One-pot strategy of copper-catalyzed synthesis of 1,2-disubstituted benzimidazoles

Synthesis and investigation of novel benzimidazole derivatives as antifungal agents

(2016) Nishad Thamban Chandrika et al.   BIOORGANIC & MEDICINAL CHEMISTRY

Synthesis, binding assays, cytotoxic activity and docking studies of benzimidazole and benzothiophene derivatives with selective affinity for the CB2 cannabinoid receptor

(2016) Javier Romero-Parra et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Catalytic Oxidative Coupling of Primary Amines under Air: A Flexible Route to Benzimidazole Derivatives

(2016) Khac Minh Huy Nguyen et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Rapid production of benzazole derivatives by a high-pressure and high-temperature water microflow chemical process

(2016) I. Nagao et al.   GREEN CHEMISTRY

Copper-catalyzed tandem Ullmann type C–N coupling and dehydrative cyclization: synthesis of imidazo[1,2-c]quinazolines

(2016) Nitesh K. Nandwana et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Synthesis of benzimidazole-based 1,3,4-oxadiazole-1,2,3-triazole conjugates as glycogen synthase kinase-3β inhibitors with antidepressant activity in in vivo models

(2016) Mushtaq A. Tantray et al.   RSC Advances

Synthesis andIn VitroActivity of Polyhalogenated 2-phenylbenzimidazoles as a New Class of anti-MRSA and Anti-VRE Agents

(2015) Hakan Göker et al.   Chemical Biology & Drug Design

Iron catalyzed oxidative assembly of N-heteroaryl and aryl metal reagents using oxygen as an oxidant

(2015) Kun Ming Liu et al.   CHEMICAL COMMUNICATIONS

A Bioinspired Catalytic Aerobic Oxidative CH Functionalization of Primary Aliphatic Amines: Synthesis of 1,2-Disubstituted Benzimidazoles

(2015) Khac Minh Huy Nguyen et al.   CHEMISTRY-A EUROPEAN JOURNAL

Synergetic catalytic effect of ionic liquids and ZnO nanoparticles on the selective synthesis of 1,2-disubstituted benzimidazoles using a ball-milling technique

(2015) Hemant Sharma et al.   GREEN CHEMISTRY

Benzimidazoles and benzoxazoles via the nucleophilic addition of anilines to nitroalkanes

(2015) Alexander V. Aksenov et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

One-Pot Synthesis of Pyrrolo[1,2-a]quinoxaline Derivatives via a Copper-Catalyzed Aerobic Oxidative Domino Reaction

(2015) Huanhuan Liu et al.   ORGANIC LETTERS

Carbon nanotube-based QuEChERS extraction and enhanced product ion scan-assisted confirmation of multi-pesticide residue in dried tangerine peel

(2015) Xiaowen Dou et al.   RSC Advances

Synthesis of 2-arylbenzimidazoles under mild conditions catalyzed by a heteropolyacid-containing task-specific ionic liquid and catalyst investigation by electrospray (tandem) mass spectrometry

(2015) Haline G. O. Alvim et al.   RSC Advances

Selenadiazole derivatives as potent thioredoxin reductase inhibitors that enhance the radiosensitivity of cancer cells

(2014) Yuan-Wei Liang et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Structure Guided Design and Kinetic Analysis of Highly Potent Benzimidazole Inhibitors Targeting the PDEδ Prenyl Binding Site

(2014) Gunther Zimmermann et al.   JOURNAL OF MEDICINAL CHEMISTRY

Copper-Catalyzed Three-Component Synthesis of Benzothiazolethiones from o-Iodoanilines, Isocyanide, and Potassium Sulfide

(2014) Pan Dang et al.   ORGANIC LETTERS

Convenient Synthesis of Benzothiazoles and Benzimidazoles through Brønsted Acid Catalyzed Cyclization of 2-Amino Thiophenols/Anilines with β-Diketones

(2014) Muhammad Shareef Mayo et al.   ORGANIC LETTERS

Solvent/Oxidant-Switchable Synthesis of Multisubstituted Quinazolines and Benzimidazoles via Metal-Free Selective Oxidative Annulation of Arylamidines

(2014) Jian-Ping Lin et al.   ORGANIC LETTERS

Benzimidazole CB2 agonists: Design, synthesis and SAR

(2013) Kausik K. Nanda et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

“All-water” one-pot diverse synthesis of 1,2-disubstituted benzimidazoles: hydrogen bond driven ‘synergistic electrophile–nucleophile dual activation’ by water

(2013) Damodara N. Kommi et al.   GREEN CHEMISTRY

Small molecule inhibition of the KRAS–PDEδ interaction impairs oncogenic KRAS signalling

(2013) Gunther Zimmermann et al.   NATURE

An Efficient One-Pot Synthesis of Benzo[4,5]imidazo[1,2-a]quinoxalines via Copper-Catalyzed Process

(2013) Aiping Huang et al.   ORGANIC LETTERS

Catalyst-Free N-Arylation Using Unactivated Fluorobenzenes

(2012) Frederik Diness et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Dimeric 1,3-Phenylene-bis(piperazinyl benzimidazole)s: Synthesis and Structure–Activity Investigations on their Binding with Human Telomeric G-Quadruplex DNA and Telomerase Inhibition Properties

(2012) Akash K Jain et al.   JOURNAL OF MEDICINAL CHEMISTRY

Palladium-Catalyzed Synthesis of Benzimidazoles and Quinazolinones from Common Precursors

(2012) Jessie E. R. Sadig et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of 3-Substituted and 2,3-Disubstituted Quinazolinones via Cu-Catalyzed Aryl Amidation

(2012) Lanting Xu et al.   ORGANIC LETTERS

Exploration of in vitro time point quantitative evaluation of newly synthesized benzimidazole and benzothiazole derivatives as potential antibacterial agents

(2011) Prabal Bandyopadhyay et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Optimisation of a novel series of selective CNS penetrant CB2 agonists

(2011) Christine Watson et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Building Heterocyclic Systems with RC(OR)2+ Carbocations in Recyclable Brønsted Acidic Ionic Liquids: Facile Synthesis of 1-Substituted 1H-1,2,3,4-Tetrazoles, Benzazoles and Other Ring Systems with CH(OEt)3 and EtC(OEt)3 in [EtNH3][NO3] and [PMIM(SO3H)][O

(2011) Gopalakrishnan Aridoss et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Copper-Mediated Synthesis of Substituted 2-Aryl-N-benzylbenzimidazoles and 2-Arylbenzoxazoles via C–H Functionalization/C–N/C–O Bond Formation

(2011) Murali Mohan Guru et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of 1,2-disubstituted benzimidazoles, 2-substituted benzimidazoles and 2-substituted benzothiazoles in SDS micelles

(2010) Kiumars Bahrami et al.   GREEN CHEMISTRY

Copper-Catalyzed Synthesis of Quinazoline Derivatives via Ullmann-Type Coupling and Aerobic Oxidation

(2010) Chen Wang et al.   JOURNAL OF ORGANIC CHEMISTRY

Small Molecular Glasses Based on Multiposition Encapsulated Phenyl Benzimidazole Iridium(III) Complexes: Toward Efficient Solution-Processable Host-Free Electrophosphorescent Diodes

(2009) Hui Xu et al.   JOURNAL OF PHYSICAL CHEMISTRY B

Cross-coupling reaction of alcohols for carbon–carbon bond formation using pincer-type NHC/palladium catalysts

(2009) Osamu Kose et al.   ORGANIC & BIOMOLECULAR CHEMISTRY