Developing Spindlin1 small-molecule inhibitors by using protein microarrays
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Title
Developing Spindlin1 small-molecule inhibitors by using protein microarrays
Authors
Keywords
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Journal
Nature Chemical Biology
Volume 13, Issue 7, Pages 750-756
Publisher
Springer Nature
Online
2017-05-15
DOI
10.1038/nchembio.2377
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Related references
Note: Only part of the references are listed.- Molecular Recognition of Lys and Arg Methylation
- (2016) Joshua E. Beaver et al. ACS Chemical Biology
- Identification and Structure-Activity Relationship Studies of Small-Molecule Inhibitors of the Methyllysine Reader Protein Spindlin1
- (2016) Dina Robaa et al. ChemMedChem
- A cellular chemical probe targeting the chromodomains of Polycomb repressive complex 1
- (2016) Jacob I Stuckey et al. Nature Chemical Biology
- Identification of a small-molecule ligand of the epigenetic reader protein Spindlin1 via a versatile screening platform
- (2016) Tobias Wagner et al. NUCLEIC ACIDS RESEARCH
- Reading the Combinatorial Histone Language
- (2015) Zhangli Su et al. ACS Chemical Biology
- Identification of a Fragment-like Small Molecule Ligand for the Methyl-lysine Binding Protein, 53BP1
- (2015) Michael T. Perfetti et al. ACS Chemical Biology
- Chemical Inhibitors of Epigenetic Methyllysine Reader Proteins
- (2015) Natalia Milosevich et al. BIOCHEMISTRY
- Quantitative Proteomic Analysis of Histone Modifications
- (2015) He Huang et al. CHEMICAL REVIEWS
- Structure-Guided Design of IACS-9571, a Selective High-Affinity Dual TRIM24-BRPF1 Bromodomain Inhibitor
- (2015) Wylie S. Palmer et al. JOURNAL OF MEDICINAL CHEMISTRY
- Targeting histone lysine methylation in cancer
- (2015) John McGrath et al. PHARMACOLOGY & THERAPEUTICS
- The histone code reader SPIN1 controls RET signaling in liposarcoma
- (2015) Henriette Franz et al. Oncotarget
- Competitive Binding of a Benzimidazole to the Histone-Binding Pocket of the Pygo PHD Finger
- (2014) Thomas C. R. Miller et al. ACS Chemical Biology
- Hitting the ‘mark’: Interpreting lysine methylation in the context of active transcription
- (2014) Glenn G. Wozniak et al. Biochimica et Biophysica Acta-Gene Regulatory Mechanisms
- Towards understanding methyllysine readout
- (2014) Catherine A. Musselman et al. Biochimica et Biophysica Acta-Gene Regulatory Mechanisms
- Molecular basis underlying histone H3 lysine-arginine methylation pattern readout by Spin/Ssty repeats of Spindlin1
- (2014) X. Su et al. GENES & DEVELOPMENT
- Chromodomain Antagonists That Target the Polycomb-Group Methyllysine Reader Protein Chromobox Homolog 7 (CBX7)
- (2014) Chakravarthi Simhadri et al. JOURNAL OF MEDICINAL CHEMISTRY
- The cellular thermal shift assay for evaluating drug target interactions in cells
- (2014) Rozbeh Jafari et al. Nature Protocols
- Discovery and Development of Potent and Selective Inhibitors of Histone Methyltransferase G9a
- (2014) Ramzi F. Sweis et al. ACS Medicinal Chemistry Letters
- Chromatin proteins and modifications as drug targets
- (2013) Kristian Helin et al. NATURE
- Discovery of a chemical probe for the L3MBTL3 methyllysine reader domain
- (2013) Lindsey I James et al. Nature Chemical Biology
- Emerging patterns of somatic mutations in cancer
- (2013) Ian R. Watson et al. NATURE REVIEWS GENETICS
- A Tudor Domain Protein SPINDLIN1 Interacts with the mRNA-Binding Protein SERBP1 and Is Involved in Mouse Oocyte Meiotic Resumption
- (2013) Ting Gang Chew et al. PLoS One
- Monitoring Drug Target Engagement in Cells and Tissues Using the Cellular Thermal Shift Assay
- (2013) D. M. Molina et al. SCIENCE
- Identification and Characterization of Small Molecule Inhibitors of a Plant Homeodomain Finger
- (2012) Elise K. Wagner et al. BIOCHEMISTRY
- SPINDLIN1 Promotes Cancer Cell Proliferation through Activation of WNT/TCF-4 Signaling
- (2012) J.-X. Wang et al. MOLECULAR CANCER RESEARCH
- Perceiving the epigenetic landscape through histone readers
- (2012) Catherine A Musselman et al. NATURE STRUCTURAL & MOLECULAR BIOLOGY
- Readers of histone modifications
- (2011) Miyong Yun et al. CELL RESEARCH
- Nucleolar protein Spindlin1 recognizes H3K4 methylation and stimulates the expression of rRNA genes
- (2011) Weixiang Wang et al. EMBO REPORTS
- Druggability of methyl-lysine binding sites
- (2011) C. Santiago et al. JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN
- Small-Molecule Ligands of Methyl-Lysine Binding Proteins
- (2011) J. Martin Herold et al. JOURNAL OF MEDICINAL CHEMISTRY
- PHENIX: a comprehensive Python-based system for macromolecular structure solution
- (2010) Paul D. Adams et al. ACTA CRYSTALLOGRAPHICA SECTION D-BIOLOGICAL CRYSTALLOGRAPHY
- Identification of Non-Peptide Malignant Brain Tumor (MBT) Repeat Antagonists by Virtual Screening of Commercially Available Compounds
- (2010) Dmitri Kireev et al. JOURNAL OF MEDICINAL CHEMISTRY
- Selective inhibition of BET bromodomains
- (2010) Panagis Filippakopoulos et al. NATURE
- Molecular replacement withMOLREP
- (2009) Alexei Vagin et al. ACTA CRYSTALLOGRAPHICA SECTION D-BIOLOGICAL CRYSTALLOGRAPHY
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