Sweetening Pharmaceutical Radiochemistry by 18F-Fluoroglycosylation: Recent Progress and Future Prospects
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Title
Sweetening Pharmaceutical Radiochemistry by 18F-Fluoroglycosylation: Recent Progress and Future Prospects
Authors
Keywords
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Journal
Pharmaceuticals
Volume 14, Issue 11, Pages 1175
Publisher
MDPI AG
Online
2021-11-17
DOI
10.3390/ph14111175
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Note: Only part of the references are listed.- Advances in Reactive Oxygen Species (ROS) Imaging
- (2021) Niren Murthy et al. JOURNAL OF NUCLEAR MEDICINE
- Synthesis, Radiosynthesis, and in vitro Studies on Novel Hypoxia PET Tracers Incorporating [ 18 F]FDR
- (2021) Manuele Musolino et al. EUROPEAN JOURNAL OF ORGANIC CHEMISTRY
- Development of 18F-Fluoroglycosylated PSMA-Ligands with Improved Renal Clearance Behavior
- (2020) Roman Potemkin et al. MOLECULAR PHARMACEUTICS
- Targeting Fibroblast Activation Protein: Radiosynthesis and Preclinical Evaluation of an 18F-labeled FAP Inhibitor
- (2020) Johannes Toms et al. JOURNAL OF NUCLEAR MEDICINE
- Characterisation of the Expression of Neurotensin and Its Receptors in Human Colorectal Cancer and Its Clinical Implications
- (2020) Shengyang Qiu et al. Biomolecules
- Identification of Boronic Acid Derivatives as an Active Form of N-Alkylaminoferrocene-Based Anticancer Prodrugs and Their Radiolabeling with 18F
- (2019) Steffen Daum et al. BIOCONJUGATE CHEMISTRY
- FAPI-PET/CT: Mean intensity of tracer-uptake (SUV) in 28 different kinds of cancer
- (2019) Clemens Kratochwil et al. JOURNAL OF NUCLEAR MEDICINE
- Synthesis and Bioevaluation of Novel [18F]FDG-Conjugated 2-Nitroimidazole Derivatives for Tumor Hypoxia Imaging
- (2019) Xianteng Yang et al. MOLECULAR PHARMACEUTICS
- 18F-labelled triazolyl-linked argininamides targeting the neuropeptide Y Y1R for PET imaging of mammary carcinoma
- (2019) Simone Maschauer et al. Scientific Reports
- One-step conjugation of glycylglycine with [18F]FDG and a pilot PET imaging study
- (2018) A. M. Şenışık et al. JOURNAL OF RADIOANALYTICAL AND NUCLEAR CHEMISTRY
- Synthesis and Characterization of Novel Fluoro-glycosylated Porphyrins that can be Utilized as Theranostic Agents
- (2018) Katriann Arja et al. ChemistryOpen
- FAPI-PET/CT: biodistribution and preliminary dosimetry estimate of two DOTA-containing FAP-targeting agents in patients with various cancers
- (2018) Frederik Giesel et al. JOURNAL OF NUCLEAR MEDICINE
- Synthesis and evaluation of an N-[18F]fluorodeoxyglycosyl amino acid for PET imaging of tumor metabolism
- (2018) Zhifang Wu et al. NUCLEAR MEDICINE AND BIOLOGY
- Radiosynthesis of an 18 F-fluoroglycosylated aminoferrocene for in-vivo imaging of reactive oxygen species activity by PET
- (2018) Johannes Toms et al. JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS
- Efficient cartridge purification for producing high molar activity [18F]fluoro-glycoconjugates via oxime formation
- (2018) Outi Keinänen et al. NUCLEAR MEDICINE AND BIOLOGY
- Targeting Prostate-Specific Membrane Antigen (PSMA) with F-18-Labeled Compounds: the Influence of Prosthetic Groups on Tumor Uptake and Clearance Profile
- (2017) Vincent Bouvet et al. MOLECULAR IMAGING AND BIOLOGY
- β-Configured clickable [18F]FDGs as novel 18F-fluoroglycosylation tools for PET
- (2017) M. Elgland et al. NEW JOURNAL OF CHEMISTRY
- Consensus nomenclature rules for radiopharmaceutical chemistry — Setting the record straight
- (2017) Heinz H. Coenen et al. NUCLEAR MEDICINE AND BIOLOGY
- Radiosynthesis and Preclinical Evaluation of 18F-Fluoroglycosylated Octreotate for Somatostatin Receptor Imaging
- (2016) Simone Maschauer et al. BIOCONJUGATE CHEMISTRY
- 18F- and 68Ga-Labeled Neurotensin Peptides for PET Imaging of Neurotensin Receptor 1
