Bivalent BET Bromodomain Inhibitors Confer Increased Potency and Selectivity for BRDT via Protein Conformational Plasticity
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Title
Bivalent BET Bromodomain Inhibitors Confer Increased Potency and Selectivity for BRDT via Protein Conformational Plasticity
Authors
Keywords
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Journal
JOURNAL OF MEDICINAL CHEMISTRY
Volume 65, Issue 15, Pages 10441-10458
Publisher
American Chemical Society (ACS)
Online
2022-07-23
DOI
10.1021/acs.jmedchem.2c00453
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