Synthesis of trifluoromethylated isoxazoles and their elaboration through inter- and intra-molecular C–H arylation

18F-Labeling of Arenes and Heteroarenes for Applications in Positron Emission Tomography

(2016) Sean Preshlock et al.   CHEMICAL REVIEWS

Asymmetric 18F-fluorination for applications in positron emission tomography

(2016) Faye Buckingham et al.   Chemical Science

Recent Developments in the Synthesis and Reactivity of Isoxazoles: Metal Catalysis and Beyond

(2015) Feng Hu et al.   ADVANCED SYNTHESIS & CATALYSIS

Late-Stage Fluorination: Fancy Novelty or Useful Tool?

(2015) Constanze N. Neumann et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Modular, Concise, and Efficient Synthesis of Highly Functionalized 5-Fluoropyridazines by a [2 + 1]/[3 + 2]-Cycloaddition Sequence

(2015) Gaël Tran et al.   ORGANIC LETTERS

Advances in Catalytic Enantioselective Fluorination, Mono-, Di-, and Trifluoromethylation, and Trifluoromethylthiolation Reactions

(2014) Xiaoyu Yang et al.   CHEMICAL REVIEWS

Synthetic Methods for Compounds Having CF3–S Units on Carbon by Trifluoromethylation, Trifluoromethylthiolation, Triflylation, and Related Reactions

(2014) Xiu-Hua Xu et al.   CHEMICAL REVIEWS

Late-Stage Fluorination: From Fundamentals to Application

(2014) Michael G. Campbell et al.   ORGANIC PROCESS RESEARCH & DEVELOPMENT

Sandmeyer Trifluoromethylation of Arenediazonium Tetrafluoroborates

(2013) Grégory Danoun et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

The Trifluoromethylating Sandmeyer Reaction: A Method for Transforming CN into CCF3

(2013) Duncan L. Browne   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Introduction of Fluorine and Fluorine-Containing Functional Groups

(2013) Theresa Liang et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Fluorine in Pharmaceutical Industry: Fluorine-Containing Drugs Introduced to the Market in the Last Decade (2001–2011)

(2013) Jiang Wang et al.   CHEMICAL REVIEWS

Total Synthesis of Calothrixin A and B via C–H Activation

(2013) Nagarajan Ramkumar et al.   JOURNAL OF ORGANIC CHEMISTRY

Copper-Promoted Sandmeyer Trifluoromethylation Reaction

(2013) Jian-Jun Dai et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Silver-Mediated Trifluoromethylation of Aryldiazonium Salts: Conversion of Amino Group into Trifluoromethyl Group

(2013) Xi Wang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Synthesis of Trifluoromethylated Isoxazolidines: 1,3-Dipolar Cycloaddition of Nitrosoarenes, (Trifluoromethyl)diazomethane, and Alkenes

(2013) Gary A. Molander et al.   ORGANIC LETTERS

Fluorine Scanning by Nonselective Fluorination: Enhancing Raf/MEK Inhibition while Keeping Physicochemical Properties

(2013) Ikumi Hyohdoh et al.   ACS Medicinal Chemistry Letters

Molecular Design of Photovoltaic Materials for Polymer Solar Cells: Toward Suitable Electronic Energy Levels and Broad Absorption

(2012) Yongfang Li   ACCOUNTS OF CHEMICAL RESEARCH

Synthesis and Use of a Trifluoromethylated Azomethine Ylide Precursor

(2012) Gaël Tran et al.   JOURNAL OF ORGANIC CHEMISTRY

Palladium-Catalyzed Direct Arylation of Heteroaromatics with Activated Aryl Chlorides Using a Sterically Relieved Ferrocenyl-Diphosphane

(2012) David Roy et al.   ACS Catalysis

The fluorous effect in biomolecular applications

(2011) Massimo Cametti et al.   CHEMICAL SOCIETY REVIEWS

Fluorination of elastomer materials

(2011) Sandra Schlögl et al.   EUROPEAN POLYMER JOURNAL

Synopsis of Some Recent Tactical Application of Bioisosteres in Drug Design

(2011) Nicholas A. Meanwell   JOURNAL OF MEDICINAL CHEMISTRY

Cascade Palladium-Catalyzed Direct Intramolecular Arylation/Alkene Isomerization Sequences: Synthesis of Indoles and Benzofurans

(2010) Myriam Yagoubi et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

Fluorine in health care: Organofluorine containing blockbuster drugs

(2010) David O’Hagan   JOURNAL OF FLUORINE CHEMISTRY

Synthesis of Unsymmetricalo-Biphenols ando-Binaphthols via Silicon-Tethered Pd-Catalyzed C−H Arylation

(2010) Chunhui Huang et al.   ORGANIC LETTERS

Fluorinated high-performance polymers: Poly(arylene ether)s and aromatic polyimides containing trifluoromethyl groups

(2010) Mahua G. Dhara et al.   PROGRESS IN POLYMER SCIENCE

Ligand-Free-Palladium-Catalyzed Direct 4-Arylation of Isoxazoles Using Aryl Bromides

(2009) Yacoub Fall et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Fluorine in medicinal chemistry: a century of progress and a 60-year retrospective of selected highlights

(2009) Robert Filler et al.   Future Medicinal Chemistry

One-Pot Synthesis of α-Carbolines via Sequential Palladium-Catalyzed Aryl Amination and Intramolecular Arylation

(2009) Joydev K. Laha et al.   JOURNAL OF ORGANIC CHEMISTRY

Domino Palladium-Catalyzed Heck-Intermolecular Direct Arylation Reactions

(2009) Olivier René et al.   ORGANIC LETTERS

Palladium-Catalyzed Direct C-4 Arylation of 2,5-Disubstituted Furans with Aryl Bromides

(2008) Aditya L. Gottumukkala et al.   ADVANCED SYNTHESIS & CATALYSIS

The Many Roles for Fluorine in Medicinal Chemistry

(2008) William K. Hagmann   JOURNAL OF MEDICINAL CHEMISTRY

Diversity-oriented synthesis; a spectrum of approaches and results

(2008) Richard J. Spandl et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Fluorination in Medicinal Chemistry: Methods, Strategies, and Recent Developments

(2008) Kenneth L. Kirk   ORGANIC PROCESS RESEARCH & DEVELOPMENT

N,N-Disubstituted propargylamines as tools in the sequential 1,3-dipolar cycloaddition/arylation processes to the formation of polyheterocyclic systems

(2008) Luca Basolo et al.   TETRAHEDRON

Mild and efficient palladium-catalyzed intramolecular direct arylation reactions

(2008) Marc Lafrance et al.   TETRAHEDRON

Fluorine in medicinal chemistry

(2007) Sophie Purser et al.   CHEMICAL SOCIETY REVIEWS