- (2016) Simone Maschauer et al. JOURNAL OF MEDICINAL CHEMISTRY
- Caged [18F]FDG Glycosylamines for Imaging Acidic Tumor Microenvironments Using Positron Emission Tomography
- (2015) Robert R. Flavell et al. BIOCONJUGATE CHEMISTRY
- Rerouting the Metabolic Pathway of 18F-Labeled Peptides: The Influence of Prosthetic Groups
- (2015) Susan Richter et al. BIOCONJUGATE CHEMISTRY
- Improved radiosynthesis and preliminary in vivo evaluation of a 18F-labeled glycopeptide–peptoid hybrid for PET imaging of neurotensin receptor 2
- (2015) Simone Maschauer et al. BIOORGANIC & MEDICINAL CHEMISTRY
- Development of 6-[18F]fluoro-carbohydrate-based prosthetic groups and their conjugation to peptides via click chemistry
- (2015) Charlotte Collet et al. JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS
- Applications of Fluorine in Medicinal Chemistry
- (2015) Eric P. Gillis et al. JOURNAL OF MEDICINAL CHEMISTRY
- Synthesis and in Vitro and in Vivo Evaluation of an 18F-Labeled Neuropeptide Y Analogue for Imaging of Breast Cancer by PET
- (2015) Sven Hofmann et al. MOLECULAR PHARMACEUTICS
- Nucleophilic fluorination using imidazolium based ionic liquid bearing tert-alcohol moiety
- (2015) Sandip S. Shinde et al. NEW JOURNAL OF CHEMISTRY
- Novel synthesis and initial preclinical evaluation of 18 F-[FDG] labeled rhodamine: a potential PET myocardial perfusion imaging agent
- (2015) Ibrahim AlJammaz et al. NUCLEAR MEDICINE AND BIOLOGY
- A New Highly Reactive and Low Lipophilicity Fluorine-18 Labeled Tetrazine Derivative for Pretargeted PET Imaging
- (2015) Outi Keinänen et al. ACS Medicinal Chemistry Letters
- Neurotensin receptors in pancreatic ductal carcinomas
- (2015) Meike Körner et al. EJNMMI Research
- Use of 18F-2-Fluorodeoxyglucose to Label Antibody Fragments for Immuno-Positron Emission Tomography of Pancreatic Cancer
- (2015) Mohammad Rashidian et al. ACS Central Science
- One molecule of ionic liquid and tert-alcohol on a polystyrene-support as catalysts for efficient nucleophilic substitution including fluorination
- (2014) Sandip S. Shinde et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- Sweetening Pharmaceutical Radiochemistry by18F-Fluoroglycosylation: A Short Review
- (2014) Simone Maschauer et al. Biomed Research International
- Click chemistry based synthesis of dopamine D4 selective receptor ligands for the selection of potential PET tracers
- (2013) Ashutosh Banerjee et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- Translating the concept of peptidelabeling with 5-deoxy-5-[18F]fluororibose into preclinical practice: 18F-labeling of Siglec-9 peptide for PET imaging of inflammation
- (2013) Xiang-Guo Li et al. CHEMICAL COMMUNICATIONS
- Oxime Ligation: A Chemoselective Click-Type Reaction for Accessing Multifunctional Biomolecular Constructs
- (2013) Sébastien Ulrich et al. CHEMISTRY-A EUROPEAN JOURNAL
- Application of Click Chemistry for PET
- (2013) Leila Mirfeizi et al. CURRENT ORGANIC CHEMISTRY
- Pyrazole-type cannabinoid ligands conjugated with fluoro-deoxy-carbohydrates as potential PET-imaging agents: Synthesis and CB1/CB2 receptor affinity evaluation
- (2013) Simona Frau et al. JOURNAL OF FLUORINE CHEMISTRY
- Synthesis of a new fluorine-18 glycosylated ‘click’ cyanoquinoline for the imaging of epidermal growth factor receptor
- (2013) Federica Pisaneschi et al. JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS
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- (2013) Christopher Lang et al. JOURNAL OF MEDICINAL CHEMISTRY
- Improved PET Imaging of Tumors in Mice Using a Novel 18 F-Folate Conjugate with an Albumin-Binding Entity
- (2013) Cindy R. Fischer et al. MOLECULAR IMAGING AND BIOLOGY
- Comparison of Three Dimeric 18F-AlF-NOTA-RGD Tracers
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- 18F-Glyco-RGD Peptides for PET Imaging of Integrin Expression: Efficient Radiosynthesis by Click Chemistry and Modulation of Biodistribution by Glycosylation
