2,5-Disubstituted furan derivatives containing imidazole, triazole or tetrazole moiety as potent α-glucosidase inhibitors

A review on synthesis, mechanism of action, and structure-activity relationships of 1,2,3-triazole-based α-glucosidase inhibitors as promising anti-diabetic agents

(2022) Zari Fallah et al.   JOURNAL OF MOLECULAR STRUCTURE

Design, synthesis and bioactivity study on 5-phenylfuran derivatives as potent reversal agents against P-glycoprotein-mediated multidrug resistance in MCF-7/ADR cell

(2021) Ya-Sheng Li et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

2,5-Disubstituted furan derivatives containing 1,3,4-thiadiazole moiety as potent α-glucosidase and E. coli β-glucuronidase inhibitors

(2021) Ya-Sheng Li et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Rational design of phenyl thiophene (pyridine) derivatives that overcome P-glycoprotein mediated MDR in MCF-7/ADR cell

(2021) Ya-Sheng Li et al.   BIOORGANIC CHEMISTRY

Discovery of a series of 5-phenyl-2-furan derivatives containing 1,3-thiazole moiety as potent Escherichia coli β-glucuronidase inhibitors

(2021) Tao-Shun Zhou et al.   BIOORGANIC CHEMISTRY

Screening of α‐Glucosidase Inhibitors from Houttuynia cordata and Evaluation of the Binding Mechanisms

(2020) Xueli Zhang et al.   ChemistrySelect

Synthesis and bioactivity of phenyl substituted furan and oxazole carboxylic acid derivatives as potential PDE4 inhibitors

(2020) Yinuo Lin et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Synthetic heterocyclic candidates as promising α-glucosidase inhibitors: An overview

(2019) Manoj Dhameja et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Novel S-Thiazol-2-yl-furan-2-carbothioate Derivatives as Potential T3SS Inhibitors Against Xanthomonas oryzae on Rice

(2019) Shan Jiang et al.   JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY

Biological evaluation of new imidazole derivatives tethered with indole moiety as potent α-glucosidase inhibitors

(2018) Sadia Naureen et al.   BIOORGANIC CHEMISTRY

A simple and efficient synthesis of benzimidazoles containing piperazine or morpholine skeleton at C-6 position as glucosidase inhibitors with antioxidant activity

(2018) Musa Özil et al.   BIOORGANIC CHEMISTRY

Potential of Potentilla inclinata and its polyphenolic compounds in α-glucosidase inhibition: Kinetics and interaction mechanism merged with docking simulations

(2018) Didem Şöhretoğlu et al.   INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES

Benzimidazole derivatives as new α-glucosidase inhibitors and in silico studies

(2016) Nik Khairunissa Nik Abdullah Zawawi et al.   BIOORGANIC CHEMISTRY

Inhibitory kinetics and mechanism of kaempferol on α-glucosidase

(2016) Xi Peng et al.   FOOD CHEMISTRY

Design, synthesis, α-glucosidase inhibitory activity, molecular docking and QSAR studies of benzimidazole derivatives

(2016) Leila Dinparast et al.   JOURNAL OF MOLECULAR STRUCTURE

Development of a credible 3D-QSAR CoMSIA model and docking studies for a series of triazoles and tetrazoles containing 11β-HSD1 inhibitors

(2016) P. R. Murumkar et al.   SAR AND QSAR IN ENVIRONMENTAL RESEARCH

Food protein-derived bioactive peptides in management of type 2 diabetes

(2015) Prasad Patil et al.   EUROPEAN JOURNAL OF NUTRITION

DPP-4 inhibitor and alpha-glucosidase inhibitor equally improve endothelial function in patients with type 2 diabetes: EDGE study

(2014) Kazufumi Nakamura et al.   Cardiovascular Diabetology

Design, synthesis, in silico molecular docking and biological evaluation of novel oxadiazole based thiazolidine-2,4-diones bis-heterocycles as PPAR-γ agonists

(2014) Syed Nazreen et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Advances in the cellular immunological pathogenesis of type 1 diabetes

(2014) Min Li et al.   JOURNAL OF CELLULAR AND MOLECULAR MEDICINE

Synthesis and structure–activity relationship of 2-adamantylmethyl tetrazoles as potent and selective inhibitors of human 11β-hydroxysteroid dehydrogenase type 1 (11β-HSD1)

(2013) Xiang-Yang Ye et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Inhibition of α-glucosidase and α-amylase by diaryl derivatives of imidazole-thione and 1,2,4-triazole-thiol

(2011) Mahmoud Balba et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Crystal structures of isomaltase from Saccharomyces cerevisiae and in complex with its competitive inhibitor maltose

(2010) Keizo Yamamoto et al.   FEBS Journal