Sweetening Pharmaceutical Radiochemistry by18F-Fluoroglycosylation: A Short Review

Click chemistry based synthesis of dopamine D4 selective receptor ligands for the selection of potential PET tracers

(2013) Ashutosh Banerjee et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

Translating the concept of peptidelabeling with 5-deoxy-5-[18F]fluororibose into preclinical practice: 18F-labeling of Siglec-9 peptide for PET imaging of inflammation

(2013) Xiang-Guo Li et al.   CHEMICAL COMMUNICATIONS

Application of Click Chemistry for PET

(2013) Leila Mirfeizi et al.   CURRENT ORGANIC CHEMISTRY

Pyrazole-type cannabinoid ligands conjugated with fluoro-deoxy-carbohydrates as potential PET-imaging agents: Synthesis and CB1/CB2 receptor affinity evaluation

(2013) Simona Frau et al.   JOURNAL OF FLUORINE CHEMISTRY

Synthesis of a new fluorine-18 glycosylated ‘click’ cyanoquinoline for the imaging of epidermal growth factor receptor

(2013) Federica Pisaneschi et al.   JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS

Synthesis and Evaluation of a 18F-Labeled Diarylpyrazole Glycoconjugate for the Imaging of NTS1-Positive Tumors

(2013) Christopher Lang et al.   JOURNAL OF MEDICINAL CHEMISTRY

Improved PET Imaging of Tumors in Mice Using a Novel 18 F-Folate Conjugate with an Albumin-Binding Entity

(2013) Cindy R. Fischer et al.   MOLECULAR IMAGING AND BIOLOGY

Comparison of Three Dimeric 18F-AlF-NOTA-RGD Tracers

(2013) Jinxia Guo et al.   MOLECULAR IMAGING AND BIOLOGY

18F-Glyco-RGD Peptides for PET Imaging of Integrin Expression: Efficient Radiosynthesis by Click Chemistry and Modulation of Biodistribution by Glycosylation

(2013) Simone Maschauer et al.   MOLECULAR PHARMACEUTICS

Recent Trends in Bioorthogonal Click-Radiolabeling Reactions Using Fluorine-18

(2013) Marc Pretze et al.   MOLECULES

Single step 18F-labeling of dimeric cycloRGD for functional PET imaging of tumors in mice

(2013) Ying Li et al.   NUCLEAR MEDICINE AND BIOLOGY

Efficient bioconjugation of 5-fluoro-5-deoxy-ribose (FDR) to RGD peptides for positron emission tomography (PET) imaging of αvβ3 integrin receptor

(2013) Sergio Dall'Angelo et al.   ORGANIC & BIOMOLECULAR CHEMISTRY

[18F]Fluoro-Deoxy-Glucose Folate: A Novel PET Radiotracer with Improved in Vivo Properties for Folate Receptor Targeting

(2012) Cindy R. Fischer et al.   BIOCONJUGATE CHEMISTRY

[18F]-5-Fluoro-5-deoxyribose, an efficient peptide bioconjugation ligand for positron emission tomography (PET) imaging

(2012) Xiang-Guo Li et al.   CHEMICAL COMMUNICATIONS

Development of a Metabolically Stable Neurotensin Receptor 2 (NTS2) Ligand

(2012) Cornelia Held et al.   ChemMedChem

A New Class of Highly Potent Matrix Metalloproteinase Inhibitors Based on Triazole-Substituted Hydroxamates: (Radio)Synthesis and in Vitro and First in Vivo Evaluation

(2012) Verena Hugenberg et al.   JOURNAL OF MEDICINAL CHEMISTRY

18FDG conjugated magnetic nanoparticle probes: synthesis and in vitro investigations on MCF-7 breast cancer cells

(2012) Feriha Ozkaya et al.   JOURNAL OF RADIOANALYTICAL AND NUCLEAR CHEMISTRY

Novel synthesis and preclinical evaluation of folic acid derivatives labeled with 18F-[FDG] for PET imaging of folate receptor-positive tumors

(2012) I. Al Jammaz et al.   NUCLEAR MEDICINE AND BIOLOGY

Direct radiolabelling of proteins at cysteine using [18F]-fluorosugars

(2011) Omar Boutureira et al.   CHEMICAL COMMUNICATIONS

Gold nanoparticle probes: Design and in vitro applications in cancer cell culture

(2011) Gulcan Unak et al.   COLLOIDS AND SURFACES B-BIOINTERFACES

Fluoroglycoproteins: ready chemical site-selective incorporation of fluorosugars into proteins

(2010) Omar Boutureira et al.   CHEMICAL COMMUNICATIONS

Click-Chemistry Reactions in Radiopharmaceutical Chemistry: Fast & Easy Introduction of Radiolabels into Biomolecules for In Vivo Imaging

(2010) C. Wangler et al.   CURRENT MEDICINAL CHEMISTRY

Imaging of enzyme replacement therapy using PET

(2010) C. P. Phenix et al.   PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA

Labeling and Glycosylation of Peptides Using Click Chemistry: A General Approach to 18F-Glycopeptides as Effective Imaging Probes for Positron Emission Tomography

(2009) Simone Maschauer et al.   ANGEWANDTE CHEMIE-INTERNATIONAL EDITION

A Novel Method for Direct Site-Specific Radiolabeling of Peptides Using [18F]FDG

(2009) Mohammad Namavari et al.   BIOCONJUGATE CHEMISTRY

Direct labelling of peptides with 2-[18F]fluoro-2-deoxy-d-glucose ([18F]FDG)

(2009) Frank Wuest et al.   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS

A series of 2-O-trifluoromethylsulfonyl-d-mannopyranosides as precursors for concomitant 18F-labeling and glycosylation by click chemistry

(2009) Simone Maschauer et al.   CARBOHYDRATE RESEARCH

18F-Fluoroglucosylation of peptides, exemplified on cyclo(RGDfK)

(2009) Christina Hultsch et al.   EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING

18F-Labeled Galacto and PEGylated RGD Dimers for PET Imaging of αvβ3 Integrin Expression

(2009) Shuanglong Liu et al.   MOLECULAR IMAGING AND BIOLOGY

Synthesis and Application of [18F]FDG-Maleimidehexyloxime ([18F]FDG-MHO): A [18F]FDG-Based Prosthetic Group for the Chemoselective18F-Labeling of Peptides and Proteins†

(2008) Frank Wuest et al.   BIOCONJUGATE CHEMISTRY

Molecular Imaging with PET

(2008) Simon M. Ametamey et al.   CHEMICAL REVIEWS