- (2013) Simone Maschauer et al. MOLECULAR PHARMACEUTICS
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- Efficient bioconjugation of 5-fluoro-5-deoxy-ribose (FDR) to RGD peptides for positron emission tomography (PET) imaging of αvβ3 integrin receptor
- (2013) Sergio Dall'Angelo et al. ORGANIC & BIOMOLECULAR CHEMISTRY
- [18F]Fluoro-Deoxy-Glucose Folate: A Novel PET Radiotracer with Improved in Vivo Properties for Folate Receptor Targeting
- (2012) Cindy R. Fischer et al. BIOCONJUGATE CHEMISTRY
- [18F]-5-Fluoro-5-deoxyribose, an efficient peptide bioconjugation ligand for positron emission tomography (PET) imaging
- (2012) Xiang-Guo Li et al. CHEMICAL COMMUNICATIONS
- Development of a Metabolically Stable Neurotensin Receptor 2 (NTS2) Ligand
- (2012) Cornelia Held et al. ChemMedChem
- Oxime formation for fluorine-18 labeling of peptides and proteins for positron emission tomography (PET) imaging: A review
- (2012) Xiang-Guo Li et al. JOURNAL OF FLUORINE CHEMISTRY
- A New Class of Highly Potent Matrix Metalloproteinase Inhibitors Based on Triazole-Substituted Hydroxamates: (Radio)Synthesis and in Vitro and First in Vivo Evaluation
- (2012) Verena Hugenberg et al. JOURNAL OF MEDICINAL CHEMISTRY
- 18FDG conjugated magnetic nanoparticle probes: synthesis and in vitro investigations on MCF-7 breast cancer cells
- (2012) Feriha Ozkaya et al. JOURNAL OF RADIOANALYTICAL AND NUCLEAR CHEMISTRY
- Novel synthesis and preclinical evaluation of folic acid derivatives labeled with 18F-[FDG] for PET imaging of folate receptor-positive tumors
- (2012) I. Al Jammaz et al. NUCLEAR MEDICINE AND BIOLOGY
- Novel Strategies for Fluorine-18 Radiochemistry
- (2011) Ryan Littich et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- Direct radiolabelling of proteins at cysteine using [18F]-fluorosugars
- (2011) Omar Boutureira et al. CHEMICAL COMMUNICATIONS
- Gold nanoparticle probes: Design and in vitro applications in cancer cell culture
- (2011) Gulcan Unak et al. COLLOIDS AND SURFACES B-BIOINTERFACES
- Altered Expression of Neurotensin Receptors Is Associated with the Differentiation State of Prostate Cancer
- (2010) S. L. Swift et al. CANCER RESEARCH
- Fluoroglycoproteins: ready chemical site-selective incorporation of fluorosugars into proteins
- (2010) Omar Boutureira et al. CHEMICAL COMMUNICATIONS
- Labeling and Glycosylation of Peptides Using Click Chemistry: A General Approach to 18F-Glycopeptides as Effective Imaging Probes for Positron Emission Tomography
- (2009) Simone Maschauer et al. ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
- A Novel Method for Direct Site-Specific Radiolabeling of Peptides Using [18F]FDG
- (2009) Mohammad Namavari et al. BIOCONJUGATE CHEMISTRY
- Direct labelling of peptides with 2-[18F]fluoro-2-deoxy-d-glucose ([18F]FDG)
- (2009) Frank Wuest et al. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
- A series of 2-O-trifluoromethylsulfonyl-d-mannopyranosides as precursors for concomitant 18F-labeling and glycosylation by click chemistry
- (2009) Simone Maschauer et al. CARBOHYDRATE RESEARCH
- 18F-Fluoroglucosylation of peptides, exemplified on cyclo(RGDfK)
- (2009) Christina Hultsch et al. EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING
- 18F-Labeled Galacto and PEGylated RGD Dimers for PET Imaging of αvβ3 Integrin Expression
- (2009) Shuanglong Liu et al. MOLECULAR IMAGING AND BIOLOGY
- Synthesis and Application of [18F]FDG-Maleimidehexyloxime ([18F]FDG-MHO): A [18F]FDG-Based Prosthetic Group for the Chemoselective18F-Labeling of Peptides and Proteins†
- (2008) Frank Wuest et al. BIOCONJUGATE CHEMISTRY
- Molecular Imaging with PET
- (2008) Simon M. Ametamey et al. CHEMICAL REVIEWS
- Fluorine in medicinal chemistry
- (2007) Sophie Purser et al. CHEMICAL SOCIETY REVIEWS
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