directed Pd(ii)-catalyzed C–H bond functionalization under ambient conditions

(2010) Benjamin Haffemayer et al.   Chemical Science

Dialkylbiaryl phosphines in Pd-catalyzed amination: a user's guide

(2010) David S. Surry et al.   Chemical Science

Catalytic CC, CN, and CO Ullmann-Type Coupling Reactions

(2009) Florian Monnier et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Kinase Domain Mutations in Cancer: Implications for Small Molecule Drug Design Strategies

(2009) Jack A. Bikker et al.   JOURNAL OF MEDICINAL CHEMISTRY

Mechanistic Study of Copper-Catalyzed Aerobic Oxidative Coupling of Arylboronic Esters and Methanol: Insights into an Organometallic Oxidase Reaction

(2009) Amanda E. King et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Orthogonal Cu- and Pd-Based Catalyst Systems for the O- and N-Arylation of Aminophenols

(2009) Debabrata Maiti et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Facile Synthesis of 1,2,4-Triazoles via a Copper-Catalyzed Tandem Addition−Oxidative Cyclization

(2009) Satoshi Ueda et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Evolution of a Fourth Generation Catalyst for the Amination and Thioetherification of Aryl Halides

(2008) John F. Hartwig   ACCOUNTS OF CHEMICAL RESEARCH

Biaryl Phosphane Ligands in Palladium-Catalyzed Amination

(2008) David S. Surry et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION