(NH4)2S2O8-Mediated Metal-Free Decarboxylative Formylation/Acylation of α-Oxo/Ketoacids and Its Application to the Synthesis of Indole Alkaloids

Recent Advances in the Synthesis of β-Carboline Alkaloids

(2021) Tímea Szabó et al.   MOLECULES

Photo-on-Demand Synthesis of Vilsmeier Reagents with Chloroform and Their Applications to One-Pot Organic Syntheses

(2021) Fengying Liang et al.   JOURNAL OF ORGANIC CHEMISTRY

Decarboxylative Coupling of Glyoxylic Acid and Its Acetal Derivatives: A Unique C1 Formylation Synthon

(2021) Yunyu Xiang et al.   TETRAHEDRON

Metal-, Photocatalyst-, and Light-Free Minisci C–H Acetylation of N-Heteroarenes with Vinyl Ethers

(2021) Jianyang Dong et al.   ORGANIC LETTERS

A comprehensive overview of β-carbolines and its derivatives as anticancer agents

(2021) Bo Luo et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Direct C–H Functionalization of Phenanthrolines: Metal- and Light-Free Dicarbamoylations

(2021) David T. Mooney et al.   JOURNAL OF ORGANIC CHEMISTRY

Photoredox‐Catalyzed Redox‐Neutral Minisci C−H Formylation of N ‐Heteroarenes

(2020) Jianyang Dong et al.   ADVANCED SYNTHESIS & CATALYSIS

Aroylation of Electron-Rich Pyrroles under Minisci Reaction Conditions

(2020) Joydev K. Laha et al.   ORGANIC LETTERS

Iron-Catalyzed Minisci Type Acetylation of N -Heteroarenes Mediated by CH(OEt)3 /TBHP

(2019) A. Srinivasulu et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Recent Advances in Minisci-Type Reactions

(2019) Rupert S. J. Proctor et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

α-Keto Acids: Acylating Agents in Organic Synthesis

(2019) Filipe Penteado et al.   CHEMICAL REVIEWS

Visible-Light-Mediated Direct Decarboxylative Acylation of Electron-Deficient Heteroarenes Using α-Ketoacids

(2019) Sabyasachi Manna et al.   JOURNAL OF ORGANIC CHEMISTRY

First total synthesis of the β-carboline alkaloids trigonostemine A, trigonostemine B and a new synthesis of pityriacitrin and hyrtiosulawesine

(2019) Tímea Szabó et al.   TETRAHEDRON LETTERS

Synthesis of 3-Formylindoles via Electrochemical Decarboxylation of Glyoxylic Acid with an Amine as a Dual Function Organocatalyst

(2019) Dian-Zhao Lin et al.   ORGANIC LETTERS

Metal-, Photocatalyst-, and Light-Free Direct C–H Acylation and Carbamoylation of Heterocycles

(2019) Matthew T. Westwood et al.   ORGANIC LETTERS

Nickel-catalyzed electrochemical Minisci acylation of aromatic N-heterocycles with α-keto acids via ligand-to-metal electron transfer pathway

(2019) Hang Ding et al.   JOURNAL OF CATALYSIS

Palladium-catalyzed hydroformylation of terminal arylacetylenes with glyoxylic acid

(2018) Yang Liu et al.   CHEMICAL COMMUNICATIONS

Decarboxylative reactions with and without light – a comparison

(2018) Johanna Schwarz et al.   GREEN CHEMISTRY

Advances in Decarboxylative Oxidative Coupling Reaction

(2018) Tong Zhang et al.   JOURNAL OF ORGANIC CHEMISTRY

Selective nickel-catalyzed dehydrogenative–decarboxylative formylation of indoles with glyoxylic acid

(2018) Zhiping Yin et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Electrochemical N-Formylation of Amines via Decarboxylation of Glyoxylic Acid

(2018) Dian-Zhao Lin et al.   ORGANIC LETTERS

Decarboxylative formylation of aryl halides with glyoxylic acid by merging organophotoredox with palladium catalysis

(2018) Bin Zhao et al.   Organic Chemistry Frontiers

Copper/Persulfate-Promoted Oxidative Decarboxylative C−H Acylation of Pyrazolones with α-Oxocarboxylic Acids: Direct Access to 4-Acylpyrazolones under Mild Conditions

(2018) Tanakorn Kittikool et al.   ADVANCED SYNTHESIS & CATALYSIS

Metal- and Acid-Free C–H Formylation of Nitrogen Heterocycles: Using Trioxane as an Aldehyde Equivalent Enabled by an Organic-Soluble Oxidant

(2018) Jacob M. Ganley et al.   ORGANIC LETTERS

Photoredox-Catalyzed Decarboxylative C–H Acylation of Heteroarenes

(2018) Chao Yang et al.   SYNLETT

Metal-, Photocatalyst-, and Light-Free, Late-Stage C–H Alkylation of Heteroarenes and 1,4-Quinones Using Carboxylic Acids

(2018) Daniel R. Sutherland et al.   ORGANIC LETTERS

Chemo- and Regioselective Organo-Photoredox Catalyzed Hydroformylation of Styrenes via a Radical Pathway

(2017) He Huang et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Diverse Secondary Metabolites from the Marine-Derived Fungus Dichotomomyces cejpii F31-1

(2017) Yan-Xiu Chen et al.   Marine Drugs

Intramolecular Minisci acylation under silver-free neutral conditions for the synthesis of azafluorenones and fluorenones

(2017) Joydev K. Laha et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Electrocatalytic Minisci Acylation Reaction of N-Heteroarenes Mediated by NH4I

(2017) Qing-Qing Wang et al.   ORGANIC LETTERS

Iron-Catalyzed C3-Formylation of Indoles with Formaldehyde and Aqueous Ammonia under Air

(2017) Jin-Ming Yang et al.   SYNLETT

Visible Light-Mediated Direct Decarboxylative C–H Functionalization of Heteroarenes

(2017) R. Aleyda Garza-Sanchez et al.   ACS Catalysis

Decarboxylative Coupling ofα-Keto Acids withortho-Phenylenediamines Promoted by an Electrochemical Method in Aqueous Media

(2016) Hai-Bin Wang et al.   ADVANCED SYNTHESIS & CATALYSIS

Copper mediated decarboxylative direct C–H arylation of heteroarenes with benzoic acids

(2016) Tuhin Patra et al.   CHEMICAL COMMUNICATIONS

Recent advances in catalytic decarboxylative acylation reactions via a radical process

(2016) Li-Na Guo et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

Regiospecific Benzoylation of Electron-Deficient N-Heterocycles with Methylbenzenes via a Minisci-Type Reaction

(2015) Wajid Ali et al.   JOURNAL OF ORGANIC CHEMISTRY

Analysis of the Structural Diversity, Substitution Patterns, and Frequency of Nitrogen Heterocycles among U.S. FDA Approved Pharmaceuticals

(2014) Edon Vitaku et al.   JOURNAL OF MEDICINAL CHEMISTRY

A Transition Metal-Free Minisci Reaction: Acylation of Isoquinolines, Quinolines, and Quinoxaline

(2014) Yogesh Siddaraju et al.   JOURNAL OF ORGANIC CHEMISTRY

Synthesis of 1-indolyl substituted β-carboline natural products and discovery of antimalarial and cytotoxic activities

(2014) Lydia P.P. Liew et al.   TETRAHEDRON

Silica-supported ceric ammonium nitrate catalyzed chemoselective formylation of indoles

(2014) Sukanya Tongkhan et al.   TETRAHEDRON LETTERS

Unexplored reactivity of 2-oxoaldehydes towards Pictet–Spengler conditions: concise approach to β-carboline based marine natural products

(2014) Narsaiah Battini et al.   RSC Advances

WCl6/DMF as a new reagent system for the phosphine-free Pd(0)-catalyzed aminocarbonylation of aryl halides

(2014) Nasser Iranpoor et al.   RSC Advances

The Cross-Dehydrogenative Coupling of C sp 3H Bonds: A Versatile Strategy for CC Bond Formations

(2013) Simon A. Girard et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A Cascade Coupling Strategy for One-Pot Total Synthesis of β-Carboline and Isoquinoline-Containing Natural Products and Derivatives

(2013) Yan-Ping Zhu et al.   CHEMISTRY-A EUROPEAN JOURNAL

Total Syntheses of Eudistomins Y1-Y7by an Efficient One-Pot Process of Tandem Benzylic Oxidation and Aromatization of 1-Benzyl-3,4-dihydro-β-Carbolines

(2013) Tien Ha Trieu et al.   EUROPEAN JOURNAL OF ORGANIC CHEMISTRY

Synthesis and Quantitative Structure–Activity Relationship (QSAR) Study of Novel N-Arylsulfonyl-3-acylindole Arylcarbonyl Hydrazone Derivatives as Nematicidal Agents

(2013) Zhiping Che et al.   JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY

CH Bond Functionalization: Emerging Synthetic Tools for Natural Products and Pharmaceuticals

(2012) Junichiro Yamaguchi et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

nBu4NI-catalyzed C3-formylation of indoles with N-methylaniline

(2012) Lan-Tao Li et al.   CHEMICAL COMMUNICATIONS

Cu(ii)-catalyzed C–H (SP3) oxidation and C–N cleavage: base-switched methylenation and formylation using tetramethylethylenediamine as a carbon source

(2012) Lei Zhang et al.   CHEMICAL COMMUNICATIONS

Synthesis and Evaluation of Indole-Based Chalcones as Inducers of Methuosis, a Novel Type of Nonapoptotic Cell Death

(2012) Michael W. Robinson et al.   JOURNAL OF MEDICINAL CHEMISTRY

Decarboxylative coupling reactions: a modern strategy for C–C-bond formation

(2011) Nuria Rodríguez et al.   CHEMICAL SOCIETY REVIEWS

Total synthesis and bioactivity of the marine alkaloid pityriacitrin and some of its derivatives

(2011) Puyong Zhang et al.   EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY

Antimalarial β-Carboline and Indolactam Alkaloids from Marinactinospora thermotolerans, a Deep Sea Isolate

(2011) Hongbo Huang et al.   JOURNAL OF NATURAL PRODUCTS

Mild and Selective Ru-Catalyzed Formylation and Fe-Catalyzed Acylation of Free (N–H) Indoles Using Anilines as the Carbonyl Source

(2011) Wenliang Wu et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

Minisci reactions: Versatile CH-functionalizations for medicinal chemists

(2011) Matthew A. J. Duncton   MedChemComm

Direct C−H Arylation of Electron-Deficient Heterocycles with Arylboronic Acids

(2010) Ian B. Seiple et al.   JOURNAL OF THE AMERICAN CHEMICAL SOCIETY

β-Carboline Alkaloids from a Korean TunicateEudistomasp.

(2008) Weihong Wang et al.   JOURNAL OF NATURAL PRODUCTS